Ligand binding to the serotonin 5HT3 receptor studied with a novel fluorescent ligand

Biochemistry

Volumn 37, Issue 45, 1998, Pages 15850-15864

  Tain, Ana Paula ^a   Hovius, Ruud ^a   Pick, Horst ^a   Blasey, Horst ^a,c   Bernard, Alain ^a,c   Surprenant, Annmarie ^a,d   Lundström, Kenneth ^b   Vogel, Horst ^a  

^a EPFL   (Switzerland)

^b F HOFFMANN LA ROCHE LTD   (Switzerland)

^c SERONO PHARMACEUTICAL RES INSTITUTE   (Switzerland)

^d UNIVERSITY OF SHEFFIELD   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

1,2,3,9 TETRAHYDRO 3 [(5 METHYL 1H IMIDAZOL 4 YL)METHYL] 9 [3 AMINO (N FLUORESCEINTHIOCARBAMOYL)PROPYL] 4H CARBAZOL 4 ONE; LIGAND; SEROTONIN 3 RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL CELL; ANISOTROPY; ARTICLE; BINDING SITE; CELL STRAIN BHK; DISSOCIATION CONSTANT; ELECTROPHYSIOLOGY; ENTHALPY; ENTROPY; LIGAND BINDING; NONHUMAN; PH; PRIORITY JOURNAL; RADIOASSAY; RECEPTOR OCCUPANCY; SPECTROFLUOROMETRY; STOICHIOMETRY; TEMPERATURE DEPENDENCE; THERMODYNAMICS;

ANIMALS; BINDING, COMPETITIVE; CARBAZOLES; CELL LINE; CRICETINAE; ELECTROPHYSIOLOGY; FLUORESCENCE POLARIZATION; FLUORESCENT DYES; HUMANS; IMIDAZOLES; INDOLES; KIDNEY; KINETICS; LIGANDS; RADIOLIGAND ASSAY; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT3; SEROTONIN ANTAGONISTS; SPECTROMETRY, FLUORESCENCE; THERMODYNAMICS; TRANSFECTION;

ANIMALIA;

EID: 20644440200     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi981812z     Document Type: Article

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