메뉴 건너뛰기




Volumn 115, Issue 3, 2014, Pages 2487-2493

Thermal, spectroscopic, and dissolution studies of ketoconazole-Pluronic F127 system

Author keywords

DSC; Eutectic; FTIR; Intrinsic dissolution; Ketoconazole; Phase diagram; Pluronic F127; Solid dispersion; XRPD

Indexed keywords

DSC; FTIR; KETOCONAZOLE; PLURONIC F-127; SOLID DISPERSION; XRPD;

EID: 84900659654     PISSN: 13886150     EISSN: None     Source Type: Journal    
DOI: 10.1007/s10973-014-3661-2     Document Type: Article
Times cited : (66)

References (23)
  • 1
    • 0020057397 scopus 로고
    • Ketoconazole: A review of its therapeutic efficacy in superficial and systemic fungal infections
    • 1:CAS:528:DyaL38XhtlGjt7Y%3D 10.2165/00003495-198223010-00001
    • Heel RC, Brogden RN, Carmine A, Morley PA, Speight TM, Avery GS. Ketoconazole: a review of its therapeutic efficacy in superficial and systemic fungal infections. Drugs. 1982;23:1-36.
    • (1982) Drugs , vol.23 , pp. 1-36
    • Heel, R.C.1    Brogden, R.N.2    Carmine, A.3    Morley, P.A.4    Speight, T.M.5    Avery, G.S.6
  • 2
    • 0018921956 scopus 로고
    • The activity in vitro and in vivo of a new imidazole antifungal, ketoconazole
    • 1:CAS:528:DyaL3cXhslGjtLY%3D 10.1093/jac/6.1.97
    • Odds FC, Milne LJR, Gentles JC, Ball EH. The activity in vitro and in vivo of a new imidazole antifungal, ketoconazole. J Antimicrob Chemother. 1980;6:97-104.
    • (1980) J Antimicrob Chemother , vol.6 , pp. 97-104
    • Odds, F.C.1    Milne, L.J.R.2    Gentles, J.C.3    Ball, E.H.4
  • 3
    • 0030633665 scopus 로고    scopus 로고
    • Use of azoles for systemic antifungal therapy
    • Kauffman A, Carver P. Use of azoles for systemic antifungal therapy. Adv Pharmacol. 1997;39:147-89.
    • (1997) Adv Pharmacol , vol.39 , pp. 147-189
    • Kauffman, A.1    Carver, P.2
  • 5
    • 77958531109 scopus 로고    scopus 로고
    • Improvement of solubility and dissolution properties of ketoconazole by solid dispersions and inclusion complexes
    • Balata G, Mahdi M, Bakera RA. Improvement of solubility and dissolution properties of ketoconazole by solid dispersions and inclusion complexes. Asian J Pharm Sci. 2010;5:1-12.
    • (2010) Asian J Pharm Sci , vol.5 , pp. 1-12
    • Balata, G.1    Mahdi, M.2    Bakera, R.A.3
  • 6
    • 0033663452 scopus 로고    scopus 로고
    • Physical stabilisation of amorphous ketoconazole in solid dispersions with polyvinylpyrrolidone K25
    • 10.1016/S0928-0987(00)00173-1
    • Van den Mooter G, Wuyts M, Blaton N, Busson R, Grobet P, Augustijns P, Kinget R. Physical stabilisation of amorphous ketoconazole in solid dispersions with polyvinylpyrrolidone K25. Eur J Pharm Sci. 2001;12:261-9.
    • (2001) Eur J Pharm Sci , vol.12 , pp. 261-269
    • Van Den Mooter, G.1    Wuyts, M.2    Blaton, N.3    Busson, R.4    Grobet, P.5    Augustijns, P.6    Kinget, R.7
  • 7
    • 0000312699 scopus 로고    scopus 로고
    • Physicochemical and drug-delivery considerations for oral drug bioavailability
    • 1:CAS:528:DyaK2sXjs1Cgtg%3D%3D 10.1016/1359-6446(96)10039-8
    • Chan OH, Stewart BH. Physicochemical and drug-delivery considerations for oral drug bioavailability. Drug Discov Today. 1996;1:461-73.
    • (1996) Drug Discov Today , vol.1 , pp. 461-473
    • Chan, O.H.1    Stewart, B.H.2
  • 8
    • 57049163132 scopus 로고    scopus 로고
    • Drug delivery strategies for improved azole antifungal action
    • 1:CAS:528:DC%2BD1cXhtlaisrbL 10.1517/17425240802457188
    • Yang W, Wiederhold NP, Williams RO. Drug delivery strategies for improved azole antifungal action. Expert Opin Drug Deliv. 2008;5:1199-216.
    • (2008) Expert Opin Drug Deliv , vol.5 , pp. 1199-1216
    • Yang, W.1    Wiederhold, N.P.2    Williams, R.O.3
  • 9
    • 0036724743 scopus 로고    scopus 로고
    • Antifungal drug resistance to azoles and polyenes
    • 1:CAS:528:DC%2BD38XnsFOjtbk%3D 10.1016/S1473-3099(02)00371-7
    • Canuto MM, Gutierrez F. Antifungal drug resistance to azoles and polyenes. Lancet Infect Dis. 2002;2:550-63.
    • (2002) Lancet Infect Dis. , vol.2 , pp. 550-563
    • Canuto, M.M.1    Gutierrez, F.2
  • 10
    • 78449296944 scopus 로고    scopus 로고
    • Effective formulation development strategies for poorly soluble active pharmaceutical ingredients (APIs)
    • 1:CAS:528:DC%2BC3cXhsFyqu7rF
    • Elder DP. Effective formulation development strategies for poorly soluble active pharmaceutical ingredients (APIs). Am Pharm Rev. 2010;13:28-34.
    • (2010) Am Pharm Rev , vol.13 , pp. 28-34
    • Elder, D.P.1
  • 11
    • 84867825837 scopus 로고    scopus 로고
    • Solid dispersions: A strategy for poorly aqueous soluble drugs and technology updates
    • 1:CAS:528:DC%2BC38XhsFCgsbfN 10.1517/17425247.2012.732064
    • Alam MA, Ali R, Al-Jenoobi FI, Al-Mohizea AM. Solid dispersions: a strategy for poorly aqueous soluble drugs and technology updates. Expert Opin Drug Deliv. 2012;9:1419-40.
    • (2012) Expert Opin Drug Deliv , vol.9 , pp. 1419-1440
    • Alam, M.A.1    Ali, R.2    Al-Jenoobi, F.I.3    Al-Mohizea, A.M.4
  • 12
    • 79959380233 scopus 로고    scopus 로고
    • Phase diagram and dissolution studies of the fenofibrate-acetylsalicylic acid system
    • 10.1007/s10973-010-1148-3
    • Górniak A, Wojakowska A, Karolewicz B, Pluta J. Phase diagram and dissolution studies of the fenofibrate-acetylsalicylic acid system. J Therm Anal Calorim. 2011;104:1195-200.
    • (2011) J Therm Anal Calorim , vol.104 , pp. 1195-1200
    • Górniak, A.1    Wojakowska, A.2    Karolewicz, B.3    Pluta, J.4
  • 13
    • 84881478244 scopus 로고    scopus 로고
    • Thermal, spectroscopic, and dissolution studies of the simvastatin-acetylsalicylic acid mixtures
    • 10.1007/s10973-012-2641-7
    • Górniak A, Karolewicz B, Zurawska-Płaksej E, Pluta J. Thermal, spectroscopic, and dissolution studies of the simvastatin- acetylsalicylic acid mixtures. J Therm Anal Calorim. 2013;111:2125-32.
    • (2013) J Therm Anal Calorim , vol.111 , pp. 2125-2132
    • Górniak, A.1    Karolewicz, B.2    Zurawska-Płaksej, E.3    Pluta, J.4
  • 14
    • 79955592721 scopus 로고    scopus 로고
    • Nanoparticle formation and growth during in vitro dissolution of ketoconazole solid dispersion
    • 1:CAS:528:DC%2BC3MXlslCgs74%3D 10.1002/jps.22491
    • Kanaujia P, Lau G, Kiong W, Widjaja E, Hanefeld A, Fischbach M, Maio M, Tan RBH. Nanoparticle formation and growth during in vitro dissolution of ketoconazole solid dispersion. J Pharm Sci. 2011;100:2876-85.
    • (2011) J Pharm Sci , vol.100 , pp. 2876-2885
    • Kanaujia, P.1    Lau, G.2    Kiong, W.3    Widjaja, E.4    Hanefeld, A.5    Fischbach, M.6    Maio, M.7    Tan, R.B.H.8
  • 15
    • 79955604485 scopus 로고    scopus 로고
    • Physicochemical characterization and dissolution study of solid dispersions of ketoconazole with nicotinamide
    • 1:CAS:528:DC%2BC38XnvFCntA%3D%3D 10.1248/cpb.59.629
    • Aggarwal AK, Jain S. Physicochemical characterization and dissolution study of solid dispersions of ketoconazole with nicotinamide. Chem Pharm Bull. 2011;59:629-38.
    • (2011) Chem Pharm Bull , vol.59 , pp. 629-638
    • Aggarwal, A.K.1    Jain, S.2
  • 16
    • 84859531522 scopus 로고    scopus 로고
    • Physicochemical characterization and release rate studies of solid dispersions of ketoconazole with Pluronic F127 and PVP K-30
    • 1:CAS:528:DC%2BC38XisFCqtro%3D
    • Kumar P, Mohan Ch, Umashankar MS, Gulati M. Physicochemical characterization and release rate studies of solid dispersions of ketoconazole with Pluronic F127 and PVP K-30. Iran J Pharm Res. 2011;10:685-94.
    • (2011) Iran J Pharm Res , vol.10 , pp. 685-694
    • Kumar, P.1    Mohan, C.2    Umashankar, M.S.3    Gulati, M.4
  • 17
  • 18
    • 23844542459 scopus 로고    scopus 로고
    • Effect of solubilizing and microemulsifying excipients in polyethylene glycol 6000 solid dispersion on enhanced dissolution and bioavailability of ketoconazole
    • 1:CAS:528:DC%2BD2MXltVamtbw%3D 10.1007/BF02977766
    • Heo M-Y, Piao Z-Z, Kim T-W, Cao Q-R, Kim A, Lee B-J. Effect of solubilizing and microemulsifying excipients in polyethylene glycol 6000 solid dispersion on enhanced dissolution and bioavailability of ketoconazole. Arch Pharm Res. 2005;28:604-11.
    • (2005) Arch Pharm Res , vol.28 , pp. 604-611
    • Heo, M.-Y.1    Piao, Z.-Z.2    Kim, T.-W.3    Cao, Q.-R.4    Kim, A.5    Lee, B.-J.6
  • 19
    • 0038759662 scopus 로고    scopus 로고
    • Amphiphilic block copolymers for drug delivery
    • 1:CAS:528:DC%2BD3sXltlWhu7g%3D 10.1002/jps.10397
    • Adams ML, Lavasanifar A, Kwon GS. Amphiphilic block copolymers for drug delivery. J Pharm Sci. 2003;92:1343-55.
    • (2003) J Pharm Sci , vol.92 , pp. 1343-1355
    • Adams, M.L.1    Lavasanifar, A.2    Kwon, G.S.3
  • 20
    • 33845351355 scopus 로고    scopus 로고
    • A review of poloxamer 407 pharmaceutical and pharmacological characteristics
    • 1:CAS:528:DC%2BD28Xht1Kmt73I 10.1007/s11095-006-9104-4
    • Dumortier G, Grossiord JL, Agnely F, Chaumeil JC. A review of poloxamer 407 pharmaceutical and pharmacological characteristics. Pharm Res. 2006;23:2709-28.
    • (2006) Pharm Res , vol.23 , pp. 2709-2728
    • Dumortier, G.1    Grossiord, J.L.2    Agnely, F.3    Chaumeil, J.C.4
  • 21
    • 79960120015 scopus 로고    scopus 로고
    • Preparation, physico chemical characterization of solid dispersions of tenoxicam with poloxamer
    • 1:CAS:528:DC%2BC3cXhsVWksL7J
    • Saritha A, Nalini Shastri N. Preparation, physico chemical characterization of solid dispersions of tenoxicam with poloxamer. J Pharm Sci Technol. 2010;2:308-11.
    • (2010) J Pharm Sci Technol , vol.2 , pp. 308-311
    • Saritha, A.1    Nalini Shastri, N.2
  • 23
    • 0037074108 scopus 로고    scopus 로고
    • The mechanism of drug release from solid dispersion in water-soluble polymers
    • 1:CAS:528:DC%2BD3MXptlaitL0%3D 10.1016/S0378-5173(01)00891-2
    • Craig DQ. The mechanism of drug release from solid dispersion in water-soluble polymers. Int J Pharm. 2002;231:131-44.
    • (2002) Int J Pharm , vol.231 , pp. 131-144
    • Craig, D.Q.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.