Characterisation and localisation of [3H]2-(2-benzofuranyl)-2-imidazoline binding in rat brain: A selective ligand for imidazoline I2 receptors

European Journal of Pharmacology

Volumn 353, Issue 1, 1998, Pages 123-135

  Lione, Lisa A ^a   Nutt, David J ^a   Hudson, Alan L ^a  

^a UNIVERSITY OF BRISTOL   (United Kingdom)

Author keywords

3H 2 BFI; Arcuate nucleus; Autoradiography; Brain, rat; Idazoxan; Imidazoline I2 receptor

Indexed keywords

2 (1,4 BENZODIOXAN 2 YLAMINO) 2 IMIDAZOLINE; 2 (2 BENZOFURANYL) 2 IMIDAZOLINE; 2 (2 IMIDAZOLIN 2 YL)QUINOLINE; 2 (2 IMIDAZOLIN 2 YL)QUINOXALINE; 4 CHLORO 2 (2 IMIDAZOLIN 2 YLAMINO)ISOINDOLINE; ADRENERGIC RECEPTOR BLOCKING AGENT; ADRENERGIC RECEPTOR STIMULATING AGENT; AGMATINE; BRIMONIDINE; EFAROXAN; GUANABENZ; HISTAMINE RECEPTOR; IDAZOXAN; IMIDAZOLINE I1 RECEPTOR; IMIDAZOLINE I2 RECEPTOR; MEDETOMIDINE; MOXONIDINE; NAPHAZOLINE; RAUWOLSCINE; UNCLASSIFIED DRUG; 2-(2-BENZOFURANYL)-2-IMIDAZOLINE; BENZOFURAN DERIVATIVE; DRUG RECEPTOR; IMIDAZOLE DERIVATIVE; IMIDAZOLINE RECEPTORS; LIGAND; TRITIUM;

ANIMAL TISSUE; ARCUATE NUCLEUS; ARTICLE; AUTORADIOGRAPHY; BRAIN HOMOGENATE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY; RECEPTOR DENSITY; ANIMAL; BINDING COMPETITION; BRAIN; COMPARATIVE STUDY; HISTOLOGY; KINETICS; MEMBRANE; METABOLISM; WISTAR RAT;

ANIMALS; AUTORADIOGRAPHY; BENZOFURANS; BINDING, COMPETITIVE; BRAIN; IDAZOXAN; IMIDAZOLES; KINETICS; LIGANDS; MALE; MEMBRANES; RATS; RATS, WISTAR; RECEPTORS, DRUG; TRITIUM;

EID: 0031595107     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(98)00389-6     Document Type: Article

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