The protein kinase c inhibitors Ro 318220 and GF 109203X are equally potent inhibitors of MAPKAP kinase-1β (Rsk-2) and p70 S6 kinase

FEBS Letters

Volumn 402, Issue 2-3, 1997, Pages 121-123

  Alessi, Dario R ^a  

^a UNIVERSITY OF DUNDEE   (United Kingdom)

Author keywords

p70 S6 kinase; PKC; Protein kinase inhibitor; Rsk

Indexed keywords

2 [1 (3 AMIDINOTHIOPROPYL) 1H INDOL 3 YL] 3 (1 METHYL 1H INDOL 3 YL)MALEIMIDE; 2 [1 (3 DIMETHYLAMINOPROPYL) 3 INDOLYL] 3 (3 INDOLYL)MALEIMIDE; ISOENZYME; MITOGEN ACTIVATED PROTEIN KINASE; PROTEIN KINASE C INHIBITOR;

ARTICLE; DRUG POTENCY; ENZYME INHIBITION; PRIORITY JOURNAL;

AMINO ACID SEQUENCE; ANIMALS; CELL LINE; ENZYME INHIBITORS; INDOLES; ISOENZYMES; KINETICS; LIVER; MALEIMIDES; MOLECULAR SEQUENCE DATA; PEPTIDES; PROTEIN KINASE C; PROTEIN-SERINE-THREONINE KINASES; RATS; RECOMBINANT PROTEINS; RIBOSOMAL PROTEIN S6 KINASES; RIBOSOMAL PROTEIN S6 KINASES, 90-KDA; SPODOPTERA; TRANSFECTION;

EID: 0031052014     PISSN: 00145793     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-5793(96)01510-4     Document Type: Article

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