메뉴 건너뛰기




Volumn 14, Issue 3, 2013, Pages 994-1003

Design and evaluation of self-nanoemulsifying pellets of repaglinide

Author keywords

anti hyperglycemic activity; extrusion spheronization; repaglinide; self nanoemulsifying pellets

Indexed keywords

GLUCOSE; LACTOSE; MICROCRYSTALLINE CELLULOSE; REPAGLINIDE; STREPTOZOCIN; SURFACTANT;

EID: 84890177977     PISSN: None     EISSN: 15309932     Source Type: Journal    
DOI: 10.1208/s12249-013-9990-9     Document Type: Article
Times cited : (26)

References (32)
  • 1
    • 0342617694 scopus 로고    scopus 로고
    • Lipid-based vehicles for the oral delivery of poorly water soluble drugs
    • 10.1016/S0169-409X(96)00494-2 1:CAS:528:DyaK2sXhtlOqs70%3D
    • Humberstone AJ, Charman WN. Lipid-based vehicles for the oral delivery of poorly water soluble drugs. Adv Drug Deliv Rev. 1997;25:103-28.
    • (1997) Adv Drug Deliv Rev. , vol.25 , pp. 103-128
    • Humberstone, A.J.1    Charman, W.N.2
  • 2
    • 0034808093 scopus 로고    scopus 로고
    • Repaglinide, a review of its therapeutic use in type 2 diabetes mellitus
    • 11577798 10.2165/00003495-200161110-00008 1:CAS:528:DC%2BD3MXnvVCqs70%3D
    • Culy C, Jarvis B. Repaglinide, a review of its therapeutic use in type 2 diabetes mellitus. Drugs. 2001;61:1625-60.
    • (2001) Drugs , vol.61 , pp. 1625-1660
    • Culy, C.1    Jarvis, B.2
  • 3
    • 0033001413 scopus 로고    scopus 로고
    • Repaglinide, a new oral antidiabetic agent: A review of recent preclinical studies
    • 10383607 10.1046/j.1365-2362.1999.00001.x 1:CAS:528:DyaK1MXktFOhsLc%3D
    • Malaisse W. Repaglinide, a new oral antidiabetic agent: a review of recent preclinical studies. Eur J Clin Invest. 1999;29:21-9.
    • (1999) Eur J Clin Invest. , vol.29 , pp. 21-29
    • Malaisse, W.1
  • 4
    • 33646403422 scopus 로고    scopus 로고
    • Ionization, lipophilicity and solubility properties of repaglinide
    • 16520012 10.1016/j.jpba.2006.01.056 1:CAS:528:DC%2BD28Xks1CjtLw%3D
    • Mandic Z, Gabelica V. Ionization, lipophilicity and solubility properties of repaglinide. J Pharm Biomed Anal. 2006;41(3):866-71.
    • (2006) J Pharm Biomed Anal , vol.41 , Issue.3 , pp. 866-871
    • Mandic, Z.1    Gabelica, V.2
  • 6
    • 0002096610 scopus 로고    scopus 로고
    • Insulin, oral hypoglycemic agents and the pharmacology of the endocrine pancreas
    • J.G. Hardman L.E. Limbrid (eds) McGraw-Hill USA
    • Davis SN, Granner DK. Insulin, oral hypoglycemic agents and the pharmacology of the endocrine pancreas. In: Hardman JG, Limbrid LE, editors. Goodman and Gilman's the pharmacological basis of therapeutics. USA: McGraw-Hill; 2001. p. 1704-5.
    • (2001) Goodman and Gilman's the Pharmacological Basis of Therapeutics , pp. 1704-1705
    • Davis, S.N.1    Granner, D.K.2
  • 7
    • 45849111476 scopus 로고    scopus 로고
    • Dissolution rates and supersaturation behavior of amorphous repaglinide particles produced by controlled precipitation
    • 10.1166/jbn.2007.001 1:CAS:528:DC%2BD2sXkvVemsbo%3D
    • Sinswat P, Matteucci ME, Johnston KP, Williams III RO. Dissolution rates and supersaturation behavior of amorphous repaglinide particles produced by controlled precipitation. J Biomed Nanotechnol. 2007;3:18-27.
    • (2007) J Biomed Nanotechnol , vol.3 , pp. 18-27
    • Sinswat, P.1    Matteucci, M.E.2    Johnston, K.P.3    Williams III, R.O.4
  • 8
    • 79956030072 scopus 로고    scopus 로고
    • Repaglinide-cyclodextrin complexes: Preparation, characterization and in vivo evaluation of antihyperglycemic activity
    • 10.1007/s10847-010-9895-0 1:CAS:528:DC%2BC3MXlslynur8%3D
    • Desai NS, Bramhane DM, Nagarsenker MS. Repaglinide-cyclodextrin complexes: preparation, characterization and in vivo evaluation of antihyperglycemic activity. J Incl Phenom Macrocycl Chem. 2011;70(1-2):217-25.
    • (2011) J Incl Phenom Macrocycl Chem , vol.70 , Issue.1-2 , pp. 217-225
    • Desai, N.S.1    Bramhane, D.M.2    Nagarsenker, M.S.3
  • 9
    • 84859455331 scopus 로고    scopus 로고
    • Preparation, characterization and in vivo evaluation of antihyperglycemic activity of microwave generated repaglinide solid dispersion
    • 22466731 10.1248/cpb.60.482 1:CAS:528:DC%2BC38XovFSksr0%3D
    • Zawar LR, Bari SB. Preparation, characterization and in vivo evaluation of antihyperglycemic activity of microwave generated repaglinide solid dispersion. Chem Pharm Bull. 2012;60(4):482-7.
    • (2012) Chem Pharm Bull , vol.60 , Issue.4 , pp. 482-487
    • Zawar, L.R.1    Bari, S.B.2
  • 10
    • 84862504521 scopus 로고    scopus 로고
    • Enhancement of solubility of repaglinide by solid dispersion technique
    • 1:CAS:528:DC%2BC38Xos1Whu70%3D
    • Kavitha R, Sathali AAH. Enhancement of solubility of repaglinide by solid dispersion technique. Int J Chem Sci. 2012;10(1):377-90.
    • (2012) Int J Chem Sci , vol.10 , Issue.1 , pp. 377-390
    • Kavitha, R.1    Sathali, A.A.H.2
  • 11
    • 79955913657 scopus 로고    scopus 로고
    • Preparation, characterization and in vitro evaluation of repaglinide binary solid dispersions with hydrophilic polymers
    • 1:CAS:528:DC%2BC3MXkvFKju7Y%3D
    • Patel M, Pandya N, Bhaskar VH. Preparation, characterization and in vitro evaluation of repaglinide binary solid dispersions with hydrophilic polymers. Int J Drug Dev & Res. 2011;3(2):107-17.
    • (2011) Int J Drug Dev & Res , vol.3 , Issue.2 , pp. 107-117
    • Patel, M.1    Pandya, N.2    Bhaskar, V.H.3
  • 12
    • 51449095969 scopus 로고    scopus 로고
    • Micellar solubilization of some poorly soluble antidiabetic drugs: A technical note
    • 18431666 10.1208/s12249-008-9057-5 1:CAS:528:DC%2BC3cXnslGjt78%3D
    • Seedher N, Kanojia M. Micellar solubilization of some poorly soluble antidiabetic drugs: a technical note. AAPS PharmSciTech. 2008;9(2):431-6.
    • (2008) AAPS PharmSciTech , vol.9 , Issue.2 , pp. 431-436
    • Seedher, N.1    Kanojia, M.2
  • 14
    • 1842684453 scopus 로고    scopus 로고
    • Self-emulsifying drug delivery systems (SEDDS) for improved oral delivery of lipophilic drugs
    • 15082340 10.1016/j.biopha.2004.02.001
    • Gursoy RN, Benita S. Self-emulsifying drug delivery systems (SEDDS) for improved oral delivery of lipophilic drugs. Biomed Pharmacother. 2004;58:173-82.
    • (2004) Biomed Pharmacother , vol.58 , pp. 173-182
    • Gursoy, R.N.1    Benita, S.2
  • 15
    • 0034614208 scopus 로고    scopus 로고
    • Microemulsion-based media as novel drug delivery systems
    • 11104900 10.1016/S0169-409X(00)00103-4 1:CAS:528:DC%2BD3cXosFertb4%3D
    • Lawrence MJ, Rees GD. Microemulsion-based media as novel drug delivery systems. Adv Drug Deliv Rev. 2000;45:89-121.
    • (2000) Adv Drug Deliv Rev. , vol.45 , pp. 89-121
    • Lawrence, M.J.1    Rees, G.D.2
  • 16
    • 33646854907 scopus 로고    scopus 로고
    • Enhanced bioavailability of silymarin by self-microemulsifying drug delivery system
    • 10.1016/j.ejpb.2005.12.005
    • Wei W, Yang W, Li Q. Enhanced bioavailability of silymarin by self-microemulsifying drug delivery system. Eur J Pharm Biopharm. 2006;63:288-94.
    • (2006) Eur J Pharm Biopharm , vol.63 , pp. 288-294
    • Wei, W.1    Yang, W.2    Li, Q.3
  • 17
    • 78650539714 scopus 로고    scopus 로고
    • Self-nanoemulsifying drug delivery systems: Formulation insights, applications and advances
    • 21143036 10.2217/nnm.10.126 1:CAS:528:DC%2BC3cXhsFGltLnE
    • Date A, Desai N, Dixit R, Nagarsenker M. Self-nanoemulsifying drug delivery systems: formulation insights, applications and advances. Nanomedicine. 2010;5(10):1595-616.
    • (2010) Nanomedicine , vol.5 , Issue.10 , pp. 1595-1616
    • Date, A.1    Desai, N.2    Dixit, R.3    Nagarsenker, M.4
  • 18
    • 0031957735 scopus 로고    scopus 로고
    • A study on gelatin capsule brittleness: Moisture transfer between the capsule shell and its content
    • 9572904 10.1021/js9704238 1:CAS:528:DyaK1cXis12jsbw%3D
    • Chang RK, Raghavan KS, Hussain MA. A study on gelatin capsule brittleness: moisture transfer between the capsule shell and its content. J Pharm Sci. 1998;87:556-8.
    • (1998) J Pharm Sci , vol.87 , pp. 556-558
    • Chang, R.K.1    Raghavan, K.S.2    Hussain, M.A.3
  • 19
    • 33749532642 scopus 로고    scopus 로고
    • Use of texture analyzer to study hydrophilic solvent effects on the mechanical properties of hard gelatin capsules
    • 16844327 10.1016/j.ijpharm.2006.06.017 1:CAS:528:DC%2BD28XhtVOgu77I
    • Mei X, Etzler FM, Wang Z. Use of texture analyzer to study hydrophilic solvent effects on the mechanical properties of hard gelatin capsules. Int J Pharm. 2006;324:128-35.
    • (2006) Int J Pharm , vol.324 , pp. 128-135
    • Mei, X.1    Etzler, F.M.2    Wang, Z.3
  • 20
    • 67549143093 scopus 로고    scopus 로고
    • Preparation and evaluation of self-nanoemulsifying tablets of carvedilol
    • 10.1208/s12249-009-9192-7 1:CAS:528:DC%2BC3cXotV2mtbk%3D
    • Mahmoud EA, Bendas ER, Mohamed MI. Preparation and evaluation of self-nanoemulsifying tablets of carvedilol. AAPS Pharm Sci Tech. 2009;10:183-92.
    • (2009) AAPS Pharm Sci Tech. , vol.10 , pp. 183-192
    • Mahmoud, E.A.1    Bendas, E.R.2    Mohamed, M.I.3
  • 21
    • 57349119914 scopus 로고    scopus 로고
    • Formulation and in vivo evaluation of self-nanoemulsifying granules for oral delivery of a combination of ezetimibe and simvastatin
    • 18720144 10.1080/03639040802071570 1:CAS:528:DC%2BD1cXhtlyjsLzN
    • Dixit RP, Nagarsenker MS. Formulation and in vivo evaluation of self-nanoemulsifying granules for oral delivery of a combination of ezetimibe and simvastatin. Drug Dev Ind Pharm. 2008;34:1285-96.
    • (2008) Drug Dev Ind Pharm. , vol.34 , pp. 1285-1296
    • Dixit, R.P.1    Nagarsenker, M.S.2
  • 23
    • 2642540226 scopus 로고    scopus 로고
    • Comparative bioavailability study in dogs of a self emulsifying formulation of progesterone presented in a pellet and liquid form compared with an aqueous suspension of progesterone
    • 15124207 10.1002/jps.20068 1:CAS:528:DC%2BD2cXks12iu7g%3D
    • Tuleu C, Newton JM, Rose J, Euler D, Saklatvala R, Clarke A, et al. Comparative bioavailability study in dogs of a self emulsifying formulation of progesterone presented in a pellet and liquid form compared with an aqueous suspension of progesterone. J Pharm Sci. 2004;93:1495-502.
    • (2004) J Pharm Sci , vol.93 , pp. 1495-1502
    • Tuleu, C.1    Newton, J.M.2    Rose, J.3    Euler, D.4    Saklatvala, R.5    Clarke, A.6    Booth, S.7
  • 24
    • 33847148114 scopus 로고    scopus 로고
    • The preparation of pellets containing a surfactant or a mixture of mono- and di-glycerides by extrusion/spheronization
    • 17223021 10.1016/j.ejps.2006.11.020 1:CAS:528:DC%2BD2sXitFyrsLs%3D
    • Newton JM, Pinto MR, Podczeck F. The preparation of pellets containing a surfactant or a mixture of mono- and di-glycerides by extrusion/spheronization. Eur J Pharm Sci. 2007;30:333-42.
    • (2007) Eur J Pharm Sci , vol.30 , pp. 333-342
    • Newton, J.M.1    Pinto, M.R.2    Podczeck, F.3
  • 25
    • 84867402149 scopus 로고    scopus 로고
    • Sirolimus solid self-microemulsifying pellets: Formulation development, characterization and bioavailability evaluation
    • 10.1016/j.ijpharm.2012.07.055
    • Xiongwei H, Chen L, Dingxiong C, Jing Z, Zhihong L, Wei W, et al. Sirolimus solid self-microemulsifying pellets: formulation development, characterization and bioavailability evaluation. Int J Pharm. 2012;438:123-33.
    • (2012) Int J Pharm , vol.438 , pp. 123-133
    • Xiongwei, H.1    Chen, L.2    Dingxiong, C.3    Jing, Z.4    Zhihong, L.5    Wei, W.6    Hongtao, S.7
  • 26
    • 34247536269 scopus 로고    scopus 로고
    • Preparation and characterization of a self emulsifying pellet formulation
    • 17196807 10.1016/j.ejpb.2006.11.015 1:CAS:528:DC%2BD2sXkslCht78%3D
    • Abdalla A, Mäder K. Preparation and characterization of a self emulsifying pellet formulation. Eur J Pharm Biopharm. 2007;66:220-6.
    • (2007) Eur J Pharm Biopharm , vol.66 , pp. 220-226
    • Abdalla, A.1    Mäder, K.2
  • 27
    • 33845576641 scopus 로고    scopus 로고
    • Design and evaluation of self-nanoemulsifying drug delivery systems (SNEDDS) for cefpodoxime proxetil
    • 17010543 10.1016/j.ijpharm.2006.08.038 1:CAS:528:DC%2BD28XhtlCmtLjN
    • Date AA, Nagarsenker MS. Design and evaluation of self-nanoemulsifying drug delivery systems (SNEDDS) for cefpodoxime proxetil. Int J Pharm. 2007;329:166-72.
    • (2007) Int J Pharm , vol.329 , pp. 166-172
    • Date, A.A.1    Nagarsenker, M.S.2
  • 28
    • 39149113817 scopus 로고    scopus 로고
    • Formulation of lipid-based delivery systems for oral administration: Materials, methods and strategies
    • 18068260 10.1016/j.addr.2007.10.010 1:CAS:528:DC%2BD1cXitVOnu7s%3D
    • Pouton CW, Porter CJH. Formulation of lipid-based delivery systems for oral administration: materials, methods and strategies. Adv Drug Deliv Rev. 2008;60:625-37.
    • (2008) Adv Drug Deliv Rev. , vol.60 , pp. 625-637
    • Pouton, C.W.1    Porter, C.J.H.2
  • 29
    • 39149092022 scopus 로고    scopus 로고
    • Enhancing intestinal drug solubilisation using lipid-based delivery systems
    • 18155801 10.1016/j.addr.2007.10.014 1:CAS:528:DC%2BD1cXitVOmsr4%3D
    • Porter CJH, Pouton CW, Cuine JF, Charman WN. Enhancing intestinal drug solubilisation using lipid-based delivery systems. Adv Drug Deliv Rev. 2008;60:673-91.
    • (2008) Adv Drug Deliv Rev. , vol.60 , pp. 673-691
    • Porter, C.J.H.1    Pouton, C.W.2    Cuine, J.F.3    Charman, W.N.4
  • 30
    • 0034601204 scopus 로고    scopus 로고
    • Self-dispersing lipid formulations for improving oral absorption of lipophilic drugs
    • 10840200 10.1016/S0939-6411(00)00089-8 1:CAS:528:DC%2BD3cXjslyisrk%3D
    • Gershanik T, Benita S. Self-dispersing lipid formulations for improving oral absorption of lipophilic drugs. Eur J Pharm Biopharm. 2000;50(1):179-88.
    • (2000) Eur J Pharm Biopharm , vol.50 , Issue.1 , pp. 179-188
    • Gershanik, T.1    Benita, S.2
  • 31
    • 0034889914 scopus 로고    scopus 로고
    • The influence of formulation variables on the properties of pellets containing a self-emulsifying mixture
    • 11536202 10.1002/jps.1051 1:CAS:528:DC%2BD3MXmtFKlurc%3D
    • Newton M, Petersson J, Podczeck F, Clarke A, Booth S. The influence of formulation variables on the properties of pellets containing a self-emulsifying mixture. J Pharm Sci. 2001;90:987-95.
    • (2001) J Pharm Sci , vol.90 , pp. 987-995
    • Newton, M.1    Petersson, J.2    Podczeck, F.3    Clarke, A.4    Booth, S.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.