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Volumn 136, Issue 18, 2014, Pages 6608-6616
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Discovery of amphipathic dynorphin A analogues to inhibit the neuroexcitatory effects of dynorphin A through bradykinin receptors in the spinal cord
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Author keywords
[No Author keywords available]
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Indexed keywords
BINDING ENERGY;
BIOACTIVITY;
RATS;
BINDING AFFINITIES;
CENTRAL NERVOUS SYSTEMS;
DOSE-DEPENDENT MANNER;
HYPERALGESIC EFFECTS;
PERIPHERAL NEUROPATHY;
STRUCTURAL DISSIMILARITIES;
STRUCTURAL FEATURE;
STRUCTURE-ACTIVITY RELATIONSHIPS;
LIGANDS;
BRADYKININ;
BRADYKININ RECEPTOR;
DYNORPHIN A;
DYNORPHIN A DERIVATIVE;
DYNORPHIN A[4-11];
ICATIBANT;
KALLIDIN;
OPIATE RECEPTOR;
UNCLASSIFIED DRUG;
[7 DES ARGININE] DYNORPHIN A[4-11];
DYNORPHIN;
ANIMAL EXPERIMENT;
ANIMAL MODEL;
ANIMAL TISSUE;
ARTICLE;
BINDING AFFINITY;
CARBOXY TERMINAL SEQUENCE;
CENTRAL NERVOUS SYSTEM;
CHRONIC PAIN;
CONTROLLED STUDY;
DRUG RECEPTOR BINDING;
HUMAN;
HUMAN CELL;
HYPERALGESIA;
IN VIVO STUDY;
LIGAND BINDING;
MALE;
MOLECULAR INTERACTION;
MOLECULAR RECOGNITION;
MOTOR DYSFUNCTION;
NERVE CELL EXCITABILITY;
NERVE INJURY;
NONHUMAN;
PERIPHERAL NEUROPATHY;
PHARMACOPHORE;
RAT;
SPINAL CORD;
STRUCTURE ACTIVITY RELATION;
UPREGULATION;
ANIMAL;
CHEMISTRY;
DRUG EFFECTS;
METABOLISM;
NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY;
RADIOASSAY;
SPRAGUE DAWLEY RAT;
ANIMALS;
DYNORPHINS;
MAGNETIC RESONANCE SPECTROSCOPY;
MALE;
RADIOLIGAND ASSAY;
RATS;
RATS, SPRAGUE-DAWLEY;
RECEPTORS, BRADYKININ;
SPINAL CORD;
STRUCTURE-ACTIVITY RELATIONSHIP;
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EID: 84900345297
PISSN: 00027863
EISSN: 15205126
Source Type: Journal
DOI: 10.1021/ja501677q Document Type: Article |
Times cited : (25)
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References (28)
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