Structure-anti-MRSA activity relationship of macrocyclic bis(bibenzyl) derivatives

Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 24, 2013, Pages 6563-6568

  Sawada, Hiromi ^a   Onoda, Kenji ^a   Morita, Daichi ^a   Ishitsubo, Erika ^b   Matsuno, Kenji ^a   Tokiwa, Hiroaki ^b   Kuroda, Teruo ^a   Miyachi, Hiroyuki ^a  

^a OKAYAMA UNIVERSITY   (Japan)

^b RIKKYO UNIVERSITY   (Japan)

Author keywords

Isoplagiochin; Marchantin; Methicillin resistance; Riccardin; Structure activity relationship

Indexed keywords

ANTIINFECTIVE AGENT; BENZENE; BIS(BIBENZYL) DERIVATIVE; HYDROXYL GROUP; ISOPLAGIOCHIN; MACROCYCLIC COMPOUND; MARCHANTIN; PHENYL GROUP; RICCARDIN; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERICIDAL ACTIVITY; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; HYDROPHILICITY; HYDROPHOBICITY; METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS; MOLECULAR DYNAMICS; NONHUMAN; STRUCTURE ACTIVITY RELATION;

METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS;

ISOPLAGIOCHIN; MARCHANTIN; METHICILLIN RESISTANCE; RICCARDIN; STRUCTURE-ACTIVITY RELATIONSHIP;

ANTI-BACTERIAL AGENTS; BIBENZYLS; HYDROPHOBIC AND HYDROPHILIC INTERACTIONS; MACROCYCLIC COMPOUNDS; METHICILLIN-RESISTANT STAPHYLOCOCCUS AUREUS; MOLECULAR DYNAMICS SIMULATION; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84888860592     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2013.10.069     Document Type: Article

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