Characterizations of plasticized polymeric film coatings for preparing multiple-unit floating drug delivery systems (muFDDSs) with controlled-release characteristics

PLoS ONE

Volumn 9, Issue 6, 2014, Pages

  Hung, Sheng Feng ^a   Hsieh, Chien Ming ^a,c   Chen, Ying Chen ^a   Wang, Yu Chun ^a   Ho, Hsiu O ^a   Sheu, Ming Thau ^a,b  

^a TAIPEI MEDICAL UNIVERSITY   (Taiwan)

^b TAIPEI MEDICAL UNIVERSITY HOSPITAL   (Taiwan)

^c PROVIDENCE UNIVERSITY   (Taiwan)

Author keywords

[No Author keywords available]

Indexed keywords

ACRYLIC ACID; BICARBONATE; CITRIC ACID TRIETHYL ESTER; ETHYL CELLULOSE; EUDRAGIT; EUDRAGIT RS; LOSARTAN; PHTHALIC ACID DIETHYL ESTER; WATER; ARTIFICIAL MEMBRANE; CELLULOSE; DELAYED RELEASE FORMULATION; DRUG CARRIER; PLASTIC;

AQUEOUS SOLUTION; ARTICLE; CHEMICAL ANALYSIS; CONTROLLED RELEASE FORMULATION; CONTROLLED STUDY; DRUG DELIVERY SYSTEM; DRUG PELLET; DRUG SOLUBILITY; EFFERVESCENT TABLET; FILM COATING; MECHANICAL STRESS; MULTIPLE UNIT FLOATING DRUG DELIVERY SYSTEM; PHYSICAL PARAMETERS; STRESS STRAIN RELATIONSHIP; SUSTAINED DRUG RELEASE; TOUGHNESS; YOUNG MODULUS; ANALOGS AND DERIVATIVES; ARTIFICIAL MEMBRANE; CHEMISTRY; DELAYED RELEASE FORMULATION;

CELLULOSE; DELAYED-ACTION PREPARATIONS; DRUG CARRIERS; LOSARTAN; MEMBRANES, ARTIFICIAL; PLASTICS; SODIUM BICARBONATE; STRESS, MECHANICAL;

EID: 84903398926     PISSN: None     EISSN: 19326203     Source Type: Journal    
DOI: 10.1371/journal.pone.0100321     Document Type: Article

References (29)

1. Pawar VK, Kansal S, Garg G, Awasthi R, Singodia D, et al. (2011) Gastroretentive dosage forms: a review with special emphasis on floating drug delivery systems. Drug delivery 18: 97-110.
2. Waterman KC (2007) A critical review of gastric retentive controlled drug delivery. Pharmaceutical development and technology 12: 1-10.
3. Singh BN, Kim KH (2000) Floating drug delivery systems: An approach to oral controlled drug delivery via gastric retention. J Controlled Release 63: 235-259.
4. Rouge N, Buri P, Doelker E (1996) Drug absorption sites in the gastrointestinal tract and dosage forms for site-specific delivery. Int J Pharm 136: 117-139. (Pubitemid 26199405)
5. Sato Y, Kawashima Y, Takeuchi H, Yamamoto H (2004) In vitro and in vivo evaluation of riboflavin-containing microballoons for a floating controlled drug delivery system in healthy humans. Int J Pharm 275: 97-107. (Pubitemid 38481523)
6. Umamaheshwari RB, Jain S, Bhadra D, Jain NK (2003) Floating microspheres bearing acetohydroxamic acid for the treatment of Helicobacter pylori. J Pharm Pharmacol 55: 1607-1613. (Pubitemid 38054390)
7. Bardonnet PL, Faivre V, Pugh WJ, Piffaretti JC, Falson F (2006) Gastroretentive dosage forms: Overview and special case of Helicobacter pylori. J Controlled Release 111: 1-18. (Pubitemid 43289989)
8. Yang L, Eshraghi J, Fassihi R (1999) A new intragastric delivery system for the treatment of Helicobacter pylori associated gastric ulcer: In vitro evaluation. J Controlled Release 57: 215-222. (Pubitemid 29073437)
9. Seta Y, Higuchi F, Kawahara Y, Nishimura K, Okada R (1988) Design and preparation of captopril sustained-release dosage forms and their biopharmaceutical properties. Int J Pharm 41: 245-254. (Pubitemid 18034878)
10. Jain SK, Awasthi AM, Jain NK, Agrawal GP (2005) Calcium silicate based microspheres of repaglinide for gastroretentive floating drug delivery: Preparation and in vitro characterization. J Controlled Release 107: 300-309. (Pubitemid 41316292)
11. Wurster DE, Alkhamis KA, Matheson LE (2003) Prediction of the adsorption of diazepam by activated carbon in aqueous media. J Pharm Sci 92: 2008-2016. (Pubitemid 37175631)
12. Munday DL (2003) Film coated pellets containing verapamil hydrochloride: Enhanced dissolution into neutral medium. Drug Dev Ind Pharm 29: 575-583.
13. Prajapati VD, Jani GK, Khutliwala TA, Zala BS (2013) Raft forming system-an upcoming approach of gastroretentive drug delivery system. Journal of controlled release : official journal of the Controlled Release Society 168: 151-165.
14. Dixit N (2011) Floating Drug Delivery System. Journal of Current Pharmaceutical Research 7: 6-20.
15. Sungthongjeen S, Sriamornsak P, Puttipipatkhachorn S (2008) Design and evaluation of floating multi-layer coated tablets based on gas formation. Eur J Pharm Biopharm 69: 255-263. (Pubitemid 351467157)
16. Ichikawa M, Watanabe S, Miyake Y (1991) A new multiple-unit oral floating dosage system. I: Preparation and in vitro evaluation of floating and sustained-release characteristics. J Pharm Sci 80: 1062-1066.
17. Kawashima Y, Niwa T, Takeuchi H, Hino T, Ito Y (1991) Preparation of multiple unit hollow microspheres (microballoons) with acrylic resin containing tranilast and their drug release characteristics (in vitro) and floating behavior (in vivo). J Controlled Release 16: 279-289.
18. Streubel A, Siepmann J, Bodmeier R (2003) Multiple unit gastroretentive drug delivery systems: A new preparation method for low density microparticles. J Microencapsul 20: 329-347. (Pubitemid 36621475)
19. Talukder R, Fassihi R (2004) Gastroretentive delivery systems: Hollow beads. Drug Dev Ind Pharm 30: 405-412. (Pubitemid 38987183)
20. Bechgaard H, Ladefoged K (1978) Distribution of pellets in the gastrointestinal tract. The influence on transit time exerted by the density or diameter of pellets. J Pharm Pharmacol 30: 690-692. (Pubitemid 9063329)
21. Chen YC, Lee LW, Ho HO, Sha C, Sheu MT (2012) Evaluation of water uptake and mechanical properties of blended polymer films for preparing gas-generated multiple-unit floating drug delivery systems. Journal of pharmaceutical sciences 101: 3811-3822.
22. Iannuccelli V, Coppi G, Bernabei MT, Cameroni R (1998) Air compartment multiple-unit system for prolonged gastric residence. Part I. Formulation study. Int J Pharm 174: 47-54. (Pubitemid 28486988)
23. Krögel I, Bodmeier R (1999) Floating or pulsatile drug delivery systems based on coated effervescent cores. Int J Pharm 187: 175-184. (Pubitemid 29443897)
24. Sica DA, Gehr TWB, Ghosh S (2005) Clinical pharmacokinetics of losartan. Clin Pharmacokinet 44: 797-814. (Pubitemid 41126929)
25. Wu JS, Ho HO, Sheu MT (2001) A statistical design to evaluate the influence of manufacturing factors on the material properties and functionalities of microcrystalline cellulose. Eur J Pharm Sci 12: 417-425.
26. Kawano Y, Wang Y, Palmer RA, Aubuchon SR (2002) Stress-Strain Curves of Nafion Membranes in Acid and Salt Forms. Polímeros: Ciência e Tecnologia 12: 96-101.
27. Bi Y, Sunada H, Yonezawa Y, Danjo K, Otsuka A, et al. (1996) Preparation and evaluation of a compressed tablet rapidly disintegrating in the oral cavity. Chemical & pharmaceutical bulletin 44: 2121-2127. (Pubitemid 26396765)
28. Hamdani J, Moes AJ, Amighi K (2006) Development and in vitro evaluation of a novel floating multiple unit dosage form obtained by melt pelletization. International journal of pharmaceutics 322: 96-103. (Pubitemid 44339598)
29. Bodmeier R, Paeratakul O (1994) Mechanical properties of dry and wet cellulosic and acrylic films prepared from aqueous colloidal polymer dispersions used in the coating of solid dosage forms. Pharm Res 11: 882-888. (Pubitemid 24210626)