Synthesis and biological investigations of [18F]MR18445, a 5-HT3 receptor partial agonist

Bioorganic and Medicinal Chemistry

Volumn 6, Issue 6, 1998, Pages 789-795

  Katounina, Tatiana ^a   Besret, Laurent ^a   Dhilly, Martine ^a   Petit Taboué, Marie Christine ^a   Barbelivien, Alexandra ^b   Baron, Jean Claude ^a   Dauphin, François ^b   Barré, Louisa ^a  

^a GIP CYCERON   (France)

^b UNIVERSITÉ DE CAEN   (France)

Author keywords

5 HT3 Receptor; Baboon; Fluorine 18; PET; Rat

Indexed keywords

FLUORINE 18; PARTIAL AGONIST; RADIOLIGAND; SEROTONIN 3 AGONIST;

ANIMAL EXPERIMENT; ARTICLE; BABOON; CONTROLLED STUDY; DRUG BRAIN LEVEL; DRUG DISTRIBUTION; DRUG METABOLISM; DRUG SYNTHESIS; INTRAVENOUS DRUG ADMINISTRATION; NONHUMAN; RAT;

ANIMALS; AUTORADIOGRAPHY; BRAIN; FLUORINE RADIOISOTOPES; MALE; PAPIO; QUINOXALINES; RADIOPHARMACEUTICALS; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT3; SEROTONIN AGONISTS; TISSUE DISTRIBUTION; TOMOGRAPHY, EMISSION-COMPUTED;

PAPIO; PAPIO HAMADRYAS;

EID: 0031862061     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(98)00035-2     Document Type: Article

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