A reliable and efficient synthesis of SR 142801

Bioorganic and Medicinal Chemistry Letters

Volumn 6, Issue 19, 1996, Pages 2307-2310

  Giardina, Giuseppe A M ^a   Grugni, Mario ^a   Rigolio, Roberto ^a   Vassallo, Marco ^a   Erhard, Karl ^b   Farina, Carlo ^a  

^a SmithKline Beecham SpA   (Italy)

^b GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

NEUROKININ 3 RECEPTOR ANTAGONIST; SZ 142801; UNCLASSIFIED DRUG;

ARTICLE; DRUG SYNTHESIS;

EID: 0030575607     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/0960-894X(96)00419-2     Document Type: Article

References (20)

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20. 10 three steps appear to exceed 100% yield.