Screening for small molecule disruptors of AKAP-PKA interactions

Methods in Molecular Biology

Volumn 1294, Issue , 2015, Pages 151-166

  Schächterle, Carolin ^a   Christian, Frank ^a   Fernandes, João Miguel Parente ^a   Klussmann, Enno ^a  

^a NONE

Author keywords

A kinase anchoring protein (AKAP); Enzyme linked immunosorbent assay (ELISA); Homogenous time resolved fluorescence (HTRF) assay; Inhibitory peptides; Nonpeptidic helix mimetics; Protein kinase A (PKA); Small molecules

Indexed keywords

CYCLIC AMP DEPENDENT PROTEIN KINASE; CYCLIC AMP DEPENDENT PROTEIN KINASE ANCHORING PROTEIN; PROTEIN INHIBITOR; MOLECULAR LIBRARY; PROTEIN BINDING;

ARTICLE; ENZYME ACTIVITY; ENZYME INHIBITION; ENZYME LINKED IMMUNOSORBENT ASSAY; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN PROTEIN INTERACTION; CHEMISTRY; DRUG EFFECTS; FLUORESCENCE; METABOLISM; MOLECULAR LIBRARY; PHARMACOLOGY; PROCEDURES; SIGNAL TRANSDUCTION;

A KINASE ANCHOR PROTEINS; CYCLIC AMP-DEPENDENT PROTEIN KINASES; ENZYME-LINKED IMMUNOSORBENT ASSAY; FLUORESCENCE; PROTEIN BINDING; SIGNAL TRANSDUCTION; SMALL MOLECULE LIBRARIES;

EID: 84925321321     PISSN: 10643745     EISSN: None     Source Type: Book Series    
DOI: 10.1007/978-1-4939-2537-7_12     Document Type: Article

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