Development of novel gastroretentive drug delivery system of gliclazide: Hollow beads

Drug Development and Industrial Pharmacy

Volumn 40, Issue 3, 2014, Pages 398-408

  Awasthi, Rajendra ^a,b   Kulkarni, Giriraj T ^b  

^a JAWAHARLAL NEHRU TECHNOLOGICAL UNIVERSITY   (India)

^b Laureate Institute of Pharmacy Kathog   (India)

Author keywords

Alginate bead; Buoyancy; Floating bead; Hollow beads; Mucoadhesion

Indexed keywords

ALGINIC ACID; DRUG CARRIER; GLICLAZIDE; HYDROXYPROPYLMETHYLCELLULOSE; PECTIN; PHOSPHATE;

ANIMAL TISSUE; ARTICLE; BUOYANCY; CHEMICAL INTERACTION; CHEMICAL STRUCTURE; CONTROLLED DRUG RELEASE; CONTROLLED STUDY; DIFFERENTIAL SCANNING CALORIMETRY; DIFFUSION; DRUG DELIVERY SYSTEM; DRUG SOLUBILITY; GELATION; GOAT; HOLLOW FLOATING BEAD; IN VITRO STUDY; INFRARED RADIATION; MICROSCOPY; MUCOADHESION; NONHUMAN; PARTICLE SIZE; PHYSICAL PARAMETERS; SCANNING ELECTRON MICROSCOPY; SPECTROSCOPY; STOMACH MUCOSA; X RAY DIFFRACTION;

ALGINATES; CALORIMETRY, DIFFERENTIAL SCANNING; CHEMISTRY, PHARMACEUTICAL; DRUG CARRIERS; DRUG DELIVERY SYSTEMS; GLICLAZIDE; GLUCURONIC ACID; HEXURONIC ACIDS; HYDROGEN-ION CONCENTRATION; HYPOGLYCEMIC AGENTS; METHYLCELLULOSE; MICROSCOPY, ELECTRON, SCANNING; PARTICLE SIZE; PECTINS; SOLUBILITY; SPECTROSCOPY, FOURIER TRANSFORM INFRARED; TIME FACTORS; X-RAY DIFFRACTION;

EID: 84893934764     PISSN: 03639045     EISSN: 15205762     Source Type: Journal    
DOI: 10.3109/03639045.2013.763817     Document Type: Article

References (33)

1. Chien Yie W. Novel drug delivery systems. New York: Informa, Healthcare Inc; 2009.
2. Streubel A, Siepmann J, Bodmeier R. Drug delivery to the upper small intestine window using gastroretentive technologies. Curr Opin Pharmacol 2006;6:501-8.
3. Talukder R, Fassihi R. Gastroretentive delivery systems: hollow beads. Drug Dev Ind Pharm 2004;30:405-12.
4. Soppimath KS, Kulkarni AR, Rudzinski WE, Aminabhavi TM. Microspheres as floating drug delivery systems to increase gastric retention of drugs. Drug Metab Rev 2001;33:149-60.
5. Jain SK, Gupta A. Development of Gelucire 43/01 beads of metformin hydrochloride for floating delivery. AAPS Pharm Sci Tech 2009;10:1128-36.
6. Kofuji K, Isobe T, Murata Y. Controlled release of alpha-lipoic acid through incorporation into natural polysaccharide-based gel beads. Food Chem 2009;115:483-7.
7. Pawar VK, Kansal S, Garg G, et al. Gastroretentive dosage forms: a review with special emphasis on floating drug delivery systems. Drug Deliv 2011;18:97-110.
8. Waterman KC. A critical review of gastric retentive controlled drug delivery. Pharm Dev Technol 2007;12:1-10.
9. Ostberg T, Lund E, Graffner C. Calcium alginate matrixes for oral multiple unit administration: release characteristics in different media. Int J Pharm 1994;112:241-8.
10. Kikuchi A, Kawabuchi M, Sugihara M, et al. Pulsed dextran release from calcium-alginate gel beads. J Controlled Release 1997;47:21-9.
11. Aslani P, Kennedy RA. Effect of gelation conditions and dissolution media on the release of paracetamol from alginate gel beads. J Microencapsulation 1996;13:601-14.
12. Pongjanyakul T, Rongthong T. Enhanced entrapment efficiency and modulated drug release of alginate beads loaded with drug-clay intercalated complexes as microreservoirs. Carbohydr Polym 2010;81:409-19.
13. Patel YL, Sher P, Pawar AP. The effect of drug concentration and curing time on processing and properties of calcium alginate beads containing metronidazole by response surface methodology. AAPS Pharm Sci Tech 2006;7:Article 86. Available from: http://www.aap-spharmscitech.org [last accessed 7 Sep 2012].
14. Sriamornsak P, Nunthanid J, heewatanakornkool K, Manchun S. Effect of drug loading method on drug content and drug release from calcium pectinate gel beads. AAPS Pharm Sci Tech 2010;11:1315-19.
15. Sriamornsak P, Thirawong N, Puttipipatkhachorn S. Emulsion gel beads of calcium pectinate capable of floating on the gastric fluid: effect of some additives, hardening agent or coating on release behavior of metronidazole. Eur J Pharm Sci 2005;24:363-73.
16. Sriamornsak P, Asavapichayont P, Nunthanid J, et al. Piriyaprasarth S. wax-incorporated emulsion gel beads of calcium pectinate for intragastric floating drug delivery. AAPS Pharm Sci Tech 2008;9:571-7.
17. Das S, Ng K-Y, Ho PC. Formulation and optimization of zinc-pectinate beads for the controlled delivery of resveratrol. AAPS Pharm Sci Tech 2010;11:729-42.
18. Rowe RC, Sheskey PJ, Quinn ME. Handbook of pharmaceutical excipients. London: Pharmaceutical Press; American Pharmacists Association; 2009.
19. Sriamornsak P, Thirawong N, Puttipipatkhachorn S. (2004). Morphology and buoyancy of oil-entrapped calcium pectinate gel beads. AAPS J 2004;6:Article 24. Available from: http://www.aapsj. org [last accessed 10 June 2012].
20. Sriamornsak P, Sungthongjeen S, Puttipipatkhachorn S. Use of pectin as a carrier for intragastric floating drug delivery: carbonate salt contained beads. Carbohydr Polym 2007;67:436-45.
21. Gribic S, Parojcic J, Ibric S, Djuric Z. In vitro-in vivo correlation for gliclazide immediate-release tablets based on mechanistic absorption simulation. AAPS Pharm Sci Tech 2011;12:165-71.
22. Fahmy RH. Statistical approach for assessing the influence of calcium silicate and hpmc on the formulation of novel alfuzosin hydrochloride mucoadhesive-floating beads as gastroretentive drug delivery systems. AAPS Pharm Sci Tech 2012;13:990-1004.
23. Kadajji VG, Betageri GV. Water soluble polymers for pharmaceutical applications. Polymers 2011;3:1972-2009.
24. Oh SH, Parka IL, Kim JM, Lee JH. (2007) In vitro and in vivo characteristics of PCL scaffolds with pore size gradient fabricated by a centrifugation method. Biomaterials 2007;28:1664-71.
25. Yeo Y, Park K. Control of encapsulation efficiency and initial burst in polymeric microparticle systems. Arch Pharm Res 2004;27:1-12.
26. McCauley JA, Brittain HG. Thermal methods of analysis. In: Brittain HG, ed. Physical characterization of pharmaceutical solids, drugs and pharmaceutical sciences. New York: Marcel Dekker; 1995:223-50.
27. Mura P, Faucci MT, Parrini PL. Effects of grinding with microcrystalline cellulose and cyclodextrins on the ketoprofen physicochemical properties. Drug Dev Ind Pharm 2001;27:119-28.
28. Baker PW, Lonsdale HK. Controlled release of biologically active agents. New York: Plenum; 1974.
29. Madan PL. Clofibrate microcapsules: III. Mechanism of release. Drug Dev Ind Pharm 1980;6:629-44.
30. Nath BS, Kulkarni GT, Rao KP. In vitro release kinetics of nitrofurantoin from gelatin microbeads prepared from extrusion-congealing technique. Estern Pharmacist 1995;37:139-42.
31. Al-Kassas RS, Al-Gohary OMN, Al-Faadhel MM. Controlling of systemic absorption of gliclazide through incorporation into alginate beads. Int J Pharm 2007;341:230-7.
32. Awasthi R, Kulkarni GT, Pawar VK, Garg G. Optimization studies on gastroretentive floating system using response surface methodology. AAPS Pharm Sci Tech 2012;13:85-93.
33. Awasthi R, Kulkarni GT. Development of novel gastroretentive floating particulate drug delivery system of gliclazide. Curr Drug Deliv 2012;9:437-51.