Investigation on the coupling reactions of aryltriflates with aromatic amines: Selection of the metal catalyst

Bioorganic and Medicinal Chemistry Letters

Volumn 7, Issue 14, 1997, Pages 1821-1824

  Torisawa, Yasuhiro ^a   Hashimoto, Akihiro ^a   Furuta, Takuya ^a   Minamikawa, Jun Ichi ^a  

^a OTSUKA PHARMACEUTICAL CO LTD   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

ANILINE DERIVATIVE; AROMATIC AMINE;

ARTICLE; CATALYST; DRUG SYNTHESIS; IN VITRO STUDY; METHODOLOGY; REACTION ANALYSIS;

EID: 0030799609     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(97)00315-6     Document Type: Article

References (17)

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3. Larock, R. C. in Comprehensive Organic Transformations, VCH Publisher 1989, pp. 397-398;
4. Mitsunobu, O. in Comprehensive Organic Synthesis, Trost, B. M., Fleming, I., Eds.; Pergamon Press, 1991, vol 6, pp. 65-101.
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17. All the experiments shown here were carried out under conventional conditions (no argon exchange) and no special precautions have been taken for the selection of the solvent and reagents.