Structure-activity relationship studies of thalidomide analogs with a taxol-like mode of action

Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 24, 2013, Pages 6902-6904

  Pandit, Bulbul ^a   Hu, Zhigen ^a   Chettiar, Somsundaram N ^a   Zink, Jennifer ^a   Xiao, Zili ^a   Etter, Jonathan P ^a   Bhasin, Deepak ^a   Li, Pui Kai ^a  

^a OHIO STATE UNIVERSITY   (United States)

Author keywords

Anti microtubule agents; Thalidomide analogs

Indexed keywords

5 HYDROXY (2,6 DIISOPROPYLPHENYL) 1H ISOINDOLE 1,3 DIONE; 5HPP 33; BENZENE DERIVATIVE; ISOINDOLE DERIVATIVE; PACLITAXEL; THALIDOMIDE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIPROLIFERATIVE ACTIVITY; ARTICLE; BREAST CANCER; CANCER CELL; CANCER CELL CULTURE; CANCER INHIBITION; CONTROLLED STUDY; DRUG CONFORMATION; DRUG MECHANISM; DRUG SYNTHESIS; ESTERIFICATION; HUMAN; HUMAN CELL; IN VITRO STUDY; MICROTUBULE ASSEMBLY; PROSTATE CANCER; STRUCTURE ACTIVITY RELATION;

ANTI-MICROTUBULE AGENTS; THALIDOMIDE ANALOGS;

CELL LINE, TUMOR; CELL PROLIFERATION; HUMANS; ISOINDOLES; MICROTUBULES; PACLITAXEL; STRUCTURE-ACTIVITY RELATIONSHIP; THALIDOMIDE; TUBULIN MODULATORS;

EID: 84888859456     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2013.09.084     Document Type: Article

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