Rational Design of Vitamin D3 Analogues Which Selectively Restore Activity to a Vitamin D Receptor Mutant Associated with Rickets

Organic Letters

Volumn 4, Issue 22, 2002, Pages 3863-3866

  Swann, Steve L ^a   Bergh, Joel J ^a   Farach Carson, M Cindy ^a   Koh, John T ^a  

^a UNIVERSITY OF DELAWARE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CALCITRIOL RECEPTOR; CALCIUM; COLECALCIFEROL; DRUG DERIVATIVE; LIGAND;

ARTICLE; CELL LINE; CHEMICAL STRUCTURE; DRUG DESIGN; DRUG EFFECT; GENETICS; HUMAN; METABOLISM; MUTATION; RICKETS; STRUCTURE ACTIVITY RELATION; TRANSACTIVATION;

CALCIUM; CELL LINE; CHOLECALCIFEROL; DRUG DESIGN; HUMANS; LIGANDS; MODELS, MOLECULAR; MUTATION; RECEPTORS, CALCITRIOL; RICKETS; STRUCTURE-ACTIVITY RELATIONSHIP; TRANS-ACTIVATION (GENETICS);

EID: 0001474784     PISSN: 15237060     EISSN: None     Source Type: Journal    
DOI: 10.1021/ol0266931     Document Type: Article

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