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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 21, 2013, Pages 5945-5948

2-Amino-6-chloro-3,4-dihydroquinazoline: A novel 5-HT3 receptor antagonist with antidepressant character

(5) Dukat, Małgorzata a Alix, Katie a Worsham, Jessica a Khatri, Shailesh b Schulte, Marvin K b

a VIRGINIA COMMONWEALTH UNIVERSITY (United States)

b UNIVERSITY OF THE SCIENCES (United States)

Author keywords

5 HT3 receptors; Antagonists; Antidepressants; TST (tail suspension test)

Indexed keywords

2 AMINO 6 CHLORO 3,4 DIHYDROQUINAZOLINE; ANTIDEPRESSANT AGENT; DESIPRAMINE; FLUOXETINE; IMIPRAMINE; MD 354; ONDANSETRON; QUINAZOLINE; SEROTONIN 3 AGONIST; SEROTONIN 3 ANTAGONIST; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANTIDEPRESSANT ACTIVITY; ARTICLE; BLOOD BRAIN BARRIER; CONTROLLED STUDY; DRUG BIOAVAILABILITY; DRUG STRUCTURE; FEMALE; LOCOMOTION; MOUSE; NONHUMAN; OOCYTE; SPECTROSCOPY; VOLTAGE CLAMP;

ANURA;

5-HT(3) RECEPTORS; ANTAGONISTS; ANTIDEPRESSANTS; TST (TAIL SUSPENSION TEST);

AMINATION; ANIMALS; ANTIDEPRESSIVE AGENTS; ANURA; HALOGENATION; HINDLIMB SUSPENSION; MICE; QUINAZOLINES; RECEPTORS, SEROTONIN, 5-HT3; SEROTONIN 5-HT3 RECEPTOR ANTAGONISTS;

EID: 84885176023 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.08.072 Document Type: Article

Times cited : (36)

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