Search for selective antagonists at α1-adrenoreceptors: Neutral or negative antagonism?

Farmaco

Volumn 53, Issue 4, 1998, Pages 278-286

  Melchiorre, Carlo ^a   Bolognesi, Maria L ^a   Budriesi, Roberta ^a   Chiarini, Alberto ^a   Giardinà, Dario ^b   Minarini, Anna ^a   Quaglia, Wilma ^b   Leonardi, Amedeo ^c  

^a UNIVERSITY OF BOLOGNA   (Italy)

^b UNIVERSITY OF CAMERINO   (Italy)

^c Recordati SpA   (Italy)

Author keywords

1 Adrenoreceptors; Inverse agonism; Neutral antagonism; Receptor classification

Indexed keywords

2 [[2 (2,6 DIMETHOXYPHENOXY)ETHYL]AMINOMETHYL] 1,4 BENZODIOXAN; ADRENERGIC RECEPTOR; ALPHA 1 ADRENERGIC RECEPTOR BLOCKING AGENT; PRAZOSIN; RECEPTOR SUBTYPE;

BINDING SITE; CONFERENCE PAPER; CONTROLLED STUDY; DRUG ANTAGONISM; DRUG CLASSIFICATION; DRUG EFFICACY; ENANTIOMER; NONHUMAN; PROPRIOCEPTION; STEREOCHEMISTRY;

ADRENERGIC ALPHA-ANTAGONISTS; ANIMALS; DIOXANES; HUMANS; PRAZOSIN; RECEPTORS, ADRENERGIC, ALPHA-1; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0031845395     PISSN: 0014827X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-827X(98)00022-6     Document Type: Conference Paper

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