Inhibition of monocarboxylate transporter by N-cyanosulphonamide S0859

European Journal of Pharmacology

Volumn 762, Issue , 2015, Pages 344-349

  Heidtmann, Hella ^a   Ruminot, Iván ^a   Becker, Holger M ^a   Deitmer, Joachim W ^a  

^a University of Koblenz Landau   (Germany)

Author keywords

Lactate; MCT; NBCe1; pHi< inf>; Xenopus oocyte

Indexed keywords

KETONE BODY; LACTIC ACID; MONOCARBOXYLATE TRANSPORTER; MONOCARBOXYLATE TRANSPORTER 1; MONOCARBOXYLATE TRANSPORTER 2; MONOCARBOXYLATE TRANSPORTER 4; PYRUVIC ACID; S 0859; SULFONAMIDE; UNCLASSIFIED DRUG; BENZAMIDE DERIVATIVE; BICARBONATE SODIUM COTRANSPORTER; ISOPROTEIN; S 0859 COMPOUND;

ANIMAL CELL; ANION TRANSPORT; ARTICLE; ASTROCYTE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG MECHANISM; FEMALE; HETEROLOGOUS EXPRESSION; IC50; INHIBITION KINETICS; MOUSE; NEWBORN; NONHUMAN; OOCYTE; PRIORITY JOURNAL; PROTEIN FUNCTION; TRANSPORT KINETICS; XENOPUS LAEVIS; ANIMAL; ANTAGONISTS AND INHIBITORS; DRUG EFFECTS; HUMAN; METABOLISM; RAT; TRANSPORT AT THE CELLULAR LEVEL; XENOPUS;

ANIMALS; ASTROCYTES; BENZAMIDES; BIOLOGICAL TRANSPORT; HUMANS; INHIBITORY CONCENTRATION 50; LACTIC ACID; MICE; MONOCARBOXYLIC ACID TRANSPORTERS; PROTEIN ISOFORMS; RATS; SODIUM-BICARBONATE SYMPORTERS; SULFONAMIDES; XENOPUS;

EID: 84935886126     PISSN: 00142999     EISSN: 18790712     Source Type: Journal    
DOI: 10.1016/j.ejphar.2015.05.049     Document Type: Article

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