Mesoporous calcium carbonate as a phase stabilizer of amorphous celecoxib - an approach to increase the bioavailability of poorly soluble pharmaceutical substances

Advanced Healthcare Materials

Volumn 2, Issue 11, 2013, Pages 1469-1476

  Forsgren, Johan ^a   Andersson, Mattias ^b   Nilsson, Peter ^b   Mihranyan, Albert ^a  

^a UPPSALA UNIVERSITY   (Sweden)

^b Orexo AB   (Sweden)

Author keywords

Amorphous drugs; Calcium carbonate; Celecoxib; Drug solubility; Mesoporous materials

Indexed keywords

AMORPHIZATION; BIOCHEMISTRY; CALCITE; CALCIUM CARBONATE; DRUG DELIVERY; SILICA; SOLUBILITY;

ACTIVE PHARMACEUTICAL INGREDIENTS; AMORPHOUS DRUGS; CELECOXIB; DRUG SOLUBILITY; MESOPOROUS STRUCTURES; ORAL BIOAVAILABILITIES; ORDERED MESOPOROUS SILICAS; PHARMACEUTICAL EXCIPIENT;

MESOPOROUS MATERIALS;

CALCIUM CARBONATE; CELECOXIB; CYCLOOXYGENASE 2; EXCIPIENT;

ARTICLE; CRYSTALLIZATION; DRUG BIOAVAILABILITY; DRUG FORMULATION; DRUG SOLUBILITY; DRUG STABILITY; DRUG STRUCTURE; DRUG SYNTHESIS; HYDROPHOBICITY; POLARIZATION; PRIORITY JOURNAL; THERMODYNAMICS; X RAY DIFFRACTION;

AMORPHOUS DRUGS; CALCIUM CARBONATE; CELECOXIB; DRUG SOLUBILITY; MESOPOROUS MATERIALS;

BIOLOGICAL AVAILABILITY; CALCIUM CARBONATE; CALORIMETRY, DIFFERENTIAL SCANNING; CRYSTALLIZATION; MICROSCOPY, ELECTRON, SCANNING; NITROGEN; PHASE TRANSITION; POROSITY; PYRAZOLES; SOLUBILITY; SULFONAMIDES; TEMPERATURE; X-RAY DIFFRACTION;

EID: 84887162438     PISSN: 21922640     EISSN: 21922659     Source Type: Journal    
DOI: 10.1002/adhm.201200391     Document Type: Article

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