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Bioorganic and Medicinal Chemistry Letters

Volumn 25, Issue 3, 2015, Pages 616-620

Discovery of O-(3-carbamimidoylphenyl)-l-serine amides as matriptase inhibitors using a fragment-linking approach

(11) Goswami, Rajeev a Wohlfahrt, Gerd b Mukherjee, Subhendu a Ghadiyaram, Chakshusmathi a Nagaraj, Jwala a Satyam, Leena K a Subbarao, Krishnaprasad a Gopinath, Sreevalsam a Krishnamurthy, Narasimha R a Subramanya, Hosahalli S a Ramachandra, Murali a

a Aurigene Discovery Technologies Limited (India)

b ORION CORPORATION (Finland)

Author keywords

Anti tumor; Crystallography; Fragment linking approach; Matriptase; Molecular docking

Indexed keywords

AMIDE; MATRIPTASE; NAPHTHYL GROUP; SERINE DERIVATIVE; SERINE PROTEINASE INHIBITOR; PROTEIN BINDING; SERINE; SERINE PROTEINASE;

ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; CONTROLLED STUDY; CRYSTAL STRUCTURE; ENZYME ACTIVE SITE; GROWTH INHIBITION; MALE; MOUSE; NONHUMAN; PRIMARY TUMOR; PROSTATE CANCER; PROTEIN EXPRESSION; ANIMAL; BINDING SITE; CHEMISTRY; HALF LIFE TIME; KINETICS; METABOLISM; MOLECULAR DOCKING; STRUCTURE ACTIVITY RELATION; SYNTHESIS; X RAY CRYSTALLOGRAPHY;

AMIDES; ANIMALS; BINDING SITES; CATALYTIC DOMAIN; CRYSTALLOGRAPHY, X-RAY; HALF-LIFE; KINETICS; MALE; MICE; MOLECULAR DOCKING SIMULATION; PROTEIN BINDING; SERINE; SERINE ENDOPEPTIDASES; SERINE PROTEINASE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84920720980 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2014.12.008 Document Type: Article

Times cited : (10)

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