Inhibition of cyclin-dependent kinases by purine analogues. Crystal structure of human cdk2 complexed with roscovitine

European Journal of Biochemistry

Volumn 243, Issue 1-2, 1997, Pages 518-526

  De Azevedo, Walter Filgueira ^a   Leclerc, Sophie ^b   Meijer, Laurent ^b   Havlicek, Libor ^c   Strnad, Miroslav ^d   Kim, Sung Hou ^a  

^a LAWRENCE BERKELEY NATIONAL LABORATORY   (United States)

^b STATION BIOLOGIQUE   (France)

^c CHARLES UNIVERSITY   (Czech Republic)

^d INSTITUTE OF EXPERIMENTAL BOTANY   (Czech Republic)

Author keywords

Anti tumor agent; Cell cycle; Cyclin dependent kinase; Protein kinase inhibitor; Purine

Indexed keywords

CYCLIN DEPENDENT KINASE; ENZYME INHIBITOR; OLOMOUCINE; PURINE DERIVATIVE; ROSCOVITINE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; ASTERIAS; COMPETITIVE INHIBITION; COMPLEX FORMATION; CONTROLLED STUDY; CRYSTAL STRUCTURE; CRYSTALLOGRAPHY; ENZYME BINDING; NONHUMAN; PRIORITY JOURNAL; STRUCTURE ANALYSIS;

EID: 0031028163     PISSN: 00142956     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1432-1033.1997.0518a.x     Document Type: Article

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