메뉴 건너뛰기




Volumn 101, Issue 10, 2012, Pages 3811-3822

Evaluation of water uptake and mechanical properties of blended polymer films for preparing gas-generated multiple-unit floating drug delivery systems

Author keywords

Dissolution rate; Effervescent; Floating ability; Formulation; Gastrointestinal transit; Mechanical properties; Permeability; Water uptake

Indexed keywords

BICARBONATE; CARBON DIOXIDE; ETHYL CELLULOSE; EUDRAGIT; EUDRAGIT RS; HYDROXYPROPYLMETHYLCELLULOSE; LOSARTAN POTASSIUM; MACROGOL 6000;

EID: 84865387514     PISSN: 00223549     EISSN: 15206017     Source Type: Journal    
DOI: 10.1002/jps.23279     Document Type: Article
Times cited : (8)

References (37)
  • 1
    • 33748430023 scopus 로고    scopus 로고
    • Drug delivery to the upper small intestine window using gastroretentive technologies
    • Streubel A, Siepmann J, Bodmeier R. 2006. Drug delivery to the upper small intestine window using gastroretentive technologies. Curr Opin Pharmacol 6(5):501-508.
    • (2006) Curr Opin Pharmacol , vol.6 , Issue.5 , pp. 501-508
    • Streubel, A.1    Siepmann, J.2    Bodmeier, R.3
  • 2
    • 77953393044 scopus 로고    scopus 로고
    • Gastroretentive drug delivery systems: A review
    • Nayak AK, Maji R, Das B. 2010. Gastroretentive drug delivery systems: A review. Asian J Pharm Clin Res 3(1):2-10.
    • (2010) Asian J Pharm Clin Res , vol.3 , Issue.1 , pp. 2-10
    • Nayak, A.K.1    Maji, R.2    Das, B.3
  • 3
    • 0032494197 scopus 로고    scopus 로고
    • Pharmacodynamic aspects of sustained release preparations
    • Hoffman A. 1998. Pharmacodynamic aspects of sustained release preparations. Adv Drug Deliv Rev 33(3):185-199.
    • (1998) Adv Drug Deliv Rev , vol.33 , Issue.3 , pp. 185-199
    • Hoffman, A.1
  • 4
    • 0029117539 scopus 로고
    • Optimization of sotalol floating and bioadhesive extended release tablet formulations
    • Chueh HR, Zia H, Rhodes CT. 1995. Optimization of sotalol floating and bioadhesive extended release tablet formulations. Drug Dev Ind Pharm 21(15):1725-1747.
    • (1995) Drug Dev Ind Pharm , vol.21 , Issue.15 , pp. 1725-1747
    • Chueh, H.R.1    Zia, H.2    Rhodes, C.T.3
  • 5
    • 0027180264 scopus 로고
    • A floating controlled-release drug delivery system: In vitro-in vivo evaluation
    • Desai S, Bolton S. 1993. A floating controlled-release drug delivery system: In vitro-in vivo evaluation. Pharm Res 10(9):1321-1325.
    • (1993) Pharm Res , vol.10 , Issue.9 , pp. 1321-1325
    • Desai, S.1    Bolton, S.2
  • 6
    • 2442714776 scopus 로고    scopus 로고
    • Pharmacokinetic and pharmacodynamic aspects of gastroretentive dosage forms
    • Hoffman A, Stepensky D, Lavy E, Eyal S, Klausner E, Friedman M. 2004. Pharmacokinetic and pharmacodynamic aspects of gastroretentive dosage forms. Int J Pharm 277(1-2):141-153.
    • (2004) Int J Pharm , vol.277 , Issue.1-2 , pp. 141-153
    • Hoffman, A.1    Stepensky, D.2    Lavy, E.3    Eyal, S.4    Klausner, E.5    Friedman, M.6
  • 7
    • 0033991593 scopus 로고    scopus 로고
    • Floating drug delivery systems: An approach to oral controlled drug delivery via gastric retention
    • Singh BN, Kim KH. 2000. Floating drug delivery systems: An approach to oral controlled drug delivery via gastric retention. J Control Release 63(3):235-259.
    • (2000) J Control Release , vol.63 , Issue.3 , pp. 235-259
    • Singh, B.N.1    Kim, K.H.2
  • 8
    • 0029953050 scopus 로고    scopus 로고
    • Drug absorption sites in the gastrointestinal tract and dosage forms for site-specific delivery
    • Rouge N, Buri P, Doelker E. 1996. Drug absorption sites in the gastrointestinal tract and dosage forms for site-specific delivery. Int J Pharm 136(1-2):117-139.
    • (1996) Int J Pharm , vol.136 , Issue.1-2 , pp. 117-139
    • Rouge, N.1    Buri, P.2    Doelker, E.3
  • 9
    • 1842689006 scopus 로고    scopus 로고
    • In vitro and in vivo evaluation of riboflavin-containing microballoons for a floating controlled drug delivery system in healthy humans
    • Sato Y, Kawashima Y, Takeuchi H, Yamamoto H. 2004. In vitro and in vivo evaluation of riboflavin-containing microballoons for a floating controlled drug delivery system in healthy humans. Int J Pharm 275(1-2):97-107.
    • (2004) Int J Pharm , vol.275 , Issue.1-2 , pp. 97-107
    • Sato, Y.1    Kawashima, Y.2    Takeuchi, H.3    Yamamoto, H.4
  • 10
    • 0347359072 scopus 로고    scopus 로고
    • Floating microspheres bearing acetohydroxamic acid for the treatment of Helicobacter pylori
    • Umamaheshwari RB, Jain S, Bhadra D, Jain NK. 2003. Floating microspheres bearing acetohydroxamic acid for the treatment of Helicobacter pylori. J Pharm Pharmacol 55(12):1607-1613.
    • (2003) J Pharm Pharmacol , vol.55 , Issue.12 , pp. 1607-1613
    • Umamaheshwari, R.B.1    Jain, S.2    Bhadra, D.3    Jain, N.K.4
  • 11
  • 12
    • 0033046507 scopus 로고    scopus 로고
    • A new intragastric delivery system for the treatment of Helicobacter pylori associated gastric ulcer: In vitro evaluation
    • Yang L, Eshraghi J, Fassihi R. 1999. A new intragastric delivery system for the treatment of Helicobacter pylori associated gastric ulcer: In vitro evaluation. J Control Release 57(3):215-222.
    • (1999) J Control Release , vol.57 , Issue.3 , pp. 215-222
    • Yang, L.1    Eshraghi, J.2    Fassihi, R.3
  • 13
    • 0023832711 scopus 로고
    • Design and preparation of captopril sustained-release dosage forms and their biopharmaceutical properties
    • Seta Y, Higuchi F, Kawahara Y, Nishimura K, Okada R. 1988. Design and preparation of captopril sustained-release dosage forms and their biopharmaceutical properties. Int J Pharm 41(3):245-254.
    • (1988) Int J Pharm , vol.41 , Issue.3 , pp. 245-254
    • Seta, Y.1    Higuchi, F.2    Kawahara, Y.3    Nishimura, K.4    Okada, R.5
  • 14
    • 24944474831 scopus 로고    scopus 로고
    • Calcium silicate based microspheres of repaglinide for gastroretentive floating drug delivery: Preparation and in vitro characterization
    • Jain SK, Awasthi AM, Jain NK, Agrawal GP. 2005. Calcium silicate based microspheres of repaglinide for gastroretentive floating drug delivery: Preparation and in vitro characterization. J Control Release 107(2):300-309.
    • (2005) J Control Release , vol.107 , Issue.2 , pp. 300-309
    • Jain, S.K.1    Awasthi, A.M.2    Jain, N.K.3    Agrawal, G.P.4
  • 15
    • 0141731264 scopus 로고    scopus 로고
    • Prediction of the adsorption of diazepam by activated carbon in aqueous media
    • Wurster DE, Alkhamis KA, Matheson LE. 2003. Prediction of the adsorption of diazepam by activated carbon in aqueous media. J Pharm Sci 92(10):2008-2016.
    • (2003) J Pharm Sci , vol.92 , Issue.10 , pp. 2008-2016
    • Wurster, D.E.1    Alkhamis, K.A.2    Matheson, L.E.3
  • 16
    • 0037908860 scopus 로고    scopus 로고
    • Film coated pellets containing verapamil hydrochloride: Enhanced dissolution into neutral medium
    • Munday DL. 2003. Film coated pellets containing verapamil hydrochloride: Enhanced dissolution into neutral medium. Drug Dev Ind Pharm 29(5):575-583.
    • (2003) Drug Dev Ind Pharm , vol.29 , Issue.5 , pp. 575-583
    • Munday, D.L.1
  • 18
    • 0031754109 scopus 로고    scopus 로고
    • Floating dosage forms: An in vivo study demonstrating prolonged gastric retention
    • Whitehead L, Fell JT, Collett JH, Sharma HL, Smith AM. 1998. Floating dosage forms: An in vivo study demonstrating prolonged gastric retention. J Control Release 55(1):3-12.
    • (1998) J Control Release , vol.55 , Issue.1 , pp. 3-12
    • Whitehead, L.1    Fell, J.T.2    Collett, J.H.3    Sharma, H.L.4    Smith, A.M.5
  • 21
    • 41549097189 scopus 로고    scopus 로고
    • Design and evaluation of floating multi-layer coated tablets based on gas formation
    • Sungthongjeen S, Sriamornsak P, Puttipipatkhachorn S. 2008. Design and evaluation of floating multi-layer coated tablets based on gas formation. Eur J Pharm Biopharm 69(1):255-263.
    • (2008) Eur J Pharm Biopharm , vol.69 , Issue.1 , pp. 255-263
    • Sungthongjeen, S.1    Sriamornsak, P.2    Puttipipatkhachorn, S.3
  • 22
    • 0025751561 scopus 로고
    • A new multiple-unit oral floating dosage system. I: Preparation and in vitro evaluation of floating and sustained-release characteristics
    • Ichikawa M, Watanabe S, Miyake Y. 1991. A new multiple-unit oral floating dosage system. I: Preparation and in vitro evaluation of floating and sustained-release characteristics. J Pharm Sci 80(11):1062-1066.
    • (1991) J Pharm Sci , vol.80 , Issue.11 , pp. 1062-1066
    • Ichikawa, M.1    Watanabe, S.2    Miyake, Y.3
  • 23
    • 0025799715 scopus 로고
    • Preparation of multiple unit hollow microspheres (microballoons) with acrylic resin containing tranilast and their drug release characteristics (in vitro) and floating behavior (in vivo)
    • Kawashima Y, Niwa T, Takeuchi H, Hino T, Ito Y. 1991. Preparation of multiple unit hollow microspheres (microballoons) with acrylic resin containing tranilast and their drug release characteristics (in vitro) and floating behavior (in vivo). J Control Release 16(3):279-289.
    • (1991) J Control Release , vol.16 , Issue.3 , pp. 279-289
    • Kawashima, Y.1    Niwa, T.2    Takeuchi, H.3    Hino, T.4    Ito, Y.5
  • 24
    • 0037769850 scopus 로고    scopus 로고
    • Multiple unit gastroretentive drug delivery systems: A new preparation method for low density microparticles
    • Streubel A, Siepmann J, Bodmeier R. 2003. Multiple unit gastroretentive drug delivery systems: A new preparation method for low density microparticles. J Microencapsul 20(3):329-347.
    • (2003) J Microencapsul , vol.20 , Issue.3 , pp. 329-347
    • Streubel, A.1    Siepmann, J.2    Bodmeier, R.3
  • 25
    • 3343013285 scopus 로고    scopus 로고
    • Gastroretentive delivery systems: Hollow beads
    • Talukder R, Fassihi R. 2004. Gastroretentive delivery systems: Hollow beads. Drug Dev Ind Pharm 30(4):405-412.
    • (2004) Drug Dev Ind Pharm , vol.30 , Issue.4 , pp. 405-412
    • Talukder, R.1    Fassihi, R.2
  • 26
    • 0018173224 scopus 로고
    • Distribution of pellets in the gastrointestinal tract. The influence on transit time exerted by the density or diameter of pellets
    • Bechgaard H, Ladefoged K. 1978. Distribution of pellets in the gastrointestinal tract. The influence on transit time exerted by the density or diameter of pellets. J Pharm Pharmacol 30(11):690-692.
    • (1978) J Pharm Pharmacol , vol.30 , Issue.11 , pp. 690-692
    • Bechgaard, H.1    Ladefoged, K.2
  • 27
    • 0031764619 scopus 로고    scopus 로고
    • Air compartment multiple-unit system for prolonged gastric residence. Part I. Formulation study
    • Iannuccelli V, Coppi G, Bernabei MT, Cameroni R. 1998. Air compartment multiple-unit system for prolonged gastric residence. Part I. Formulation study. Int J Pharm 174(1-2):47-54.
    • (1998) Int J Pharm , vol.174 , Issue.1-2 , pp. 47-54
    • Iannuccelli, V.1    Coppi, G.2    Bernabei, M.T.3    Cameroni, R.4
  • 28
    • 0345035517 scopus 로고    scopus 로고
    • Floating or pulsatile drug delivery systems based on coated effervescent cores
    • Krögel I, Bodmeier R. 1999. Floating or pulsatile drug delivery systems based on coated effervescent cores. Int J Pharm 187(2):175-184.
    • (1999) Int J Pharm , vol.187 , Issue.2 , pp. 175-184
    • Krögel, I.1    Bodmeier, R.2
  • 29
    • 23744484192 scopus 로고    scopus 로고
    • Clinical pharmacokinetics of losartan
    • Sica DA, Gehr TWB, Ghosh S. 2005. Clinical pharmacokinetics of losartan. Clin Pharmacokinet 44(8):797-814.
    • (2005) Clin Pharmacokinet , vol.44 , Issue.8 , pp. 797-814
    • Sica, D.A.1    Gehr, T.W.B.2    Ghosh, S.3
  • 30
    • 0035105840 scopus 로고    scopus 로고
    • A statistical design to evaluate the influence of manufacturing factors on the material properties and functionalities of microcrystalline cellulose
    • Wu JS, Ho HO, Sheu MT. 2001. A statistical design to evaluate the influence of manufacturing factors on the material properties and functionalities of microcrystalline cellulose. Eur J Pharm Sci 12(4):417-425.
    • (2001) Eur J Pharm Sci , vol.12 , Issue.4 , pp. 417-425
    • Wu, J.S.1    Ho, H.O.2    Sheu, M.T.3
  • 31
    • 85030491835 scopus 로고    scopus 로고
    • Handbook of basic pharmacokinetics
    • Ritschel WA, Kearns GL, Eds. 7th ed. Washington, DC: American Pharmacists Association
    • Ritschel WA, Kearns GL, Eds. 1999. Handbook of basic pharmacokinetics including clinical applications. 7th ed. Washington, DC: American Pharmacists Association, pp 92-105.
    • (1999) including clinical applications , pp. 92-105
  • 32
    • 0028245301 scopus 로고
    • Mechanical properties of dry and wet cellulosic and acrylic films prepared from aqueous colloidal polymer dispersions used in the coating of solid dosage forms
    • Bodmeier R, Paeratakul O. 1994. Mechanical properties of dry and wet cellulosic and acrylic films prepared from aqueous colloidal polymer dispersions used in the coating of solid dosage forms. Pharm Res 11(6):882-888.
    • (1994) Pharm Res , vol.11 , Issue.6 , pp. 882-888
    • Bodmeier, R.1    Paeratakul, O.2
  • 33
    • 0001003171 scopus 로고    scopus 로고
    • Eudragit aqueous dispersions as pharmaceutical controlled release coatings
    • Ghebre-Sellassie I, Nesbitt RU, Wang J. McGinity JW, Ed. 2nd ed. New York: Marcel Dekker
    • Ghebre-Sellassie I, Nesbitt RU, Wang J. 1997. Eudragit aqueous dispersions as pharmaceutical controlled release coatings. Aqueous polymeric coatings for pharmaceutical dosage forms; McGinity JW, Ed. 2nd ed. New York: Marcel Dekker, pp 267-286.
    • (1997) Aqueous polymeric coatings for pharmaceutical dosage forms , pp. 267-286
  • 34
    • 33749514759 scopus 로고    scopus 로고
    • Preparation and in vitro evaluation of a multiple-unit floating drug delivery system based on gas formation technique
    • Sungthongjeen S, Paeratakul O, Limmatvapirat S, Puttipipatkhachorn S. 2006. Preparation and in vitro evaluation of a multiple-unit floating drug delivery system based on gas formation technique. Int J Pharm 324(2):136-143.
    • (2006) Int J Pharm , vol.324 , Issue.2 , pp. 136-143
    • Sungthongjeen, S.1    Paeratakul, O.2    Limmatvapirat, S.3    Puttipipatkhachorn, S.4
  • 35
    • 67049160802 scopus 로고    scopus 로고
    • Design and evaluation of polymeric coated minitablets as multiple unit gastroretentive floating drug delivery systems for furosemide
    • Meka L, Kesavan B, Kalamata VN, Eaga CM, Bandari S, Vobalaboina V, Yamsani MR. 2009. Design and evaluation of polymeric coated minitablets as multiple unit gastroretentive floating drug delivery systems for furosemide. J Pharm Sci 98(6):2122-2132.
    • (2009) J Pharm Sci , vol.98 , Issue.6 , pp. 2122-2132
    • Meka, L.1    Kesavan, B.2    Kalamata, V.N.3    Eaga, C.M.4    Bandari, S.5    Vobalaboina, V.6    Yamsani, M.R.7
  • 36
    • 51449117204 scopus 로고    scopus 로고
    • Preparation of a matrix type multiple-unit gastro retentive floating drug delivery system for captopril based on gas formation technique: In Vitro evaluation
    • Meka L, Kesavan B, Chinnala KM, Vobalaboina V, Yamsani MR. 2008. Preparation of a matrix type multiple-unit gastro retentive floating drug delivery system for captopril based on gas formation technique: In Vitro evaluation. AAPS PharmSciTech 9(2):612-619.
    • (2008) AAPS PharmSciTech , vol.9 , Issue.2 , pp. 612-619
    • Meka, L.1    Kesavan, B.2    Chinnala, K.M.3    Vobalaboina, V.4    Yamsani, M.R.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.