Evaluation of thermosensitive poloxamer 407 gel systems for the sustained release of estradiol in a fish model

European Journal of Pharmaceutics and Biopharmaceutics

Volumn 88, Issue 3, 2014, Pages 954-961

  Cespi, Marco ^a   Bonacucina, Giulia ^a   Pucciarelli, Stefania ^a   Cocci, Paolo ^a   Perinelli, Diego Romano ^a   Casettari, Luca ^b   Illum, Lisbeth ^c   Palmieri, Giovanni Filippo ^a   Palermo, Francesco Alessandro ^a   Mosconi, Gilberto ^a  

^a UNIVERSITY OF CAMERINO   (Italy)

^b UNIVERSITY OF URBINO   (Italy)

^c University of Camerino Unità Ricerca e Didattica San Benedetto Del Tronto ^*  (United Kingdom)

Author keywords

17b Estradiol; Goldfish; Poloxamer; Sustained release; Thermosensitive gel; Vitellogenin

Indexed keywords

CORN OIL; ESTRADIOL; ESTROGEN RECEPTOR; POLOXAMER; VITELLOGENIN; DELAYED RELEASE FORMULATION; GEL;

ANIMAL EXPERIMENT; AREA UNDER THE CURVE; ARTICLE; BLOOD RHEOLOGY; CONTROL SYSTEM; CONTROLLED STUDY; DISPERSION; DRUG BIOAVAILABILITY; DRUG BLOOD LEVEL; DRUG DELIVERY SYSTEM; DRUG FORMULATION; DRUG HALF LIFE; ENZYME LINKED IMMUNOSORBENT ASSAY; ESTRADIOL BLOOD LEVEL; FEMALE; GEL; GOLDFISH; HEAT SENSITIVITY; IN VITRO STUDY; LIVER CLEARANCE; MALE; MAXIMUM PLASMA CONCENTRATION; MICELLIZATION; NONHUMAN; SEXUAL DEVELOPMENT; SILICONE PROSTHESIS; SUSTAINED DRUG RELEASE; TIME TO MAXIMUM PLASMA CONCENTRATION; VISCOMETRY; VISCOSITY; VITELLOGENESIS; WATER TEMPERATURE; ADMINISTRATION AND DOSAGE; ANIMAL; ANIMAL MODEL; BLOOD; CHEMISTRY; DELAYED RELEASE FORMULATION; DRUG SCREENING; MEDICINAL CHEMISTRY; METABOLISM; PROCEDURES; SYNTHESIS; TEMPERATURE;

ANIMALS; CHEMISTRY, PHARMACEUTICAL; DELAYED-ACTION PREPARATIONS; DRUG EVALUATION, PRECLINICAL; ESTRADIOL; GELS; GOLDFISH; MODELS, ANIMAL; POLOXAMER; TEMPERATURE;

EID: 84912127698     PISSN: 09396411     EISSN: 18733441     Source Type: Journal    
DOI: 10.1016/j.ejpb.2014.08.008     Document Type: Article

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