[125/123I]IPH: A radioiodinated analog of epibatidine for in vivo studies of nicotinic acetylcholine receptors

Synapse

Volumn 26, Issue 4, 1997, Pages 392-399

  Musachio, John L ^a,c   Villemagne, Victor L ^a   Scheffel, Ursula ^a   Stathis, Marigo ^a   Finley, Paige ^a   Horti, Andrew ^b   London, Edythe D ^b   Dannals, Robert F ^a  

^a DEPARTMENT OF PATHOLOGY   (United States)

^b NATIONAL INSTITUTE ON DRUG ABUSE   (United States)

^c JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

Epibatidine; Iodine 123; Iodine 125; Nicotinic acetylcholine receptor; SPECT

Indexed keywords

EPIBATIDINE; IODINE 123; IODINE 125; KETANSERIN; MECAMYLAMINE; NALOXONE; NICOTINIC RECEPTOR; 2 (2 IODO 5 PYRIDYL) 7 AZABICYCLO(2.2.1)HEPTANE; 2-(2-IODO-5-PYRIDYL)-7-AZABICYCLO(2.2.1)HEPTANE; DIAGNOSTIC AGENT; FUSED HETEROCYCLIC RINGS; LIGAND; NICOTINIC AGENT; PYRIDINE DERIVATIVE; RADIOACTIVE IODINE;

ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; BINDING SITE; CONTROLLED STUDY; DRUG PENETRATION; DRUG RECEPTOR BINDING; IN VIVO STUDY; MOUSE; NEUROTRANSMISSION; NONHUMAN; PRIORITY JOURNAL; RADIOIODINATION; RECEPTOR UPREGULATION; SINGLE PHOTON EMISSION COMPUTER TOMOGRAPHY; THALAMUS; ANIMAL; BRAIN; BRAIN LEVEL; DOSE RESPONSE; DRUG EFFECT; HISTOLOGY; MALE; PAPIO; TISSUE DISTRIBUTION;

ANIMALS; BICYCLO COMPOUNDS, HETEROCYCLIC; BRAIN; BRAIN CHEMISTRY; DOSE-RESPONSE RELATIONSHIP, DRUG; IODINE RADIOISOTOPES; LIGANDS; MALE; MICE; NICOTINIC AGONISTS; PAPIO; PYRIDINES; RECEPTORS, NICOTINIC; TISSUE DISTRIBUTION; TOMOGRAPHY, EMISSION-COMPUTED, SINGLE-PHOTON;

EID: 0030612592     PISSN: 08874476     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1098-2396(199708)26:4<392::AID-SYN7>3.0.CO;2-1     Document Type: Article

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