Predicting the antinociceptive efficacy of σ1 receptor ligands by a novel receptor fluorescence resonance energy transfer (FRET) based biosensor

Journal of Medicinal Chemistry

Volumn 57, Issue 1, 2014, Pages 238-242

  Gómez Soler, Maricel ^a   Fernández Dueñas, Víctor ^a   Portillo Salido, Enrique ^b   Pérez, Pilar ^b   Zamanillo, Daniel ^b   Vela, José Miguel ^b   Burgueño, Javier ^b   Ciruela, Francisco ^a  

^a Unitat de Bioquimica   (Spain)

^b Esteve   (Spain)

Author keywords

[No Author keywords available]

Indexed keywords

1 [ 2 ( 3,4 DICHLOROPHENYL)ETHYL] 4 METHYLPIPERAZINE; 2 [4 METHOXY 3 (2 PHENYLETHOXY)PHENYL] N,N DIPROPYLETHYLAMINE; BD 1063; CHAPERONE; FORMALDEHYDE; HALOPERIDOL; OPIATE ANTAGONIST; OPIATE RECEPTOR AFFECTING AGENT; PENTAZOCINE; SIGMA 1 OPIATE RECEPTOR; SIGMA 1 OPIATE RECEPTOR LIGAND; UNCLASSIFIED DRUG;

ANALGESIA; ANALYTIC METHOD; ANIMAL EXPERIMENT; ARTICLE; ATTENUATION; BIOASSAY; BIOSENSOR; BLEACHING; CONTROLLED STUDY; DRUG EFFICACY; FLUORESCENCE RESONANCE ENERGY TRANSFER; HUMAN; HUMAN CELL; MOUSE; NOCICEPTION; NONHUMAN; PAIN; PROTEIN CONFORMATION;

ANALGESICS; ANIMALS; BIOSENSING TECHNIQUES; FLUORESCENCE RESONANCE ENERGY TRANSFER; LIGANDS; MICE; RECEPTORS, SIGMA;

EID: 84892599073     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm401529t     Document Type: Article

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