A practical and scalable synthesis of SR 142801, a tachykinin NK3 antagonist

Bioorganic and Medicinal Chemistry Letters

Volumn 7, Issue 5, 1997, Pages 555-560

  Chen, Huai G ^a   Chung, F Z ^a   Goel, O P ^a   Johnson, D ^a   Kesten, S ^a   Knobelsdorf, J ^a   Lee, H T ^a   Rubin, J R ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

NEUROKININ 3 RECEPTOR; OSANETANT;

ANIMAL CELL; ARTICLE; CHIRALITY; CHO CELL; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; GAS LIQUID CHROMATOGRAPHY; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; IN VITRO STUDY; NONHUMAN; REACTION ANALYSIS; STEREOCHEMISTRY; X RAY CRYSTALLOGRAPHY;

ANIMALIA;

EID: 0031552139     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(97)00064-4     Document Type: Article

References (13)

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10. R = 14.58 min.
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