Study the interactions between human serum albumin and two antifungal drugs: Fluconazole and its analogue DTP

Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 21, 2014, Pages 4963-4968

  Zhang, Shao Lin ^a   Yao, Huankai ^a,b   Wang, Chenyin ^a   Tam, Kin Y ^a  

^a University of Macau   (Macao)

^b XUZHOU MEDICAL UNIVERSITY   (China)

Author keywords

Binding affinity; Fluconazole; Fluorescence spectrum; Human serum albumin; Molecular docking

Indexed keywords

2 (2,4 DICHLOROPHENYL) 1,3 DI(1H 1,2,4 TRIAZOL YL) 2 PROPANOL; ANTIFUNGAL AGENT; ARGININE; FLUCONAZOLE; HUMAN SERUM ALBUMIN; LYSINE; MAGNESIUM ION; METAL ION; UNCLASSIFIED DRUG; ZINC ION; DICHLOROPHENYL-BIS-TRIAZOLYLPROPANOL; PROTEIN BINDING; SERUM ALBUMIN; TRIAZOLE DERIVATIVE;

ARTICLE; BINDING AFFINITY; CIRCULATION; COMPLEX FORMATION; DRUG HALF LIFE; DRUG PROTEIN BINDING; DRUG STRUCTURE; ENTHALPY; ENTROPY; HALF LIFE TIME; HYDROGEN BOND; HYDROPHOBICITY; MOLECULAR DOCKING; MOLECULAR MODEL; THERMODYNAMICS; BINDING SITE; CHEMICAL PHENOMENA; CHEMICAL STRUCTURE; CIRCULAR DICHROISM; HUMAN; METABOLISM; PROTEIN CONFORMATION; SPECTROFLUOROMETRY;

ANTIFUNGAL AGENTS; BINDING SITES; CIRCULAR DICHROISM; FLUCONAZOLE; HUMANS; HYDROGEN BONDING; HYDROPHOBIC AND HYDROPHILIC INTERACTIONS; MODELS, MOLECULAR; PROTEIN BINDING; PROTEIN CONFORMATION; SERUM ALBUMIN; SPECTROMETRY, FLUORESCENCE; THERMODYNAMICS; TRIAZOLES;

EID: 84907980878     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2014.09.034     Document Type: Article

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