The verapamil transporter expressed in human alveolar epithelial cells (A549) does not interact with β2- receptor agonists

Drug Metabolism and Pharmacokinetics

Volumn 29, Issue 1, 2014, Pages 101-104

  Salomon, Johanna J ^a   Ehrhardt, Carsten ^a   Hosoya, Ken Ichi ^b  

^a TRINITY COLLEGE DUBLIN   (Ireland)

^b UNIVERSITY OF TOYAMA   (Japan)

Author keywords

Bronchodilators; Drug transporter interactions; Inhalation biopharmaceutics; Organic cation transporters; Respiratory epithelium

Indexed keywords

AMANTADINE; BETA 2 ADRENERGIC RECEPTOR STIMULATING AGENT; FORMOTEROL; MEPYRAMINE; ORGANIC CATION TRANSPORTER; QUINIDINE; SALBUTAMOL; VERAPAMIL;

ARTICLE; BINDING AFFINITY; CONCENTRATION RESPONSE; HUMAN; LUNG ALVEOLUS EPITHELIUM; MONOLAYER CULTURE; PIGMENT EPITHELIUM; PROTEIN EXPRESSION; PROTEIN PROTEIN INTERACTION; RESPIRATORY TRACT MUCOSA;

ADRENERGIC BETA-2 RECEPTOR AGONISTS; ALBUTEROL; CALCIUM CHANNEL BLOCKERS; CARRIER PROTEINS; CATIONS; CELL LINE; DRUG INTERACTIONS; EPITHELIAL CELLS; ETHANOLAMINES; HUMANS; PULMONARY ALVEOLI; RESPIRATORY MUCOSA; VERAPAMIL;

EID: 84898438269     PISSN: 13474367     EISSN: 18800920     Source Type: Journal    
DOI: 10.2133/dmpk.DMPK-13-SH-026     Document Type: Article

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