메뉴 건너뛰기




Volumn 7, Issue 1, 2015, Pages 82-93

Techniques used to enhance bioavailability of bcs class II drugs: A review

Author keywords

Amorphous state; Characterization; Dissolution enhancement; NCE

Indexed keywords

POLYMER; PRODRUG; SOLVENT; SURFACTANT;

EID: 84929074633     PISSN: None     EISSN: 09759344     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (14)

References (39)
  • 2
    • 1142309798 scopus 로고    scopus 로고
    • Rapid dissolving high potency danazol powders produced by spray freezing into liquid process
    • 2) Hu, J., Johnston, K.P., WilliamsIII, R.O., 2004. Rapid dissolving high potency danazol powders produced by spray freezing into liquid process, Int. J. Pharm. 271, 145–154.
    • (2004) Int. J. Pharm. , vol.271 , pp. 145-154
    • Hu, J.1    Johnston, K.P.2    Williams, R.O.3
  • 3
    • 0036742053 scopus 로고    scopus 로고
    • Poor aqueous solubility– an industry wide problem in drug delivery
    • Lipinski, C., 2002. Poor aqueous solubility– an industry wide problem in drug delivery, Am. Pharm. Rev. 5, 82–85.
    • (2002) Am. Pharm. Rev , vol.5 , pp. 82-85
    • Lipinski, C.1
  • 5
    • 85056065435 scopus 로고    scopus 로고
    • Bioavailability and bioequivalence testing. In: Remington: The science and practice of pharmacy
    • Gennaro AR, editor
    • Malinowski, H.J., Bioavailability and bioequivalence testing. In: Remington: The Science and Practice of Pharmacy. In: Gennaro AR, editor. 20th ed Philadelphia: Lippincott Williams Wilkinson, 2000; 995-1004.
    • (2000) 20Th Ed Philadelphia: Lippincott Williams Wilkinson , pp. 995-1004
    • Malinowski, H.J.1
  • 6
    • 0034601240 scopus 로고    scopus 로고
    • Improving drug solubility for oral delivery using solid dispersions
    • Leuner, C., Dressman, J., 2000. Improving drug solubility for oral delivery using solid dispersions. Eur. J. Pharm. Biopharm. 50, 47–60.
    • (2000) Eur. J. Pharm. Biopharm , vol.50 , pp. 47-60
    • Leuner, C.1    Dressman, J.2
  • 7
    • 0028948839 scopus 로고
    • A theoretical basis for a biopharmaceutical drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability
    • Amidon, G.L., Lenneranas, H., Shah, V.P., Crison J.R., 1995. A theoretical basis for a biopharmaceutical drug classification: The correlation of in vitro drug product dissolution and in vivo bioavailability. J. Pharm. Res. 12(3), 413-420.
    • (1995) J. Pharm. Res , vol.12 , Issue.3 , pp. 413-420
    • Amidon, G.L.1    Lenneranas, H.2    Shah, V.P.3    Crison, J.R.4
  • 10
    • 34248535178 scopus 로고    scopus 로고
    • Studies on dissolution enhancement and mathematical modeling of drug release of a poorly water-soluble drug using water-soluble carriers
    • Ahuja, N., Katare, O.P., Singh, B., 2007. Studies on dissolution enhancement and mathematical modeling of drug release of a poorly water-soluble drug using water-soluble carriers. Eur. J. Pharm. Biopharm. 65, 26-38.
    • (2007) Eur. J. Pharm. Biopharm , vol.65 , pp. 26-38
    • Ahuja, N.1    Katare, O.P.2    Singh, B.3
  • 12
    • 78649556396 scopus 로고    scopus 로고
    • Solubility and dissolution enhancement: An overview
    • Babu, V.R., Areefulla, S.H., Mallikarjun, V., 2010. Solubility and Dissolution Enhancement: An overview. J Pharm Research 3(1),141- 145.
    • (2010) J Pharm Research , vol.3 , Issue.1 , pp. 141-145
    • Babu, V.R.1    Areefulla, S.H.2    Mallikarjun, V.3
  • 13
    • 0025930844 scopus 로고
    • Solubilization and wetting effects of bile salts on the dissolution of steroids
    • Bakatselou, V., Oppenheim, R.C., Dressman, J.B., 1991. Solubilization and wetting effects of bile salts on the dissolution of steroids. Pharm Res. 8, 1461-1469.
    • (1991) Pharm Res , vol.8 , pp. 1461-1469
    • Bakatselou, V.1    Oppenheim, R.C.2    Dressman, J.B.3
  • 14
    • 27744575591 scopus 로고    scopus 로고
    • Cyclodextrins in drug delivery: An updated review
    • Challa, R., Ahuja, A., Ali, J., Khar, R.K., 2005. Cyclodextrins in Drug Delivery: An Updated Review. AAPS PharmSciTech. 6 (2), 29-57.
    • (2005) AAPS Pharmscitech , vol.6 , Issue.2 , pp. 29-57
    • Challa, R.1    Ahuja, A.2    Ali, J.3    Khar, R.K.4
  • 15
    • 77950362700 scopus 로고    scopus 로고
    • Dissolution enhancement of gliclazide using ph change approach in presence of twelve stabilizers with various physico-chemical properties
    • Talari, R., Varshosaz, J., Mostafavi, S.A., Nokhodchi, A., 2009. Dissolution Enhancement of Gliclazide Using pH Change Approach in Presence of Twelve Stabilizers with Various Physico-Chemical Properties. J Pharm Pharmaceut Sci. 12(3), 250 – 265.
    • (2009) J Pharm Pharmaceut Sci , vol.12 , Issue.3 , pp. 250-265
    • Talari, R.1    Varshosaz, J.2    Mostafavi, S.A.3    Nokhodchi, A.4
  • 17
    • 0016252489 scopus 로고
    • Prodrug approach to enhancement of rate of dissolution of allopurinol
    • Hussain, A., Rytting, J.H., 1974, Prodrug approach to enhancement of rate of dissolution of allopurinol. J Pharm Sci. 63 (5), 798–799.
    • (1974) J Pharm Sci , vol.63 , Issue.5 , pp. 798-799
    • Hussain, A.1    Rytting, J.H.2
  • 18
    • 17444400021 scopus 로고    scopus 로고
    • Comparison of powder produced by evaporative precipitation into aqueous solution (epas) and spray freezing into liquid (sfl) technologies using novel z-contrast stem and complimentary techniques
    • Vaughn, J.M., Gao, X., Yacaman, M.J., Johnston, K.P., Williams, R.O., 2005. Comparison of powder produced by evaporative precipitation into aqueous solution (EPAS) and spray freezing into liquid (SFL) technologies using novel Z-contrast STEM and complimentary techniques. Eur J Pharm Biopharm. 60(1), 81-89.
    • (2005) Eur J Pharm Biopharm , vol.60 , Issue.1 , pp. 81-89
    • Vaughn, J.M.1    Gao, X.2    Yacaman, M.J.3    Johnston, K.P.4    Williams, R.O.5
  • 19
    • 0026793126 scopus 로고
    • Powdered solution technology: Principles and mechanism
    • Spireas, S., Jarowski, C.I., Rohera, D.I., 1992. Powdered solution technology: principles and mechanism. Pharm Res. 9, 1351-1368.
    • (1992) Pharm Res , vol.9 , pp. 1351-1368
    • Spireas, S.1    Jarowski, C.I.2    Rohera, D.I.3
  • 20
  • 21
    • 27444438012 scopus 로고    scopus 로고
    • The effect of type and concentration of vehicles on the dissolution rate of a poorly soluble drug (indomethacin) from liquisolid compacts
    • Nokhodchi, A., Javadzadeh, Y., Siahi- Shadbad, M.R., Barzegar-Jalali, M., 2005. The effect of type and concentration of vehicles on the dissolution rate of a poorly soluble drug (indomethacin) from liquisolid compacts. J Pharm Pharm Sci. 8,18- 25.
    • (2005) J Pharm Pharm Sci , vol.8 , pp. 18-25
    • Nokhodchi, A.1    Javadzadeh, Y.2    Siahi- Shadbad, M.R.3    Barzegar-Jalali, M.4
  • 22
    • 0036804726 scopus 로고    scopus 로고
    • Factors affecting incorporation of drug into solid solution with hpmcp during solvent change coprecipitation
    • Sertsou, G., Butler, J., Scott, A., Hempenstall, J., Rades, T., 2002. Factors affecting incorporation of drug into solid solution with HPMCP during solvent change coprecipitation. Int J Pharm. 245, 99-108.
    • (2002) Int J Pharm , vol.245 , pp. 99-108
    • Sertsou, G.1    Butler, J.2    Scott, A.3    Hempenstall, J.4    Rades, T.5
  • 23
    • 0028200490 scopus 로고
    • Hydrosols - Alternatives for the parenteral application of poorly water soluble drugs
    • Gabmann, P., List, M., Schweitzer, A., Sucker, H., 1994. Hydrosols - Alternatives for the parenteral application of poorly water soluble drugs. Eur. J. Pharm. Biopharm. 40, 64–72.
    • (1994) Eur. J. Pharm. Biopharm , vol.40 , pp. 64-72
    • Gabmann, P.1    List, M.2    Schweitzer, A.3    Sucker, H.4
  • 24
    • 2042502059 scopus 로고    scopus 로고
    • High pressure process technology: Fundamentals and applications. Industrial chemistry library, elsevier
    • Bertucco, A., Vetter, G., 2001. High Pressure Process Technology: Fundamentals and Applications. Industrial Chemistry Library, Elsevier, Amsterdam. 9, 1-3.
    • (2001) Amsterdam , vol.9 , pp. 1-3
    • Bertucco, A.1    Vetter, G.2
  • 25
    • 77953415731 scopus 로고    scopus 로고
    • Novel drug delivery technologies for insoluble drugs
    • Chowdary, K.P.R., Madhavi, B.L.R., 2005. Novel drug delivery technologies for insoluble drugs. Indian Drugs. 42(9), 557-564.
    • (2005) Indian Drugs , vol.42 , Issue.9 , pp. 557-564
    • Chowdary, K.P.R.1    Madhavi, B.L.R.2
  • 26
    • 0033805858 scopus 로고    scopus 로고
    • Lipid formulations for oral administration of drugs: Nonemulsifying, self emulsifying and ‘self-microemulsifying’ drug delivery systems
    • Pouton, W.C., 2000. Lipid formulations for oral administration of drugs: nonemulsifying, self emulsifying and ‘self-microemulsifying’ drug delivery systems. Eur. J. Pharm. Sci. 11(2), S93– S98.
    • (2000) Eur. J. Pharm. Sci , vol.11 , Issue.2 , pp. S93-S98
    • Pouton, W.C.1
  • 27
    • 0035984949 scopus 로고    scopus 로고
    • Lipid based formulations for intestinal lymphatic delivery
    • O'Driscoll, C. M., 2002. Lipid based formulations for intestinal lymphatic delivery, Eur. J. Pharm. Sci. 15, 405– 415.
    • (2002) Eur. J. Pharm. Sci , vol.15 , pp. 405-415
    • O'driscoll, C.M.1
  • 28
    • 0033812424 scopus 로고    scopus 로고
    • Lipids, lipophilic drugs, and oral drug delivery—some emerging concepts
    • Charman, W.N., 2000. Lipids, lipophilic drugs, and oral drug delivery—some emerging concepts. J. Pharm. Sci. 89, 967–978.
    • (2000) J. Pharm. Sci , vol.89 , pp. 967-978
    • Charman, W.N.1
  • 29
    • 33847394968 scopus 로고    scopus 로고
    • Lipids and lipid-based formulations: Optimizing the oral delivery of lipophilic drugs, nature
    • Porter, C.J.H., Trevaskis, N.L., Charman, W.N., 2007. Lipids and lipid-based formulations: optimizing the oral delivery of lipophilic drugs, Nature Rev. Drug Disc. 6, 231–248.
    • (2007) Rev. Drug Disc , vol.6 , pp. 231-248
    • Porter, C.J.H.1    Trevaskis, N.L.2    Charman, W.N.3
  • 31
    • 0015124656 scopus 로고
    • Pharmaceutical applications of solid dispersion systems
    • Chiou, W.L., Riegelman, S., 1971. Pharmaceutical applications of solid dispersion systems. J. Pharm. Sci. 60(9), 1281-1302.
    • (1971) J. Pharm. Sci , vol.60 , Issue.9 , pp. 1281-1302
    • Chiou, W.L.1    Riegelman, S.2
  • 33
    • 1842865536 scopus 로고    scopus 로고
    • Melt extrusion: From process to drug delivery technology
    • Breitenbach, J., 2000. Melt extrusion: from process to drug delivery technology. Eur J Pharm Biopharm. 54 (2), 107 - 117.
    • (2000) Eur J Pharm Biopharm , vol.54 , Issue.2 , pp. 107-- 117
    • Breitenbach, J.1
  • 34
  • 35
    • 0013795160 scopus 로고
    • Increasing dissolution rates and gastrointestinal absorption of drugs via solid solutions and eutectic mixtures. I. Theoretical considerations and discussion of the literature
    • Goldberg, A.H., Gibaldi, M., Kanig, J.L., 1965. Increasing dissolution rates and gastrointestinal absorption of drugs via solid solutions and eutectic mixtures. I. Theoretical considerations and discussion of the literature. J. Pharm. Sci. 54(8), 1145-1148.
    • (1965) J. Pharm. Sci , vol.54 , Issue.8 , pp. 1145-1148
    • Goldberg, A.H.1    Gibaldi, M.2    Kanig, J.L.3
  • 36
    • 0003785744 scopus 로고
    • Solid-liquid equilibria in solutions of non-electrolytes
    • Rastogi, R.P., Rama Varma, K.T., 1956. Solid-liquid equilibria in solutions of non-electrolytes. J. Chem.Soc. 2, 2097-2101.
    • (1956) J. Chem.Soc. , vol.2 , pp. 2097-2101
    • Rastogi, R.P.1    Rama Varma, K.T.2
  • 37
    • 0014515660 scopus 로고
    • Dissolution rates of high energy polyvinylpyrrolidone (pvp)- sulfathiazole coprecipitates
    • Simonelli, A.P., Mehta, S.C., Higuchi, W.I., 1969. Dissolution rates of high energy polyvinylpyrrolidone (PVP)- sulfathiazole coprecipitates. J. Pharm. Sci. 58(5), 538-549.
    • (1969) J. Pharm. Sci , vol.58 , Issue.5 , pp. 538-549
    • Simonelli, A.P.1    Mehta, S.C.2    Higuchi, W.I.3
  • 38
    • 84984082270 scopus 로고
    • Increasing dissolution rates and gastrointestinal absorption of drugs via solid solutions and eutectic mixtures ii experimental evaluation of a eutectic mixture: Urea-acetaminophen system
    • Goldberg, A.H., Gibaldi, M., Kanig, L., 1966. Increasing dissolution rates and gastrointestinal absorption of drugs via solid solutions and eutectic mixtures II experimental evaluation of a eutectic mixture: urea-acetaminophen system. J. Pharm. Sci. 55, 482-487.
    • (1966) J. Pharm. Sci , vol.55 , pp. 482-487
    • Goldberg, A.H.1    Gibaldi, M.2    Kanig, L.3
  • 39
    • 0014628768 scopus 로고
    • Preparation and dissolution characteristics of several fast-release solid dispersions of griseofulvin
    • Chiou, W.L., Riegelman, S., 1969. Preparation and dissolution characteristics of several fast-release solid dispersions of griseofulvin. J. Pharm. Sci. 1505-1510.
    • (1969) J. Pharm. Sci , pp. 1505-1510
    • Chiou, W.L.1    Riegelman, S.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.