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Volumn 35, Issue 3, 2015, Pages 501-511

Quantification of 11 Cyohimbine binding to α 2 adrenoceptors in rat brain in vivo

Author keywords

alpha 2 adrenoceptors; amphetamine challenge; Inhibition plot; reference region; 11C yohimbine

Indexed keywords

ALPHA 2 ADRENERGIC RECEPTOR; AMPHETAMINE; NORADRENALIN; UNCLASSIFIED DRUG; YOHIMBINE; YOHIMBINE C 11; CARBON; RADIOPHARMACEUTICAL AGENT;

EID: 84937520203     PISSN: 07438346     EISSN: 14765543     Source Type: Journal    
DOI: 10.1038/jcbfm.2014.225     Document Type: Article
Times cited : (15)

References (40)
  • 1
    • 0345391014 scopus 로고    scopus 로고
    • Up-regulation of immunolabeled alpha2a-Adrenoceptors, gi coupling proteins, and regulatory receptor kinases in the prefrontal cortex of depressed suicides
    • Garcia-Sevilla JA, Escriba PV, Ozaita A, La Harpe R, Walzer C, Eytan A et al. Up-regulation of immunolabeled alpha2A-Adrenoceptors, Gi coupling proteins, and regulatory receptor kinases in the prefrontal cortex of depressed suicides. J Neurochem 1999; 72: 282-291.
    • (1999) J Neurochem , vol.72 , pp. 282-291
    • Garcia-Sevilla, J.A.1    Escriba, P.V.2    Ozaita, A.3    La Harpe, R.4    Walzer, C.5    Eytan, A.6
  • 2
    • 32544460565 scopus 로고    scopus 로고
    • Compensatory changes in the noradrenergic nervous system in the locus ceruleus and hippocampus of postmortem subjects with Alzheimer's disease and dementia with lewy bodies
    • Szot P, White SS, Greenup JL, Leverenz JB, Peskind ER, Raskind MA. Compensatory changes in the noradrenergic nervous system in the locus ceruleus and hippocampus of postmortem subjects with Alzheimer's disease and dementia with Lewy bodies. J Neurosci 2006; 26: 467-478.
    • (2006) J Neurosci , vol.26 , pp. 467-478
    • Szot, P.1    White, S.S.2    Greenup, J.L.3    Leverenz, J.B.4    Peskind, E.R.5    Raskind, M.A.6
  • 4
    • 17144475031 scopus 로고    scopus 로고
    • Agonist and antagonist actions of yohimbine as compared to fluparoxan at alpha 2)-Adrenergic receptors (ar)s, serotonin (5-ht)(1a), 5-ht1b, 5-ht1d and dopamine d-2 and d-3 receptors significance for the modulation of frontocortical monoaminergic transmission and depressive states
    • Millan MJ, Newman-Tancredi A, Audinot V, Cussac D, Lejeune F, Nicolas JP et al. Agonist and antagonist actions of yohimbine as compared to fluparoxan at alpha (2)-Adrenergic receptors (AR)s, serotonin (5-HT)(1A), 5-HT1B, 5-HT1D and dopamine D-2 and D-3 receptors. Significance for the modulation of frontocortical monoaminergic transmission and depressive states. Synapse 2000; 35: 79-95.
    • (2000) Synapse , vol.35 , pp. 79-95
    • Millan, M.J.1    Newman-Tancredi, A.2    Audinot, V.3    Cussac, D.4    Lejeune, F.5    Nicolas, J.P.6
  • 5
    • 34247556375 scopus 로고    scopus 로고
    • Detection of alpha2-Adrenergic receptors in brain of living pig with 11c-yohimbine
    • Jakobsen S, Pedersen K, Smith DF, Jensen SB, Munk OL, Cumming P. Detection of alpha2-Adrenergic receptors in brain of living pig with 11C-yohimbine. J Nucl Med 2006; 47: 2008-2015.
    • (2006) J Nucl Med , vol.47 , pp. 2008-2015
    • Jakobsen, S.1    Pedersen, K.2    Smith, D.F.3    Jensen, S.B.4    Munk, O.L.5    Cumming, P.6
  • 6
    • 84861880601 scopus 로고    scopus 로고
    • Amphetamine challenge decreases yohimbine binding to alpha2 adrenoceptors in landrace pig brain
    • Landau AM, Doudet DJ, Jakobsen S. Amphetamine challenge decreases yohimbine binding to alpha2 adrenoceptors in Landrace pig brain. Psychopharmacology (Berl) 2012; 222: 155-163.
    • (2012) Psychopharmacology (Berl , vol.222 , pp. 155-163
    • Landau, A.M.1    Doudet, D.J.2    Jakobsen, S.3
  • 7
    • 0028051572 scopus 로고
    • Effects of blood-flow on [c-11] raclopride binding in the brain-model simulations and kinetic-Analysis of pet data
    • Logan J, Volkow ND, Fowler JS, Wang GJ, Dewey SL, Macgregor R et al. Effects of blood-flow on [C-11] raclopride binding in the brain-model simulations and kinetic-Analysis of pet data. J Cereb Blood Flow Metab 1994; 14: 995-1010.
    • (1994) J Cereb Blood Flow Metab , vol.14 , pp. 995-1010
    • Logan, J.1    Volkow, N.D.2    Fowler, J.S.3    Wang, G.J.4    Dewey, S.L.5    Macgregor, R.6
  • 8
    • 0002732079 scopus 로고
    • Transient analysis of irreversible and reversible tracer binding in human brain
    • In: Battistin L, Gerstenbrand F (eds) Alan R Liss: New York, NY, USA
    • Gjedde A, Wong D, Wagner H. Transient analysis of irreversible and reversible tracer binding in human brain. In: Battistin L, Gerstenbrand F (eds). PET and NMR: New Perspectives in Neuroimaging and in Clinical Neurochemistry. Alan R Liss: New York, NY, USA, 1986; 223-235.
    • (1986) PET and NMR: New Perspectives in Neuroimaging and in Clinical Neurochemistry , pp. 223-235
    • Gjedde, A.1    Wong, D.2    Wagner, H.3
  • 9
    • 33646047272 scopus 로고    scopus 로고
    • Receptor occupancy in absence of reference region
    • Gjedde A, Wong DF. Receptor occupancy in absence of reference region. Neuroimage 2000; 11: S48.
    • (2000) Neuroimage , vol.11 , pp. S48
    • Gjedde, A.1    Wong, D.F.2
  • 10
    • 0032521354 scopus 로고    scopus 로고
    • Mechanisms of amphetamine action revealed in mice lacking the dopamine transporter
    • Jones SR, Gainetdinov RR, Wightman RM, Caron MG. Mechanisms of amphetamine action revealed in mice lacking the dopamine transporter. J Neurosci 1998; 18: 1979-1986.
    • (1998) J Neurosci , vol.18 , pp. 1979-1986
    • Jones, S.R.1    Gainetdinov, R.R.2    Wightman, R.M.3    Caron, M.G.4
  • 11
    • 0025127930 scopus 로고
    • Graphical analysis of reversible radioligand binding from time-Activity measurements applied to [n-11c-methyl]-(-)-cocaine pet studies in human subjects
    • Logan J, Fowler JS, Volkow ND, Wolf AP, Dewey SL, Schlyer DJ et al. Graphical analysis of reversible radioligand binding from time-Activity measurements applied to [N-11C-methyl]-(-)-cocaine PET studies in human subjects. J Cereb Blood Flow Metab 1990; 10: 740-747.
    • (1990) J Cereb Blood Flow Metab , vol.10 , pp. 740-747
    • Logan, J.1    Fowler, J.S.2    Volkow, N.D.3    Wolf, A.P.4    Dewey, S.L.5    Schlyer, D.J.6
  • 13
    • 57349138730 scopus 로고    scopus 로고
    • Basic cns drug transport and binding kinetics in vivo
    • Begley DJ, Bradbury MW, Kreuter J (eds Marcel Dekker: New York, NY, USA
    • Gjedde A, Gee A, Smith D. Basic CNS drug transport and binding kinetics in vivo. Begley DJ, Bradbury MW, Kreuter J (eds). The Blood-Brain Barrier and Drug Delivery to the CNS. Marcel Dekker: New York, NY, USA, 2000; 225-242.
    • (2000) The Blood-Brain Barrier and Drug Delivery to the CNS , pp. 225-242
    • Gjedde, A.1    Gee, A.2    Smith, D.3
  • 15
    • 0028894431 scopus 로고
    • Benzodiazepine receptor quantification in vivo in humans using [11c]flumazenil and pet: Application of the steady-state principle
    • Lassen NA, Bartenstein PA, Lammertsma AA, Prevett MC, Turton DR, Luthra SK et al. Benzodiazepine receptor quantification in vivo in humans using [11C]flumazenil and PET: application of the steady-state principle. J Cereb Blood Flow Metab 1995; 15: 152-165.
    • (1995) J Cereb Blood Flow Metab , vol.15 , pp. 152-165
    • Lassen, N.A.1    Bartenstein, P.A.2    Lammertsma, A.A.3    Prevett, M.C.4    Turton, D.R.5    Luthra, S.K.6
  • 17
    • 0028292989 scopus 로고
    • Platelet alpha 2-Adrenergic receptor binding and the effects of d-Amphetamine in boys with attention deficit hyperactivity disorder
    • Shekim WO, Bylund DB, Hodges K, Glaser R, Ray-Prenger C, Oetting G. Platelet alpha 2-Adrenergic receptor binding and the effects of d-Amphetamine in boys with attention deficit hyperactivity disorder. Neuropsychobiology 1994; 29: 120-124.
    • (1994) Neuropsychobiology , vol.29 , pp. 120-124
    • Shekim, W.O.1    Bylund, D.B.2    Hodges, K.3    Glaser, R.4    Ray-Prenger, C.5    Oetting, G.6
  • 18
    • 0034102018 scopus 로고    scopus 로고
    • Dose-dependent pharmacokinetics of cyclosporin a in rats: Events in tissues
    • Tanaka C, Kawai R, Rowland M. Dose-Dependent pharmacokinetics of cyclosporin A in rats: events in tissues. Drug Metab Dispos 2000; 28: 582-589.
    • (2000) Drug Metab Dispos , vol.28 , pp. 582-589
    • Tanaka, C.1    Kawai, R.2    Rowland, M.3
  • 19
    • 0028289554 scopus 로고
    • Evaluation of ultrafiltration for the free-fraction determination of single photon emission computed tomography (spect) radiotracers: Beta-cit, ibf, and iomazenil
    • Gandelman MS, Baldwin RM, Zoghbi SS, Zea-Ponce Y, Innis RB. Evaluation of ultrafiltration for the free-fraction determination of single photon emission computed tomography (SPECT) radiotracers: beta-CIT, IBF, and iomazenil. J Pharm Sci 1994; 83: 1014-1019.
    • (1994) J Pharm Sci , vol.83 , pp. 1014-1019
    • Gandelman, M.S.1    Baldwin, R.M.2    Zoghbi, S.S.3    Zea-Ponce, Y.4    Innis, R.B.5
  • 20
    • 0017724596 scopus 로고
    • Decrease in neostriatal blood flow after d-Amphetamine administration or electrical stimulation of the substantia nigra
    • Lavyne MH, Koltun WA, Clement JA, Rosene DL, Pickren KS, Zervas NT et al. Decrease in neostriatal blood flow after D-Amphetamine administration or electrical stimulation of the substantia nigra. Brain Res 1977; 135: 77-86.
    • (1977) Brain Res , vol.135 , pp. 77-86
    • Lavyne, M.H.1    Koltun, W.A.2    Clement, J.A.3    Rosene, D.L.4    Pickren, K.S.5    Zervas, N.T.6
  • 21
    • 0016703166 scopus 로고
    • Central noradrenergic regulation of cerebral blood flow and vascular permeability
    • Raichle ME, Hartman BK, Eichling JO, Sharpe LG. Central noradrenergic regulation of cerebral blood flow and vascular permeability. Proc Natl Acad Sci USA 1975; 72: 3726-3730.
    • (1975) Proc Natl Acad Sci USA , vol.72 , pp. 3726-3730
    • Raichle, M.E.1    Hartman, B.K.2    Eichling, J.O.3    Sharpe, L.G.4
  • 22
    • 73749084522 scopus 로고    scopus 로고
    • Multi-graphical analysis of dynamic pet
    • Zhou Y, Ye W, Brasic JR, Wong DF. Multi-graphical analysis of dynamic PET. Neuroimage 2010; 49: 2947-2957.
    • (2010) Neuroimage , vol.49 , pp. 2947-2957
    • Zhou, Y.1    Ye, W.2    Brasic, J.R.3    Wong, D.F.4
  • 23
    • 0020334176 scopus 로고
    • Characteristics of the [h-3]-labeled yohimbine binding on rat-brain alpha-2-Adrenoceptors
    • Rouot B, Quennedey MC, Schwartz J. Characteristics of the [H-3]-labeled yohimbine binding on rat-brain alpha-2-Adrenoceptors. Naunyn Schmiedebergs Arch Pharmacol 1982; 321: 253-259.
    • (1982) Naunyn Schmiedebergs Arch Pharmacol , vol.321 , pp. 253-259
    • Rouot, B.1    Quennedey, M.C.2    Schwartz, J.3
  • 24
    • 0023684053 scopus 로고
    • Subtypes of alpha 2-Adrenoceptors: Pharmacological and molecular biological evidence converge
    • Bylund DB. Subtypes of alpha 2-Adrenoceptors: pharmacological and molecular biological evidence converge. Trends Pharmacol Sci 1988; 9: 356-361.
    • (1988) Trends Pharmacol Sci , vol.9 , pp. 356-361
    • Bylund, D.B.1
  • 26
    • 0027753216 scopus 로고
    • Characterization of subtypes of alpha-2 adrenoceptors in the human brain
    • Ordway GA, Jaconetta SM, Halaris AE. Characterization of subtypes of alpha-2 adrenoceptors in the human brain. J Pharmacol Exp Ther 1993; 264: 967-976.
    • (1993) J Pharmacol Exp Ther , vol.264 , pp. 967-976
    • Ordway, G.A.1    Jaconetta, S.M.2    Halaris, A.E.3
  • 27
    • 0023358080 scopus 로고
    • Pharmacological evidence for alpha-2 adrenoceptor heterogeneity: Differential binding properties of [3h]rauwolscine and [3h]idazoxan in rat brain
    • Boyajian CL, Leslie FM. Pharmacological evidence for alpha-2 adrenoceptor heterogeneity: differential binding properties of [3H]rauwolscine and [3H]idazoxan in rat brain. J Pharmacol Exp Ther 1987; 241: 1092-1098.
    • (1987) J Pharmacol Exp Ther , vol.241 , pp. 1092-1098
    • Boyajian, C.L.1    Leslie, F.M.2
  • 29
    • 0023354702 scopus 로고
    • Anatomical evidence for alpha-2 adrenoceptor heterogeneity: Differential autoradiographic distributions of [3h] rauwolscine and [3h] idazoxan in rat brain
    • Boyajian CL, Loughlin SE, Leslie FM. Anatomical evidence for alpha-2 adrenoceptor heterogeneity: differential autoradiographic distributions of [3H]rauwolscine and [3H]idazoxan in rat brain. J Pharmacol Exp Ther 1987; 241: 1079-1091.
    • (1987) J Pharmacol Exp Ther , vol.241 , pp. 1079-1091
    • Boyajian, C.L.1    Loughlin, S.E.2    Leslie, F.M.3
  • 30
    • 39149130282 scopus 로고    scopus 로고
    • Dopamine binds to alpha 2)-Adrenergic receptors in the song control system of zebra finches (taeniopygia guttata)
    • Cornil CA, Castelino CB, Ball GF. Dopamine binds to alpha(2)-Adrenergic receptors in the song control system of zebra finches (Taeniopygia guttata). J Chem Neuroanat 2008; 35: 202-215.
    • (2008) J Chem Neuroanat , vol.35 , pp. 202-215
    • Cornil, C.A.1    Castelino, C.B.2    Ball, G.F.3
  • 31
    • 0032589266 scopus 로고    scopus 로고
    • Ordway ga. Alpha2c adrenoceptors inhibit adenylyl cyclase in mouse striatum: Potential activation by dopamine
    • Zhang W, Klimek V, Farley JT, Zhu MY, Ordway GA. alpha2C adrenoceptors inhibit adenylyl cyclase in mouse striatum: potential activation by dopamine. J Pharmacol Exp Ther 1999; 289: 1286-1292.
    • (1999) J Pharmacol Exp Ther , vol.289 , pp. 1286-1292
    • Zhang, W.1    Klimek, V.2    Farley, J.T.3    Zhu, M.Y.4
  • 32
    • 10844294216 scopus 로고    scopus 로고
    • Estimation of endogenous noradrenaline release in rat brain in vivo using [3h] rx 821002
    • Tyacke RJ, Robinson ES, Lalies MD, Hume SP, Hudson AL, Nutt DJ. Estimation of endogenous noradrenaline release in rat brain in vivo using [3H]RX 821002. Synapse 2005; 55: 126-132.
    • (2005) Synapse , vol.55 , pp. 126-132
    • Tyacke, R.J.1    Robinson, E.S.2    Lalies, M.D.3    Hume, S.P.4    Hudson, A.L.5    Nutt, D.J.6
  • 33
    • 0028183038 scopus 로고
    • Characterization of [3h]rx821002 binding to alpha-2 adrenergic receptor subtypes
    • O'Rourke MF, Blaxall HS, Iversen LJ, Bylund DB. Characterization of [3H]RX821002 binding to alpha-2 adrenergic receptor subtypes. J Pharmacol Exp Ther 1994; 268: 1362-1367.
    • (1994) J Pharmacol Exp Ther , vol.268 , pp. 1362-1367
    • O'Rourke, M.F.1    Blaxall, H.S.2    Iversen, L.J.3    Bylund, D.B.4
  • 34
    • 0025647855 scopus 로고
    • The role of cytochromes p-450 in cyclosporine metabolism
    • discussion 1309-1311
    • Watkins PB. The role of cytochromes P-450 in cyclosporine metabolism. J Am Acad Dermatol 1990; 23: 1301-1309, discussion 1309-1311.
    • (1990) J Am Acad Dermatol , vol.23 , pp. 1301-1309
    • Watkins, P.B.1
  • 35
    • 0036129441 scopus 로고    scopus 로고
    • Toxicokinetics of amphetamines: Metabolism and toxicokinetic data of designer drugs, amphetamine, methamphetamine, and their n-Alkyl derivatives
    • Kraemer T, Maurer HH. Toxicokinetics of amphetamines: metabolism and toxicokinetic data of designer drugs, amphetamine, methamphetamine, and their N-Alkyl derivatives. Ther Drug Monit 2002; 24: 277-289.
    • (2002) Ther Drug Monit , vol.24 , pp. 277-289
    • Kraemer, T.1    Maurer, H.H.2
  • 36
    • 0029996133 scopus 로고    scopus 로고
    • The binding of cyclosporin a to human plasma: An in vitro microdialysis study
    • Yang H, Elmquist WF. The binding of cyclosporin A to human plasma: an in vitro microdialysis study. Pharm Res 1996; 13: 622-627.
    • (1996) Pharm Res , vol.13 , pp. 622-627
    • Yang, H.1    Elmquist, W.F.2
  • 37
    • 3543004156 scopus 로고    scopus 로고
    • Human sympathetic activation by alpha2-Adrenergic blockade with yohimbine: Bimodal, epistatic influence of cytochrome p450-mediated drug metabolism
    • Le Corre P, Parmer RJ, Kailasam MT, Kennedy BP, Skaar TP, Ho H et al. Human sympathetic activation by alpha2-Adrenergic blockade with yohimbine: bimodal, epistatic influence of cytochrome P450-mediated drug metabolism. Clin Pharmacol Ther 2004; 76: 139-153.
    • (2004) Clin Pharmacol Ther , vol.76 , pp. 139-153
    • Le Corre, P.1    Parmer, R.J.2    Kailasam, M.T.3    Kennedy, B.P.4    Skaar, T.P.5    Ho, H.6
  • 38
    • 0023948926 scopus 로고
    • Regional distribution of cytochrome p-450 in the rat brain: Spectral quantitation and contribution of p-450b,e, and p-450c,d
    • Warner M, Kohler C, Hansson T, Gustafsson JA. Regional distribution of cytochrome P-450 in the rat brain: spectral quantitation and contribution of P-450b,e, and P-450c,d. J Neurochem 1988; 50: 1057-1065.
    • (1988) J Neurochem , vol.50 , pp. 1057-1065
    • Warner, M.1    Kohler, C.2    Hansson, T.3    Gustafsson, J.A.4
  • 39
    • 0034962049 scopus 로고    scopus 로고
    • Increased noradrenaline release from rat preoptic area during and after sevoflurane and isoflurane anesthesia
    • Anzawa N, Kushikata T, Ohkawa H, Yoshida H, Kubota T, Matsuki A. Increased noradrenaline release from rat preoptic area during and after sevoflurane and isoflurane anesthesia. Can J Anaesth 2001; 48: 462-465.
    • (2001) Can J Anaesth , vol.48 , pp. 462-465
    • Anzawa, N.1    Kushikata, T.2    Ohkawa, H.3    Yoshida, H.4    Kubota, T.5    Matsuki, A.6
  • 40
    • 80052618211 scopus 로고    scopus 로고
    • Isoflurane anaesthesia differentially affects the amphetamine sensitivity of agonist and antagonist d2/d3 positron emission tomography radiotracers: Implications for in vivo imaging of dopamine release
    • McCormick PN, Ginovart N, Wilson AA. Isoflurane anaesthesia differentially affects the amphetamine sensitivity of agonist and antagonist D2/D3 positron emission tomography radiotracers: implications for in vivo imaging of dopamine release. Mol Imaging Biol 2011; 13: 737-746.
    • (2011) Mol Imaging Biol , vol.13 , pp. 737-746
    • McCormick, P.N.1    Ginovart, N.2    Wilson, A.A.3


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