SCOPUS 정보 검색 플랫폼

Volumn 351, Issue 6270, 2016, Pages 241-246

Organic chemistry: Strain-release amination

(14) Gianatassio, Ryan a Lopchuk, Justin M a Wang, Jie a Pan, Chung Mao a Malins, Lara R a Prieto, Liher a Brandt, Thomas A b Collins, Michael R b Gallego, Gary M b Sach, Neal W b Spangler, Jillian E b Zhu, Huichin b Zhu, Jinjiang b Baran, Phil S a

a SCRIPPS RESEARCH INSTITUTE (United States)

b PFIZER INC (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ACETAL; ACETAL DERIVATIVE; ALKENE; ANILINE; AZETIDINE; AZETIDINE DERIVATIVE; BENZYLAMINE; BUTANE; CYCLOBUTANE; CYCLOBUTANE DERIVATIVE; CYCLOPENTANE; CYCLOPENTANE DERIVATIVE; DEUTERIUM; ELECTROPHILE; ETHER DERIVATIVE; FLUORINE; GRIGNARD REAGENT; HYDROXYL GROUP; LEWIS ACID; MALEIMIDE; MECYSTEINE; MOLECULAR SCAFFOLD; NUCLEOPHILE; SULFONE; TERTIARY AMINE; TETRAHYDROISOQUINOLINE; THIOL; DRUG; PEPTIDE;

AMINATION; ARTICLE; BIOCONJUGATION; CARBON BOND; CARBON NITROGEN BOND; CHEMICAL BOND; CONJUGATION; ELECTROPHILICITY; NUCLEOPHILICITY; PRIORITY JOURNAL; STRAIN RELEASE AMINATION; SYNTHESIS; MEDICINAL CHEMISTRY;

AMINATION; CHEMISTRY TECHNIQUES, SYNTHETIC; CHEMISTRY, PHARMACEUTICAL; PEPTIDES; PHARMACEUTICAL PREPARATIONS;

EID: 84954409400 PISSN: 00368075 EISSN: 10959203 Source Type: Journal
DOI: 10.1126/science.aad6252 Document Type: Article

Times cited : (326)

References (38)

1
- 79955419410
- N. A. Meanwell, J. Med. Chem. 54, 2529-2591 (2011).
- (2011) J. Med. Chem. , vol.54 , pp. 2529-2591
- Meanwell, N.A.¹

2
- 84921743196
- C. Ni, M. Hu, J. Hu, Chem. Rev. 115, 765-825 (2015).
- (2015) Chem. Rev. , vol.115 , pp. 765-825
- Ni, C.¹ Hu, M.² Hu, J.³

3
- 84870541226
- Y. Fujiwara et al., Nature 492, 95-99 (2012).
- (2012) Nature , vol.492 , pp. 95-99
- Fujiwara, Y.¹

4
- 84923319254
- M. V. Westphal, B. T. Wolfstädter, J. M. Plancher, J. Gatfield, E. M. Carreira, ChemMedChem 10, 461-469 (2015).
- (2015) ChemMedChem , vol.10 , pp. 461-469
- Westphal, M.V.¹ Wolfstädter, B.T.² Plancher, J.M.³ Gatfield, J.⁴ Carreira, E.M.⁵

5
- 84925459184
- Q. Michaudel, Y. Ishihara, P. S. Baran, Acc. Chem. Res. 48, 712-721 (2015).
- (2015) Acc. Chem. Res. , vol.48 , pp. 712-721
- Michaudel, Q.¹ Ishihara, Y.² Baran, P.S.³

6
- 84859797196
- A. F. Stepan et al., J. Med. Chem. 55, 3414-3424 (2012).
- (2012) J. Med. Chem. , vol.55 , pp. 3414-3424
- Stepan, A.F.¹

7
- 0000733272
- K. B. Wiberg, V. Z. Williams, J. Org. Chem. 35, 369-373 (1970).
- (1970) J. Org. Chem. , vol.35 , pp. 369-373
- Wiberg, K.B.¹ Williams, V.Z.²

8
- 0000741608
- M. D. Levin, P. Kaszynski, J. Michl, Chem. Rev. 100, 169-234 (2000).
- (2000) J. Michl, Chem. Rev. , vol.100 , pp. 169-234
- Levin, M.D.¹ Kaszynski, P.²

9
- 0001343052
- K. B. Wiberg, Chem. Rev. 89, 975-983 (1989).
- (1989) Chem. Rev. , vol.89 , pp. 975-983
- Wiberg, K.B.¹

10
- 80052249648
- K. D. Bunker, N. W. Sach, Q. Huang, P. F. Richardson, Org. Lett. 13, 4746-4748 (2011).
- (2011) Org. Lett. , vol.13 , pp. 4746-4748
- Bunker, K.D.¹ Sach, N.W.² Huang, Q.³ Richardson, P.F.⁴

11
- 79955794782
- L. Zehnder et al., J. Med. Chem. 54, 3368-3385 (2011).
- (2011) J. Med. Chem. , vol.54 , pp. 3368-3385
- Zehnder, L.¹

12
- 84877147885
- B. L. Bennett et. al., PCT Int. Appl. WO 2012145569 (2012).
- (2012) PCT Int. Appl.
- Bennett, B.L.¹

13
- 84994682847
- K. Hayashi et. al., PCT Int. Appl. WO 2013024895 (2013).
- (2013) PCT Int. Appl.
- Hayashi, K.¹

14
- 0001530046
- K. B. Wiberg, F. H. Walker, J. Am. Chem. Soc. 104, 5239-5240 (1982).
- (1982) J. Am. Chem. Soc. , vol.104 , pp. 5239-5240
- Wiberg, K.B.¹ Walker, F.H.²

15
- 84985532474
- K. B. Wiberg, Angew. Chem. Int. Ed. Engl. 25, 312-322 (1986).
- (1986) Angew. Chem. Int. Ed. Engl. , vol.25 , pp. 312-322
- Wiberg, K.B.¹

16
- 0000096835
- H. C. Kolb, M. G. Finn, K. B. Sharpless, Angew. Chem. Int. Ed. 40, 2004-2021 (2001).
- (2001) Angew. Chem. Int. Ed. , vol.40 , pp. 2004-2021
- Kolb, H.C.¹ Finn, M.G.² Sharpless, K.B.³

17
- 0025170701
- E. W. Della, D. K. Taylor, J. Tsanaktsidis, Tetrahedron Lett. 31, 5219-5220 (1990).
- (1990) Tetrahedron Lett. , vol.31 , pp. 5219-5220
- Della, E.W.¹ Taylor, D.K.² Tsanaktsidis, J.³

18
- 0034054844
- M. Messner, S. I. Kozhushkov, A. de Meijere, Eur. J. Org. Chem. 2000, 1137-1155 (2000).
- (2000) Eur. J. Org. Chem. , vol.2000 , pp. 1137-1155
- Messner, M.¹ Kozhushkov, S.I.² De Meijere, A.³

19
- 84866973898
- S. G. Davies, A. M. Fletcher, P. M. Roberts, J. E. Thomson, Tetrahedron Asymmetry 23, 1111-1153 (2012).
- (2012) Tetrahedron Asymmetry , vol.23 , pp. 1111-1153
- Davies, S.G.¹ Fletcher, A.M.² Roberts, P.M.³ Thomson, J.E.⁴

20
- 53249110866
- C. J. Rohbogner, G. C. Clososki, P. Knochel, Angew. Chem. Int. Ed. Engl. 47, 1503-1507 (2008).
- (2008) Angew. Chem. Int. Ed. Engl. , vol.47 , pp. 1503-1507
- Rohbogner, C.J.¹ Clososki, G.C.² Knochel, P.³

21
- 53549128637
- A. Brandi, S. Cicchi, F. M. Cordero, Chem. Rev. 108, 3988-4035 (2008).
- (2008) Chem. Rev. , vol.108 , pp. 3988-4035
- Brandi, A.¹ Cicchi, S.² Cordero, F.M.³

22
- 41549087781
- Y. Ikee et al., Chem. Pharm. Bull. (Tokyo) 56, 346-356 (2008).
- (2008) Chem. Pharm. Bull. (Tokyo) , vol.56 , pp. 346-356
- Ikee, Y.¹

23
- 33746509098
- M. L. Wrobleski et al., Bioorg. Med. Chem. Lett. 16, 3859-3863 (2006).
- (2006) Bioorg. Med. Chem. Lett. , vol.16 , pp. 3859-3863
- Wrobleski, M.L.¹

24
- 0001291047
- K. B. Wiberg, R. P. Ciula, J. Am. Chem. Soc. 81, 5261-5262 (1959).
- (1959) J. Am. Chem. Soc. , vol.81 , pp. 5261-5262
- Wiberg, K.B.¹ Ciula, R.P.²

25
- 0001111398
- Academic Press, New York
- K. B. Wiberg, in Advances in Alicyclic Chemistry (Academic Press, New York, 1968), vol. 2, pp. 185-254.
- (1968) Advances in Alicyclic Chemistry , vol.2 , pp. 185-254
- Wiberg, K.B.¹

26
- 84928336677
- M. A. A. Walczak, T. Krainz, P. Wipf, Acc. Chem. Res. 48, 1149-1158 (2015).
- (2015) Acc. Chem. Res. , vol.48 , pp. 1149-1158
- Walczak, M.A.A.¹ Krainz, T.² Wipf, P.³

27
- 0042904726
- G. M. Lampman, J. C. Aumiller, Org. Synth. 51, 55-59 (1971).
- (1971) Org. Synth. , vol.51 , pp. 55-59
- Lampman, G.M.¹ Aumiller, J.C.²

28
- 0023891764
- Y. Gaoni, Tetrahedron Lett. 29, 1591-1594 (1988).
- (1988) Tetrahedron Lett. , vol.29 , pp. 1591-1594
- Gaoni, Y.¹

29
- 21844526388
- Y. Gaoni, Org. Prep. Proced. Int. 27, 185-212 (1995).
- (1995) Org. Prep. Proced. Int. , vol.27 , pp. 185-212
- Gaoni, Y.¹

30
- 33750537101
- S. M. Jeffery, C. J. M. Stirling, J. Chem. Soc., Perkin Trans. 2, 1617-1624 (1993).
- (1993) J. Chem. Soc., Perkin Trans. , vol.2 , pp. 1617-1624
- Jeffery, S.M.¹ Stirling, C.J.M.²

31
- 84924565933
- O. Boutureira, G. J. L. Bernardes, Chem. Rev. 115, 2174-2195 (2015).
- (2015) Chem. Rev. , vol.115 , pp. 2174-2195
- Boutureira, O.¹ Bernardes, G.J.L.²

32
- 84910015748
- C. S. McKay, M. G. Finn, Chem. Biol. 21, 1075-1101 (2014).
- (2014) Chem. Biol. , vol.21 , pp. 1075-1101
- McKay, C.S.¹ Finn, M.G.²

33
- 81355139629
- N. Stephanopoulos, M. B. Francis, Nat. Chem. Biol. 7, 876-884 (2011).
- (2011) Nat. Chem. Biol. , vol.7 , pp. 876-884
- Stephanopoulos, N.¹ Francis, M.B.²

34
- 77949341762
- J. Kalia, R. T. Raines, Curr. Org. Chem. 14, 138-147 (2010).
- (2010) Curr. Org. Chem. , vol.14 , pp. 138-147
- Kalia, J.¹ Raines, R.T.²

35
- 84916912015
- Y. H. Lau, P. de Andrade, Y. Wu, D. R. Spring, Chem. Soc. Rev. 44, 91-102 (2015).
- (2015) Chem. Soc. Rev. , vol.44 , pp. 91-102
- Lau, Y.H.¹ De Andrade, P.² Wu, Y.³ Spring, D.R.⁴

36
- 84876702107
- A. M. Spokoyny et al., J. Am. Chem. Soc. 135, 5946-5949 (2013).
- (2013) J. Am. Chem. Soc. , vol.135 , pp. 5946-5949
- Spokoyny, A.M.¹

37
- 84940723071
- Y. Wang, D. H.-C. Chou, Angew. Chem. Int. Ed. 54, 10931-10934 (2015).
- (2015) Angew. Chem. Int. Ed. , vol.54 , pp. 10931-10934
- Wang, Y.¹ Chou, D.H.-C.²

38
- 84926354846
- S. P. Brown, A. B. Smith 3rd, J. Am. Chem. Soc. 137, 4034-4037 (2015).
- (2015) J. Am. Chem. Soc. , vol.137 , pp. 4034-4037
- Brown, S.P.¹ Smith, A.B.²

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