The making of i-bet762, a BET bromodomain inhibitor now in clinical development

Journal of Medicinal Chemistry

Volumn 56, Issue 19, 2013, Pages 7498-7500

  Zhao, Yujun ^a   Yang, Chao Yie ^a   Wang, Shaomeng ^a  

^a UNIVERSITY OF MICHIGAN   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIINFLAMMATORY AGENT; ANTINEOPLASTIC AGENT; BENZODIAZEPINE DERIVATIVE; IBET 762; PROTEIN INHIBITOR; UNCLASSIFIED DRUG;

DRUG STRUCTURE; DRUG SYNTHESIS; DRUG TARGETING; EPIGENETICS; HUMAN; NEOPLASM; PHASE 1 CLINICAL TRIAL; REVIEW;

ANIMALS; ANTINEOPLASTIC AGENTS; BENZODIAZEPINES; HUMANS; NUCLEAR PROTEINS; TRANSCRIPTION FACTORS;

EID: 84885623316     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm4014407     Document Type: Review

References (7)

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