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ChemMedChem

Volumn 9, Issue 5, 2014, Pages 928-931

Fluorescence polarization for the evaluation of small-molecule inhibitors of PCAF BRD/Tat-AcK50 association

(6) Hu, Ping a Wang, Xinghui a Zhang, Baiqun a Zhang, Shuai a Wang, Qiang b Wang, Zhiyong a

a UNIVERSITY OF SCIENCE AND TECHNOLOGY OF CHINA (China)

b High Magnetic Field Laboratory Chinese Academy of Sciences (China)

Author keywords

fluorescence polarization; HIV Tat; PCAF; protein peptide interactions; small molecule inhibitors

Indexed keywords

2 (3 AMINOPROPYLAMINO) 5 (HYDROXYMETHYL)PYRIDINE 1 OXIDE; ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; HISTONE ACETYLTRANSFERASE PCAF; LIGAND; LYSINE 50 ACETYLATED TRANSACTIVATOR; PYRIDINE 1 OXIDE; TRANSACTIVATOR PROTEIN; UNCLASSIFIED DRUG; MOLECULAR LIBRARY; PROTEIN BINDING;

ARTICLE; BINDING AFFINITY; DRUG CYTOTOXICITY; DRUG EFFICACY; DRUG SCREENING; DRUG SYNTHESIS; FLUORESCENCE POLARIZATION; HUMAN; HUMAN CELL; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN PROTEIN INTERACTION; STRUCTURE ACTIVITY RELATION; VIRUS INHIBITION; CELL LINE; CHEMICAL STRUCTURE; CHEMISTRY; DOSE RESPONSE; DRUG EFFECTS; GROWTH, DEVELOPMENT AND AGING; HUMAN IMMUNODEFICIENCY VIRUS 1; METABOLISM; MICROBIAL SENSITIVITY TEST; MOLECULAR LIBRARY; PHARMACOLOGY; SYNTHESIS; VIRUS REPLICATION;

ANTI-HIV AGENTS; CELL LINE; DOSE-RESPONSE RELATIONSHIP, DRUG; FLUORESCENCE POLARIZATION; GENE PRODUCTS, TAT; HIV-1; HUMANS; LIGANDS; MICROBIAL SENSITIVITY TESTS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; P300-CBP TRANSCRIPTION FACTORS; PROTEIN BINDING; SMALL MOLECULE LIBRARIES; STRUCTURE-ACTIVITY RELATIONSHIP; VIRUS REPLICATION;

EID: 84899902756 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201300499 Document Type: Article

Times cited : (20)

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