Combinatorial libraries on rigid scaffolds: Solid phase synthesis of variably substituted pyrazoles and isoxazoles

Molecules

Volumn 2, Issue 1, 1997, Pages 17-30

  Marzinzik, Andreas L ^a   Felder, Eduard R ^a,b  

^a F HOFFMANN LA ROCHE LTD   (Switzerland)

^b NOVARTIS PHARMA AG   (Switzerland)

Author keywords

Combinatorial chemistry; Lead finding; Split synthesis

Indexed keywords

ACETIC ACID DERIVATIVE; AMINE; CARBOXYLIC ACID DERIVATIVE; ESTER; HYDRAZINE DERIVATIVE; ISOXAZOLE DERIVATIVE; KETONE DERIVATIVE; PYRAZOLE DERIVATIVE;

ALKYLATION; ARTICLE; CHEMICAL REACTION; CLAISEN CONDENSATION; COMBINATORIAL LIBRARY; CYCLIZATION; MOLECULAR LIBRARY; MOLECULAR WEIGHT; SOLID; SUBSTITUTION REACTION; SYNTHESIS; VALIDATION PROCESS;

EID: 0002099615     PISSN: 14203049     EISSN: None     Source Type: Journal    
DOI: 10.3390/jan97p5     Document Type: Article

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