-
1
-
-
24844463791
-
-
Dissertation, Stuttgart
-
Taken in part from: [1a] M. Schön, Dissertation, Stuttgart 1997; [1b] R. Riess, Dissertation, Würzburg, 1993; [1c] S. Laschat, Diplomarbeit, Würzburg, 1987. Preliminary results reported in: [1d] M. Schön, S. Laschat, R. Riess, V. Jäger, 3-Hydroxyisoxazole-5-carbaldehydes - Versatile Key Intermediates in the Synthesis of New 3-Hydroxyisoxazoles, 5th Blue Danube Symposium on Heterocyclic Chemistry, Castá-Papiernicka, Slovak Republic, 14.-17.6.1995, PO-56, Proceedings p. 127 [1e] M. Schön, S. Laschat, R. Riess, V. Jäger, New Approach to 3-Hydroxyisoxazole-5-carbaldehydes -Key Intermediates in the Synthesis of New 3-Hydroxyisoxazoles of Pharmacological interest, Article 059, "1st Electronic Conference on Heterocyclic Chemistry", H. S. Rzepa, J. P. Snyder, C. Leach (Eds.); The Royal Society of Chemistry, 1997, ISBN 0-85404-894-4.
-
(1997)
-
-
Schön, M.1
-
2
-
-
2742555268
-
-
Dissertation, Würzburg
-
Taken in part from: [1a] M. Schön, Dissertation, Stuttgart 1997; [1b] R. Riess, Dissertation, Würzburg, 1993; [1c] S. Laschat, Diplomarbeit, Würzburg, 1987. Preliminary results reported in: [1d] M. Schön, S. Laschat, R. Riess, V. Jäger, 3-Hydroxyisoxazole-5-carbaldehydes - Versatile Key Intermediates in the Synthesis of New 3-Hydroxyisoxazoles, 5th Blue Danube Symposium on Heterocyclic Chemistry, Castá-Papiernicka, Slovak Republic, 14.-17.6.1995, PO-56, Proceedings p. 127 [1e] M. Schön, S. Laschat, R. Riess, V. Jäger, New Approach to 3-Hydroxyisoxazole-5-carbaldehydes -Key Intermediates in the Synthesis of New 3-Hydroxyisoxazoles of Pharmacological interest, Article 059, "1st Electronic Conference on Heterocyclic Chemistry", H. S. Rzepa, J. P. Snyder, C. Leach (Eds.); The Royal Society of Chemistry, 1997, ISBN 0-85404-894-4.
-
(1993)
-
-
Riess, R.1
-
3
-
-
2742586978
-
-
Diplomarbeit, Würzburg, 1987. Preliminary results reported in
-
Taken in part from: [1a] M. Schön, Dissertation, Stuttgart 1997; [1b] R. Riess, Dissertation, Würzburg, 1993; [1c] S. Laschat, Diplomarbeit, Würzburg, 1987. Preliminary results reported in: [1d] M. Schön, S. Laschat, R. Riess, V. Jäger, 3-Hydroxyisoxazole-5-carbaldehydes - Versatile Key Intermediates in the Synthesis of New 3-Hydroxyisoxazoles, 5th Blue Danube Symposium on Heterocyclic Chemistry, Castá-Papiernicka, Slovak Republic, 14.-17.6.1995, PO-56, Proceedings p. 127 [1e] M. Schön, S. Laschat, R. Riess, V. Jäger, New Approach to 3-Hydroxyisoxazole-5-carbaldehydes -Key Intermediates in the Synthesis of New 3-Hydroxyisoxazoles of Pharmacological interest, Article 059, "1st Electronic Conference on Heterocyclic Chemistry", H. S. Rzepa, J. P. Snyder, C. Leach (Eds.); The Royal Society of Chemistry, 1997, ISBN 0-85404-894-4.
-
-
-
Laschat, S.1
-
4
-
-
24844432152
-
-
5th Blue Danube Symposium on Heterocyclic Chemistry, Castá-Papiernicka, Slovak Republic, 14.-17.6. PO-56, Proceedings
-
Taken in part from: [1a] M. Schön, Dissertation, Stuttgart 1997; [1b] R. Riess, Dissertation, Würzburg, 1993; [1c] S. Laschat, Diplomarbeit, Würzburg, 1987. Preliminary results reported in: [1d] M. Schön, S. Laschat, R. Riess, V. Jäger, 3-Hydroxyisoxazole-5-carbaldehydes - Versatile Key Intermediates in the Synthesis of New 3-Hydroxyisoxazoles, 5th Blue Danube Symposium on Heterocyclic Chemistry, Castá-Papiernicka, Slovak Republic, 14.-17.6.1995, PO-56, Proceedings p. 127 [1e] M. Schön, S. Laschat, R. Riess, V. Jäger, New Approach to 3-Hydroxyisoxazole-5-carbaldehydes -Key Intermediates in the Synthesis of New 3-Hydroxyisoxazoles of Pharmacological interest, Article 059, "1st Electronic Conference on Heterocyclic Chemistry", H. S. Rzepa, J. P. Snyder, C. Leach (Eds.); The Royal Society of Chemistry, 1997, ISBN 0-85404-894-4.
-
(1995)
3-Hydroxyisoxazole-5-carbaldehydes - Versatile Key Intermediates in the Synthesis of New 3-Hydroxyisoxazoles
, pp. 127
-
-
Schön, M.1
Laschat, S.2
Riess, R.3
Jäger, V.4
-
5
-
-
24844439031
-
-
Article 059, "1st Electronic Conference on Heterocyclic Chemistry", H. S. Rzepa, J. P. Snyder, C. Leach (Eds.); The Royal Society of Chemistry, ISBN 0-85404-894-4
-
Taken in part from: [1a] M. Schön, Dissertation, Stuttgart 1997; [1b] R. Riess, Dissertation, Würzburg, 1993; [1c] S. Laschat, Diplomarbeit, Würzburg, 1987. Preliminary results reported in: [1d] M. Schön, S. Laschat, R. Riess, V. Jäger, 3-Hydroxyisoxazole-5-carbaldehydes - Versatile Key Intermediates in the Synthesis of New 3-Hydroxyisoxazoles, 5th Blue Danube Symposium on Heterocyclic Chemistry, Castá-Papiernicka, Slovak Republic, 14.-17.6.1995, PO-56, Proceedings p. 127 [1e] M. Schön, S. Laschat, R. Riess, V. Jäger, New Approach to 3-Hydroxyisoxazole-5-carbaldehydes -Key Intermediates in the Synthesis of New 3-Hydroxyisoxazoles of Pharmacological interest, Article 059, "1st Electronic Conference on Heterocyclic Chemistry", H. S. Rzepa, J. P. Snyder, C. Leach (Eds.); The Royal Society of Chemistry, 1997, ISBN 0-85404-894-4.
-
(1997)
New Approach to 3-Hydroxyisoxazole-5-carbaldehydes -Key Intermediates in the Synthesis of New 3-Hydroxyisoxazoles of Pharmacological Interest
-
-
Schön, M.1
Laschat, S.2
Riess, R.3
Jäger, V.4
-
6
-
-
0019407477
-
-
[2a] L. Brehm, P. Krogsgaard-Larsen, K. Schaumburg, Acta Chem. Scand., B 1981, 35, 311-324.
-
(1981)
Acta Chem. Scand., B
, vol.35
, pp. 311-324
-
-
Brehm, L.1
Krogsgaard-Larsen, P.2
Schaumburg, K.3
-
10
-
-
0000472403
-
Amino Acid Receptors
-
(Eds.: C. Hansch, P. G. Sammes, J. B. Taylor), Pergamon Press, Oxford
-
[3b] p Krogsgaard-Larsen, "Amino Acid Receptors", in Comprehensive Medicinal Chemistry, vol. 3 (Eds.: C. Hansch, P. G. Sammes, J. B. Taylor), Pergamon Press, Oxford, 1990, 493-537.
-
(1990)
Comprehensive Medicinal Chemistry
, vol.3
, pp. 493-537
-
-
Krogsgaard-Larsen, P.1
-
11
-
-
0028129538
-
-
[3c] Krogsgaard-Larsen, B. Frløund, F. S. Jørgensen, A. Schousboe, J. Med. Chem. 1994, 37, 2489-2505.
-
(1994)
J. Med. Chem.
, vol.37
, pp. 2489-2505
-
-
Krogsgaard-Larsen1
Frløund, B.2
Jørgensen, F.S.3
Schousboe, A.4
-
12
-
-
0028062168
-
-
T. N. Johansen, K. Frydenvang, B. Ebert, P. Krogsgaard-Larsen, U. Madsen, J. Med. Chem. 1994, 37, 3252-3262.
-
(1994)
J. Med. Chem.
, vol.37
, pp. 3252-3262
-
-
Johansen, T.N.1
Frydenvang, K.2
Ebert, B.3
Krogsgaard-Larsen, P.4
Madsen, U.5
-
13
-
-
24844440443
-
-
[5a] N. Skjœbœk, B. Ebert, E. Falch, L. Brehm, P. Krogsgaard-Larsen, J. Chem. Soc., Perkin Trans, 1 1995, 221-225.
-
(1995)
J. Chem. Soc., Perkin Trans, 1
, pp. 221-225
-
-
Skjœbœk, N.1
Ebert, B.2
Falch, E.3
Brehm, L.4
Krogsgaard-Larsen, P.5
-
15
-
-
0029863920
-
-
[6a] U. Madsen, B. Bang-Andersen, L. Brehm, I. T. Christensen, B. Ebert, I. T. S. Kristoffersen, Y. Lang, P. Krogsgaard-Larsen. J. Med. Chem. 1996, 39, 1682-1691.
-
(1996)
J. Med. Chem.
, vol.39
, pp. 1682-1691
-
-
Madsen, U.1
Bang-Andersen, B.2
Brehm, L.3
Christensen, I.T.4
Ebert, B.5
Kristoffersen, I.T.S.6
Lang, Y.7
Krogsgaard-Larsen, P.8
-
16
-
-
0029809205
-
-
[6b] R. Amici, P. Pevarello, M. Colombo, M. Varasi, Synthesis 1996, 1177-1179.
-
(1996)
Synthesis
, pp. 1177-1179
-
-
Amici, R.1
Pevarello, P.2
Colombo, M.3
Varasi, M.4
-
17
-
-
0030024147
-
-
[7a] U. Madsen, K. Frydenvang, B. Ebert, T. N. Johansen, L. Brehm, P. Krogsgaard-Larsen, J. Med. Chem. 1996, 39, 183-190.
-
(1996)
J. Med. Chem.
, vol.39
, pp. 183-190
-
-
Madsen, U.1
Frydenvang, K.2
Ebert, B.3
Johansen, T.N.4
Brehm, L.5
Krogsgaard-Larsen, P.6
-
18
-
-
0028202566
-
-
[7b] B. Ebert, S. Lenz, L. Brehm, P. Bregnedal, J. J. Hansen, K.; Frederiksen, K. P. Bøgesø, P. Krogsgaard-Larsen, J. Med. Chem. 1994, 37, 878-884.
-
(1994)
J. Med. Chem.
, vol.37
, pp. 878-884
-
-
Ebert, B.1
Lenz, S.2
Brehm, L.3
Bregnedal, P.4
Hansen, J.J.5
Frederiksen, K.6
Bøgesø, K.P.7
Krogsgaard-Larsen, P.8
-
19
-
-
0020549223
-
-
[7c] J. J Hansen, J. Lauridsen, E. Nielsen, P. Krogsgaard-Larsen, J. Med Chem. 1983, 26, 901-903.
-
(1983)
J. Med Chem.
, vol.26
, pp. 901-903
-
-
Hansen, J.J.1
Lauridsen, J.2
Nielsen, E.3
Krogsgaard-Larsen, P.4
-
20
-
-
0029150501
-
-
[8a] B. Frølund, U. Kristiansen, L. Brehm, A. B. Hansen, P. Krogsgaard-Larsen, E. Falch, J. Med. Chem. 1995, 38, 3287-3296.
-
(1995)
J. Med. Chem.
, vol.38
, pp. 3287-3296
-
-
Frølund, B.1
Kristiansen, U.2
Brehm, L.3
Hansen, A.B.4
Krogsgaard-Larsen, P.5
Falch, E.6
-
21
-
-
2742537709
-
-
[8b] H. Hjeds, I. T. Christensen. C. Cornett, B. Frølund, E. Falch, J. B. Pedersen, P. Krogsgaard-Larsen, Acta Chem. Scand. 1992, 46, 772-777.
-
(1992)
Acta Chem. Scand.
, vol.46
, pp. 772-777
-
-
Hjeds, H.1
Christensen, I.T.2
Cornett, C.3
Frølund, B.4
Falch, E.5
Pedersen, J.B.6
Krogsgaard-Larsen, P.7
-
23
-
-
37049086661
-
-
[9b] L. Brehm, J. S. Johansen, P. Krogsgaard-Larsen, J. Chem. Soc., Perkin Trans, 1 1992 , 2059-2063.
-
(1992)
J. Chem. Soc., Perkin Trans, 1
, pp. 2059-2063
-
-
Brehm, L.1
Johansen, J.S.2
Krogsgaard-Larsen, P.3
-
24
-
-
0025970909
-
-
[9c] P. Krogsgaard-Larsen, J. W. Ferkany, E. Ø. Nielsen, U. Madsen, B. Ebert, J. S. Johansen, N. H. Diemer, T. Bruhn, D. T. Beattie, D. R. Curtis, J. Med. Chem. 1991, 34, 123-130.
-
(1991)
J. Med. Chem.
, vol.34
, pp. 123-130
-
-
Krogsgaard-Larsen, P.1
Ferkany, J.W.2
Nielsen, E.Ø.3
Madsen, U.4
Ebert, B.5
Johansen, J.S.6
Diemer, N.H.7
Bruhn, T.8
Beattie, D.T.9
Curtis, D.R.10
-
26
-
-
0021910630
-
-
[10b] J.Lauridsen, T. Honoré, P. Krogsgaard-Larsen, J. Med. Chem. 1985, 28, 668-672.
-
(1985)
J. Med. Chem.
, vol.28
, pp. 668-672
-
-
Lauridsen, J.1
Honoré, T.2
Krogsgaard-Larsen, P.3
-
27
-
-
0021953106
-
-
[10c] P. Krogsgaard-Larsen, L. Brehm, J. S. Johansen, P. Vinzents, J. Lauridsen, D. R. Curtis, J. Med. Chem. 1985, 28, 673-679.
-
(1985)
J. Med. Chem.
, vol.28
, pp. 673-679
-
-
Krogsgaard-Larsen, P.1
Brehm, L.2
Johansen, J.S.3
Vinzents, P.4
Lauridsen, J.5
Curtis, D.R.6
-
28
-
-
0021367090
-
-
[10d] P. Krogsgard-Larsen, E. ø. Nielsen, D. R. Curtis, J. Med Chem. 1984, 27, 585-591.
-
(1984)
J. Med Chem.
, vol.27
, pp. 585-591
-
-
Krogsgard-Larsen, P.1
Nielsen, E.ø.2
Curtis, D.R.3
-
29
-
-
0024435507
-
-
[11a] J. J. Hansen, B. Nielsen, P. Krogsgaard-Larsen, L. Brehm, E. Ø. Nielsen, D. R. Curtis, J. Med. Chem. 1989, 32, 2254-2260.
-
(1989)
J. Med. Chem.
, vol.32
, pp. 2254-2260
-
-
Hansen, J.J.1
Nielsen, B.2
Krogsgaard-Larsen, P.3
Brehm, L.4
Nielsen, E.Ø.5
Curtis, D.R.6
-
30
-
-
2742547523
-
-
[11b] J J. Hansen, P. Krogsgaard-Larsen, J. Chem Soc., Chem. Commun. 1979, 87-88; J. Chem. Soc., Perkin Trans, 1 1980, 1826-1833.
-
(1979)
J. Chem Soc., Chem. Commun.
, pp. 87-88
-
-
Hansen, J.J.1
Krogsgaard-Larsen, P.2
-
31
-
-
2742547523
-
-
[11b] J J. Hansen, P. Krogsgaard-Larsen, J. Chem Soc., Chem. Commun. 1979, 87-88; J. Chem. Soc., Perkin Trans, 1 1980, 1826-1833.
-
(1980)
J. Chem. Soc., Perkin Trans, 1
, pp. 1826-1833
-
-
-
33
-
-
0019223440
-
-
[13a] P. Krogsgaard-Larsen, T. Honoré, J. J. Hansen, D. R. Curtis, D. Lodge, Nature 1980, 284, 64-66.
-
(1980)
Nature
, vol.284
, pp. 64-66
-
-
Krogsgaard-Larsen, P.1
Honoré, T.2
Hansen, J.J.3
Curtis, D.R.4
Lodge, D.5
-
37
-
-
84944067467
-
-
(Eds.: A. R. Katritzky, C. W. Rees), Pergamon Press, London, New York
-
For synthesis of 3-hydroxyisoxazoles in general see, e. g.: M. Sutharchanadevi, R. Murugan in Comprehensive Heterocyclic Chemistry, vol. 6 (Eds.: A. R. Katritzky, C. W. Rees), Pergamon Press, London, New York, 1996, p. 221.
-
(1996)
Comprehensive Heterocyclic Chemistry
, vol.6
, pp. 221
-
-
Sutharchanadevi, M.1
Murugan, R.2
-
40
-
-
0022380013
-
-
[17b] V. Jäger, M. Frey, Liebigs Ann. Chem. 1982, 817-820; M. Frey, V. Jäger, Synthesis 1985, 1100-1104.
-
(1985)
Synthesis
, pp. 1100-1104
-
-
Frey, M.1
Jäger, V.2
-
41
-
-
0013858776
-
-
[18a] Y. Kishida, T. Hiroako, J. Ide, A. Terada, N. Nakamura, Chem. Pharm. Bull. 1966, 14, 92.
-
(1966)
Chem. Pharm. Bull.
, vol.14
, pp. 92
-
-
Kishida, Y.1
Hiroako, T.2
Ide, J.3
Terada, A.4
Nakamura, N.5
-
42
-
-
2742542095
-
-
[18b] P. Krogsgaard-Larsen, S. B. Christensen, Acta Chem. Scand., B 1974, 28, 636-640; idem, ibid. 1976, 30, 281.
-
(1974)
Acta Chem. Scand., B
, vol.28
, pp. 636-640
-
-
Krogsgaard-Larsen, P.1
Christensen, S.B.2
-
43
-
-
0344334960
-
-
[18b] P. Krogsgaard-Larsen, S. B. Christensen, Acta Chem. Scand., B 1974, 28, 636-640; idem, ibid. 1976, 30, 281.
-
(1976)
Acta Chem. Scand., B
, vol.30
, pp. 281
-
-
Krogsgaard-Larsen, P.1
Christensen, S.B.2
-
44
-
-
0014111433
-
-
[19a] Y. Kishida, T. Hiracho, J. Ide, A. Terada, N. Nakamura, Chem. Pharm Bull. 1967, 75, 1025-1031; N. Nakamura, Chem. Pharm. Bull. 1971, 19, 46-51.
-
(1967)
Chem. Pharm Bull.
, vol.75
, pp. 1025-1031
-
-
Kishida, Y.1
Hiracho, T.2
Ide, J.3
Terada, A.4
Nakamura, N.5
-
45
-
-
85010542547
-
-
[19a] Y. Kishida, T. Hiracho, J. Ide, A. Terada, N. Nakamura, Chem. Pharm Bull. 1967, 75, 1025-1031; N. Nakamura, Chem. Pharm. Bull. 1971, 19, 46-51.
-
(1971)
Chem. Pharm. Bull.
, vol.19
, pp. 46-51
-
-
Nakamura, N.1
-
46
-
-
0002341842
-
-
[19b] A. R. Gagneux, F. Häfliger, R. Meier, C. M. Eugster, Tetrahedron Lett. 1965, 2081-2084.
-
(1965)
Tetrahedron Lett.
, pp. 2081-2084
-
-
Gagneux, A.R.1
Häfliger, F.2
Meier, R.3
Eugster, C.M.4
-
47
-
-
84918485561
-
-
[19c] A. Barco, S. Benetti, G. P. Pollini, P. G. Baraldi, M. Guarner, J. Chem. Research S 1979, 176-177.
-
(1979)
J. Chem. Research S
, pp. 176-177
-
-
Barco, A.1
Benetti, S.2
Pollini, G.P.3
Baraldi, P.G.4
Guarner, M.5
-
48
-
-
0000683502
-
-
N. Nakamura, Y. Tajima, S. Sakai, Heterocycles 1982, 17, 235-245.
-
(1982)
Heterocycles
, vol.17
, pp. 235-245
-
-
Nakamura, N.1
Tajima, Y.2
Sakai, S.3
-
49
-
-
0021672652
-
-
G. Schiewer, P. Krogsgaard-Larsen, Acta Chem. Scand., B 1984, 38, 815-819.
-
(1984)
Acta Chem. Scand., B
, vol.38
, pp. 815-819
-
-
Schiewer, G.1
Krogsgaard-Larsen, P.2
-
52
-
-
85066897001
-
-
[24a] A. J. Fatiadi, Synthesis 1976, 65-104; idem, ibid. 133-167.
-
(1976)
Synthesis
, pp. 65-104
-
-
Fatiadi, A.J.1
-
53
-
-
85066897001
-
-
[24a] A. J. Fatiadi, Synthesis 1976, 65-104; idem, ibid. 133-167.
-
Synthesis
, pp. 133-167
-
-
Fatiadi, A.J.1
-
54
-
-
0028805477
-
-
[24b] N. J. P. Broom, J. S. Elder, P. C. T. Hannan, J. E. Pons, P. J. O'Hanlon, G. Walker, J. Wilson, P. Woodall, J. Antibiot. 1995, 48, 1336-1344.
-
(1995)
J. Antibiot.
, vol.48
, pp. 1336-1344
-
-
Broom, N.J.P.1
Elder, J.S.2
Hannan, P.C.T.3
Pons, J.E.4
O'Hanlon, P.J.5
Walker, G.6
Wilson, J.7
Woodall, P.8
-
55
-
-
0026526289
-
-
[25a] A. Melikian, G. Schlewer, J.-P. Chambon, C. G. Wermuth, J. Med. Chem. 1992, 35, 4092-4097.
-
(1992)
J. Med. Chem.
, vol.35
, pp. 4092-4097
-
-
Melikian, A.1
Schlewer, G.2
Chambon, J.-P.3
Wermuth, C.G.4
-
58
-
-
84982334123
-
-
H. Göth, A. R. Gagneux, C. H. Eugster, H. Schmid, Helv. Chim Acta 1967, 50, 137-142; J. R. Geigy A.-G., Belg. Pat. 665,-249 (Dec. 10, 1965); Chem. Abstr. 1966, 65, 2266e.
-
(1967)
Helv. Chim Acta
, vol.50
, pp. 137-142
-
-
Göth, H.1
Gagneux, A.R.2
Eugster, C.H.3
Schmid, H.4
-
59
-
-
84982334123
-
-
Belg. Pat. 665,-249 (Dec. 10, 1965)
-
H. Göth, A. R. Gagneux, C. H. Eugster, H. Schmid, Helv. Chim Acta 1967, 50, 137-142; J. R. Geigy A.-G., Belg. Pat. 665,-249 (Dec. 10, 1965); Chem. Abstr. 1966, 65, 2266e.
-
(1966)
Chem. Abstr.
, vol.65
-
-
Geigy A-G, J.R.1
|