Antimicrobial activity of rhodanine-3-acetic acid derivatives

Bioorganic and Medicinal Chemistry

Volumn 25, Issue 6, 2017, Pages 1839-1845

  Krátký, Martin ^a   Vinšová, Jarmila ^a   Stolaříková, Jiřina ^b  

^a Charles University in Prague Faculty of Pharmacy   (Czech Republic)

^b Zdravotniho ustavu se sidlem v Ostrave   (Czech Republic)

Author keywords

2 (4 Oxo 2 thioxothiazolidin 3 yl)acetic acid; Amides; Antibacterial activity; Antifungal activity; Antimycobacterial activity; Condensation; Esters; In vitro activity; Rhodanine

Indexed keywords

2 (4 OXO 2 THIOXOTHIAZOLIDIN 3 YL) N PHENYLACETAMIDE DERIVATIVE; 2 (4 OXO 2 THIOXOTHIAZOLIDIN 3 YL)ACETIC ACID; 2 [4 OXO 5 (PYRIDIN 2 YLMETHYLENE) 2 THIOXOTHIAZOLIDIN 3 YL]ACETIC ACID; 2 [5 (2 ACETOXYBENZYLIDENE) 4 OXO 2 THIOXOTHIAZOLIDIN 3 YL]ACETIC ACID; 2 [5 (2 HYDROXYBENZYLIDENE) 4 OXO 2 THIOXOTHIAZOLIDIN 3 YL]ACETIC ACID; 2 [5 (3 HYDROXYBENZYLIDENE) 4 OXO 2 THIOXOTHIAZOLIDIN 3 YL]ACETIC ACID; 2 [5 (4 HYDROXYBENZYLIDENE) 4 OXO 2 THIOXOTHIAZOLIDIN 3 YL]ACETIC ACID; 2 [5 (5 BROMO 2 HYDROXYBENZYLIDENE) 4 OXO 2 THIOXOTHIAZOLIDIN 3 YL] N (4 CHLOROPHENYL)ACETAMIDE; 2 [5 (5 BROMO 2 HYDROXYBENZYLIDENE) 4 OXO 2 THIOXOTHIAZOLIDIN 3 YL]ACETIC ACID; 2 [5 (5 CHLORO 2 HYDROXYBENZYLIDENE) 4 OXO 2 THIOXOTHIAZOLIDIN 3 YL] N (4 CHLOROPHENYL)ACETAMIDE; 2 [5 (5 CHLORO 2 HYDROXYBENZYLIDENE) 4 OXO 2 THIOXOTHIAZOLIDIN 3 YL]ACETIC ACID; 4 (TRIFLUOROMETHYL)PHENYL 2 (4 OXO 2 THIOXOTHIAZOLIDIN 3 YL)ACETATE; 4 NITROPHENYLAMIDE; ACETIC ACID DERIVATIVE; ANTIINFECTIVE AGENT; ANTIMYCOBACTERIAL AGENT; BACITRACIN; FLUCONAZOLE; ISONIAZID; N (4 CHLOROPHENYL) 2 (4 OXO 2 THIOXOTHIAZOLIDIN 3 YL)ACETAMIDE; N (4 CHLOROPHENYL) 2 [4 OXO 5 (PYRIDIN 2 YLMETHYLENE) 2 THIOXOTHIAZOLIDIN 3 YL]ACETAMIDE; N (4 CHLOROPHENYL) 2 [5 (2 HYDROXYBENZYLIDENE) 4 OXO 2 THIOXOTHIAZOLIDIN 3 YL]ACETAMIDE; N (4 CHLOROPHENYL)AMIDE; RHODANINE 3 ACETIC DERIVATIVE; UNCLASSIFIED DRUG; ACETIC ACID; RHODANINE;

ANTIBACTERIAL ACTIVITY; ANTIBIOTIC SENSITIVITY; ANTIFUNGAL ACTIVITY; ANTIMICROBIAL ACTIVITY; ARTICLE; ATYPICAL MYCOBACTERIUM; CONTROLLED STUDY; DRUG SCREENING; DRUG SYNTHESIS; FUNGUS; GRAM NEGATIVE BACTERIUM; GRAM POSITIVE BACTERIUM; IN VITRO STUDY; METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; STRUCTURE ACTIVITY RELATION; CANDIDA; CARBON NUCLEAR MAGNETIC RESONANCE; CHEMISTRY; DRUG EFFECTS; INFRARED SPECTROPHOTOMETRY; MICROBIAL SENSITIVITY TEST; PROTON NUCLEAR MAGNETIC RESONANCE;

ACETIC ACID; ANTI-INFECTIVE AGENTS; CANDIDA; CARBON-13 MAGNETIC RESONANCE SPECTROSCOPY; GRAM-POSITIVE BACTERIA; METHICILLIN-RESISTANT STAPHYLOCOCCUS AUREUS; MICROBIAL SENSITIVITY TESTS; PROTON MAGNETIC RESONANCE SPECTROSCOPY; RHODANINE; SPECTROPHOTOMETRY, INFRARED;

EID: 85012012607     PISSN: 09680896     EISSN: 14643391     Source Type: Journal    
DOI: 10.1016/j.bmc.2017.01.045     Document Type: Article

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