Synthesis and receptor-binding affinity of dipeptoid cholecystokinin ligands

European Journal of Medicinal Chemistry

Volumn 31, Issue 3, 1996, Pages 215-220

  Araldi, G ^a   Donati, D ^a   Oliosi, B ^a   Pasquarello, A ^a   Polinelli, S ^a   Tarzia, G ^b   Ursini, A ^a   Van Amsterdam, F T M ^a  

^a GSK   (Italy)

^b UNIVERSITY OF URBINO   (Italy)

Author keywords

CCK B antagonist; PD134308 derivative; Peptoid

Indexed keywords

4 [[2 [2 [[(2 ADAMANTYLOXY)CARBONYL]AMINO] 3 (1H INDOL 3 YL) 2 METHYLPROPIONAMIDO] 1 PHENYLETHYL]AMINO] 4 OXOBUTYRIC ACID MEGLUMINE; 4 [[2 [[3 (2 BENZO[B]THIENYL) 2 METHYL 1 OXO 2 ADAMANTYLOXYCARBONYLAMINO]PROPYL] 1 PHENYLETHYL]AMINO 4 OXOBUTYRIC ACID; 4[[2 [[3 (2 NAPHTHYL) 2 METHYL 1 OXO 2 ADAMANTYLOXYCARBONYLAMINO]PROPYL]AMINO] 1 PHENYLETHYL]AMINO 4 OXOBUTYRIC ACID; ANXIOLYTIC AGENT; ARYLBUTYRIC ACID DERIVATIVE; CHOLECYSTOKININ A RECEPTOR; CHOLECYSTOKININ B RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CELL MEMBRANE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; NONHUMAN; PANCREAS; STRUCTURE ACTIVITY RELATION;

EID: 0029865873     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/0223-5234(96)89137-9     Document Type: Article

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