Functional characterization of cholera toxin inhibitors using human intestinal organoids

Journal of Medicinal Chemistry

Volumn 59, Issue 14, 2016, Pages 6968-6972

  Zomer Van Ommen, Domenique D ^a   Pukin, Aliaksei V ^b   Fu, Ou ^b   Quarles Van Ufford, Linda H C ^b   Janssens, Hettie M ^c   Beekman, Jeffrey M ^a   Pieters, Roland J ^b  

^a UNIVERSITY MEDICAL CENTER UTRECHT   (Netherlands)

^b UTRECHT UNIVERSITY   (Netherlands)

^c SOPHIA CHILDREN S HOSPITAL   (Netherlands)

Author keywords

[No Author keywords available]

Indexed keywords

CHOLERA TOXIN; CHOLERA TOXIN B SUBUNIT; FORSKOLIN; ANTITOXIN;

ARTICLE; CYTOPLASM; DIARRHEA; DRUG SCREENING; ENZYME LINKED IMMUNOSORBENT ASSAY; HUMAN; IC50; INTESTINE CELL; LIPOPHILICITY; RECTUM BIOPSY; ANTAGONISTS AND INHIBITORS; CHEMICAL STRUCTURE; CHEMISTRY; DOSE RESPONSE; DRUG EFFECTS; INTESTINE; STRUCTURE ACTIVITY RELATION;

ANTITOXINS; CHOLERA TOXIN; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; INTESTINES; MOLECULAR STRUCTURE; ORGANOIDS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84979940070     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/acs.jmedchem.6b00770     Document Type: Article

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