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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 21, 2013, Pages 5844-5849

Studies on substituted benzo[h]quinazolines, benzo[g]indazoles, pyrazoles, 2,6-diarylpyridines as anti-tubercular agents

(9) Maurya, Hardesh K a Verma, Ruby a Alam, Saba a Pandey, Shweta a Pathak, Vinay a Sharma, Sandeep b Srivastava, Kishore K b Negi, Arvind S a Gupta, Atul a

a CSIR CENTRAL INSTITUTE OF MEDICINAL AND AROMATIC PLANTS (India)

b CENTRAL DRUG RESEARCH INSTITUTE (India)

Author keywords

Antitubercular; Diarylpyridine; Indazole; Pyrazole; Quinazoline

Indexed keywords

(4 (2 AMINO 8 METHOXY 5,6 DIHYDROBENZO [H] QUINAZOLIN 4 YL)PHENOXY)ALKANOATE; (4 (2 AMINO 8 METHOXY 5,6 DIHYDROBENZO[H] QUINAZOLIN 4 YL)PHENOXY)ALKANEHYDRAZIDE; 1 (3 (4 ALKOXYPHENYL) 7 METHOXY 3,3A,4,5 TETRAHYDRO 2H BENZO[G]INDAZOL 2 YL)ETHANONE; 1 (3 (4 HYDROXYPHENYL) 7 METHOXY 3,3A,4,5 TETRAHYDRO 2H BENZO[G]INDAZOL 2 YL)ETHANONE; 1 (3 (4 HYDROXYPHENYL) 7 METHOXY 3,3A,4,5TETRAHYDRO 2H BENZO[G]INDAZOL 2 YL); 2 (4 HYDROXYBENZYLIDENE) 6METHOXY 3,4 DIHYDRO NAPHTHALEN 1(2H) ONE; 2 CYANO 5 OXO 5 PHENYL 3 PIPERIDIN 1 YL PENT 2 ENOIC ACID ETHYL ESTER; 5,6 DIHYDRO 8 METHOXYBENZO[H]QUINAZOLIN 2 AMINE; CHALCONE; DIOXANE DERIVATIVE; ETHAMBUTOL; ETHIONAMIDE; ISONIAZID; PYRAZINAMIDE; PYRAZOLE DERIVATIVE; PYRIDINE DERIVATIVE; PYRIMIDINE DERIVATIVE; RIFAMPICIN; STREPTOMYCIN; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIAL STRAIN; BIOLOGICAL ACTIVITY; CYTOTOXICITY; DRUG STRUCTURE; DRUG SYNTHESIS; IN VITRO STUDY; LIPOPHILICITY; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; STRUCTURE ACTIVITY RELATION;

MYCOBACTERIUM TUBERCULOSIS;

AFRWBGJRWRHQOV-UHFFFAOYSA-N; AJTJGWQHYALTSC-UHFFFAOYSA-N; AKKATVMDHBEASX-UHFFFAOYSA-N; ANTITUBERCULAR; AYZGFAJCOVMXLA-UHFFFAOYSA-N; CFOCPVQZZLPMIO-UHFFFAOYSA-N; CMWJZWOGUWCFQV-UHFFFAOYSA-N; CTEHHBOBZOCAIT-UHFFFAOYSA-N; CTODEFQZHRGULH-UHFFFAOYSA-N; DBXRLXVTWNUHCR-UHFFFAOYSA-N; DIARYLPYRIDINE; DSCMLTAZYFVUPH-UHFFFAOYSA-N; DSLIJABHAVBSDV-UHFFFAOYSA-N; DWRUNZAIXLCFIP-UHFFFAOYSA-N; DXBULVYHTICWKT-UHFFFAOYSA-N; DXPKJYJXQICXLT-UHFFFAOYSA-N; FIGVJXMTQDHJMQ-UHFFFAOYSA-N; GYXWNSDLDXGMGU-UHFFFAOYSA-N; HJBWBXRSRQEPRF-UHFFFAOYSA-N; ICSNLGPSRYBMBD-UHFFFAOYSA-N; IEVUNGKXTAPNJR-UHFFFAOYSA-N; INDAZOLE; ITENFASQOQYRFM-UHFFFAOYSA-N; JADFRCNEVYMOAL-UHFFFAOYSA-N; KGHNKNWLMDRAQN-UHFFFAOYSA-N; KXDAEFPNCMNJSK-UHFFFAOYSA-N; LFUDVFOVNMIIIB-UHFFFAOYSA-N; LONGYNYRAPHNDS-UHFFFAOYSA-N; LOQHWUSEIHJYSE-UHFFFAOYSA-N; MHOUKRXEYUPHQG-UHFFFAOYSA-N; MKOXPFXGJVHBRH-UHFFFAOYSA-N; MMVNARZZQWUGQI-UHFFFAOYSA-N; MZCGMLMIRVVUSZ-UHFFFAOYSA-N; MZWNQLWLROXGST-UHFFFAOYSA-N; NFJFJJLADCFCHO-UHFFFAOYSA-N; NKPNESPVSMHQPA-ZRDIBKRKSA-N; NQRYJNQNLNOLGT-UHFFFAOYSA-N; NXWRCPFWNLSYMG-UHFFFAOYSA-N; PAEYRUAPLGXYIJ-UHFFFAOYSA-N; PLGIFHJDPLCSPL-UHFFFAOYSA-N; POMGSLQHWNDZAP-UHFFFAOYSA-N; PYRAZOLE; QLIZWGWIQMJGMB-UHFFFAOYSA-N; QUINAZOLINE; QXQPWPCSFNZDEU-JLHYYAGUSA-N; RLGJGDBTBWUXKU-UHFFFAOYSA-N; RMGFLMXDCGQKPS-UHFFFAOYSA-N; STGYTXNBWMZKBA-UHFFFAOYSA-N; UBABLIWJMXJJNH-UHFFFAOYSA-N; UPFBAUZYKBLCEO-ZRDIBKRKSA-N; VGLWVBWXBZWXJE-WUKNDPDISA-N; VMNKGGRIISDZAU-UHFFFAOYSA-N; VOISDZHTKJQPAM-UHFFFAOYSA-N; WDWWEAMPRRKLGH-UHFFFAOYSA-N; WGCBFZZUJQDDSF-UHFFFAOYSA-N; WJNQRYCMQPMUDS-PKNBQFBNSA-N; WNRWEBKEQARBKV-UHFFFAOYSA-N; WQMAANNAZKNUDL-UHFFFAOYSA-N; XBPOBCXHALHJFP-UHFFFAOYSA-N; XPAKBGQUORPCMO-PKNBQFBNSA-N; XRWQAJSVMIKRKF-UHFFFAOYSA-N; YNAVUWVOSKDBBP-UHFFFAOYSA-N; YWQRMQADBLJRKZ-UHFFFAOYSA-N; ZVGCJBIDARLIMB-UHFFFAOYSA-N; ZWKKHRLWUFOSPA-UHFFFAOYSA-N; ZXANSLBVWCBHPP-UHFFFAOYSA-N;

ANTITUBERCULAR AGENTS; CELL LINE; HUMANS; INDAZOLES; MYCOBACTERIUM TUBERCULOSIS; PYRAZOLES; PYRIDINES; QUINAZOLINES; TUBERCULOSIS;

EID: 84885171675 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.08.101 Document Type: Article

Times cited : (50)

References (27)

1
- 25844434417
- P. Nunn, B. Williams, K. Floyd, C. Dye, G. Elzinga, and M. Raviglione Nat. Rev. Immunol. 5 2005 819
- (2005) Nat. Rev. Immunol. , vol.5 , pp. 819
- Nunn, P.¹ Williams, B.² Floyd, K.³ Dye, C.⁴ Elzinga, G.⁵ Raviglione, M.⁶

2
- 84885186144
- World Health Organization (WHO) Global Tuberculosis Report 2012
- World Health Organization (WHO) Global Tuberculosis Report 2012.

3
- 0141853344
- T.R. Frieden, T.R. Sterling, S.S. Munsiff, C.J. Watt, and C. Dye Lancet 362 2003 887
- (2003) Lancet , vol.362 , pp. 887
- Frieden, T.R.¹ Sterling, T.R.² Munsiff, S.S.³ Watt, C.J.⁴ Dye, C.⁵

4
- 84874312689
- Accessed November 30, 2009
- Tuberculosis Control-India. Available from: http://www.tbcindia.org. Accessed November 30, 2009.
- Tuberculosis Control-India

5
- 84877665340
- Accessed December 2
- Annual risk of tuberculosis infection in different zones of India. Available from: http://ntiindia.kar.nic.in/docs/ari2000-03/index.html. Accessed December 2, 2009.
- (2009) Annual Risk of Tuberculosis Infection in Different Zones of India

6
- 33847681052
- Y.L. Janin Bioorg. Med. Chem. 15 2007 2479
- (2007) Bioorg. Med. Chem. , vol.15 , pp. 2479
- Janin, Y.L.¹

7
- 84855641071
- C. Brullo, M. Rocca, P. Fossa, E. Cichero, E. Barocelli, V. Ballabeni, L. Flammini, C. Giorgio, F. Saccani, G. Domenichini, and O. Brono Bioorg. Med. Chem. Lett. 22 2012 1125
- (2012) Bioorg. Med. Chem. Lett. , vol.22 , pp. 1125
- Brullo, C.¹ Rocca, M.² Fossa, P.³ Cichero, E.⁴ Barocelli, E.⁵ Ballabeni, V.⁶ Flammini, L.⁷ Giorgio, C.⁸ Saccani, F.⁹ Domenichini, G.¹⁰ Brono, O.¹¹

8
- 84883895968
- N. Chidananda, B. Poojary, V. Sumangala, and N. Kumari Suchetha Ind. J. Heterocycl. Chem. 20 2011 337
- (2011) Ind. J. Heterocycl. Chem. , vol.20 , pp. 337
- Chidananda, N.¹ Poojary, B.² Sumangala, V.³ Kumari Suchetha, N.⁴

9
- 0024848198
- M. Ghannoum, K. Abu Elteen, and N.R. El-Rayyes Microbios 60 1989 23
- (1989) Microbios , vol.60 , pp. 23
- Ghannoum, M.¹ Abu Elteen, K.² El-Rayyes, N.R.³

10
- 79958002291
- S. Eathiraj, R. Palma, M. Hirschi, E. Volckova, E. Nakuci, J. Castro, C.-R. Chen, T.C.K. Chan, D.S. France, and M.A. Ashwell J. Biol. Chem. 286 2011 20677
- (2011) J. Biol. Chem. , vol.286 , pp. 20677
- Eathiraj, S.¹ Palma, R.² Hirschi, M.³ Volckova, E.⁴ Nakuci, E.⁵ Castro, J.⁶ Chen, C.-R.⁷ Chan, T.C.K.⁸ France, D.S.⁹ Ashwell, M.A.¹⁰

11
- 84885184867
- PCT Int. Appl. 2010, WO 2010078229 A1 20100708
- Maddry, J. A.; Severson, W.; Jonsson, C. B.; Noah, J. W.; Noah, D. L.; Chen, X. PCT Int. Appl. 2010, WO 2010078229 A1 20100708.
- Maddry, J.A.¹ Severson, W.² Jonsson, C.B.³ Noah, J.W.⁴ Noah, D.L.⁵ Chen, X.⁶

12
- 84885172354
- PCT Int. Appl. 2010, WO 2010078421 A1 20100708
- Ali, S. M.; Ashwell, M.; Tandon, M.; Yang, R.-Y.; Liu, Y.; Vensel, D.; Eathiraj, S.; Palma, R.; Lapierre, J.-M.; Westlund, N.; Wu, H; Namdev, N.; Kelleher, E; Kelleher, E. PCT Int. Appl. 2010, WO 2010078421 A1 20100708.
- Ali, S.M.¹ Ashwell, M.² Tandon, M.³ Yang, R.-Y.⁴ Liu, Y.⁵ Vensel, D.⁶ Eathiraj, S.⁷ Palma, R.⁸ Lapierre, J.-M.⁹ Westlund, N.¹⁰ Wu, H.¹¹ Namdev, N.¹² Kelleher, E.¹³ Kelleher, E.¹⁴

13
- 84886724398
- J.R. Koenig, H. Liu, I. Drizin, D.G. Witte, T.L. Carr, A.M. Manelli, I. Milicic, M.I. Strakhova, T.R. Miller, T.A. Esbenshade, J.D. Brioni, and M. Cowart Bioorg. Med. Chem. Lett. 2010 1900 20
- (1900) Bioorg. Med. Chem. Lett. , vol.2010 , pp. 20
- Koenig, J.R.¹ Liu, H.² Drizin, I.³ Witte, D.G.⁴ Carr, T.L.⁵ Manelli, A.M.⁶ Milicic, I.⁷ Strakhova, M.I.⁸ Miller, T.R.⁹ Esbenshade, T.A.¹⁰ Brioni, J.D.¹¹ Cowart, M.¹²

14
- 54949125390
- M.D. Cowart, R.J. Altenbach, H. Liu, G.C. Hsieh, I. Drizin, I. Milicic, T.R. Miller, D.G. Witte, N. Wishart, S.R. Fix-Stenzel, M.J. McPherson, R.M. Adair, J.M. Wetter, B.M. Bettencourt, K.C. Marsh, J.P. Sullivan, P. Honore, T.A. Esbenshade, and J.D. Brioni J. Med. Chem. 51 2008 6547
- (2008) J. Med. Chem. , vol.51 , pp. 6547
- Cowart, M.D.¹ Altenbach, R.J.² Liu, H.³ Hsieh, G.C.⁴ Drizin, I.⁵ Milicic, I.⁶ Miller, T.R.⁷ Witte, D.G.⁸ Wishart, N.⁹ Fix-Stenzel, S.R.¹⁰ McPherson, M.J.¹¹ Adair, R.M.¹² Wetter, J.M.¹³ Bettencourt, B.M.¹⁴ Marsh, K.C.¹⁵ Sullivan, J.P.¹⁶ Honore, P.¹⁷ Esbenshade, T.A.¹⁸ Brioni, J.D.¹⁹

15
- 84885179979
- PCT Int. Appl. 2008, WO 2008060767 A2 20080522
- Hancock, A. A.; Altenbach, R. J.; Liu, H.; Drizin, I.; Cowart, M. D.; Wishart, N.; Babinski, D. J.; Gregg, R. J.; Esbenshade, T. A.; Hsieh, G. C.; Brioni, J. D.; Honore, M. P.; Black, L. A.; Zhao, C.; Wakefield, B. D. PCT Int. Appl. 2008, WO 2008060767 A2 20080522.
- Hancock, A.A.¹ Altenbach, R.J.² Liu, H.³ Drizin, I.⁴ Cowart, M.D.⁵ Wishart, N.⁶ Babinski, D.J.⁷ Gregg, R.J.⁸ Esbenshade, T.A.⁹ Hsieh, G.C.¹⁰ Brioni, J.D.¹¹ Honore, M.P.¹² Black, L.A.¹³ Zhao, C.¹⁴ Wakefield, B.D.¹⁵

16
- 84885185739
- PCT Int. Appl. 2009, WO 2009064388 A2 20090522
- Liu, J. O.; Hu, X.; Chen, X.; Ma, D.; Bhat, S. PCT Int. Appl. 2009, WO 2009064388 A2 20090522.
- Liu, J.O.¹ Hu, X.² Chen, X.³ Ma, D.⁴ Bhat, S.⁵

17
- 84885187964
- U.S. 1995, US 5405851 A 19950411
- Pendergast, W.; Dickerson, S. H.; Johnson, J. V.; Ferone, R. U.S. 1995, US 5405851 A 19950411.
- Pendergast, W.¹ Dickerson, S.H.² Johnson, J.V.³ Ferone, R.⁴

18
- 84885176547
- PCT Int. Appl. 1991, WO 9119700 A1 19911226
- Pendergast, W.; Dickerson, S. H.; Johnson, J. V.; Ferone, R. PCT Int. Appl. 1991, WO 9119700 A1 19911226.
- Pendergast, W.¹ Dickerson, S.H.² Johnson, J.V.³ Ferone, R.⁴

19
- 0036170331
- N. Agarwal, P. Srivastava, S.K. Raghuwanshi, D.N. Upadhyay, S. Sinha, P.K. Shukla, and V.J. Ram Bioorg. Med. Chem. 10 2002 869
- (2002) Bioorg. Med. Chem. , vol.10 , pp. 869
- Agarwal, N.¹ Srivastava, P.² Raghuwanshi, S.K.³ Upadhyay, D.N.⁴ Sinha, S.⁵ Shukla, P.K.⁶ Ram, V.J.⁷

20
- 84880117082
- P. Horrocks, M.R. Pickard, H.H. Parekh, S.P. Patel, and V.B. Pathak Org. Biomol. Chem. 11 2013 4891
- (2013) Org. Biomol. Chem. , vol.11 , pp. 4891
- Horrocks, P.¹ Pickard, M.R.² Parekh, H.H.³ Patel, S.P.⁴ Pathak, V.B.⁵

21
- 84873739914
- I. Ahmad, J.P. Thakur, D. Chanda, D. Saikia, F. Khan, S. Dixit, A. Kumar, R. Konwar, A.S. Negi, and A. Gupta Bioorg. Med. Chem. 23 2013 1322
- (2013) Bioorg. Med. Chem. , vol.23 , pp. 1322
- Ahmad, I.¹ Thakur, J.P.² Chanda, D.³ Saikia, D.⁴ Khan, F.⁵ Dixit, S.⁶ Kumar, A.⁷ Konwar, R.⁸ Negi, A.S.⁹ Gupta, A.¹⁰

22
- 84886716881
- S. Velaparthi, M. Brunsteiner, R. Uddin, B. Wan, S.G. Franzblau, and P.A. Petukhov J. Med. Chem. 2008 1999 51
- (1999) J. Med. Chem. , vol.2008 , pp. 51
- Velaparthi, S.¹ Brunsteiner, M.² Uddin, R.³ Wan, B.⁴ Franzblau, S.G.⁵ Petukhov, P.A.⁶

23
- 51449117872
- D. Castagnolo, A.D. Logu, M. Radi, B. Bechi, F. Manetti, M. Magnani, S. Supino, R. Meleddu, L. Chisu, and M. Botta Bioorg. Med. Chem. 16 2008 8587
- (2008) Bioorg. Med. Chem. , vol.16 , pp. 8587
- Castagnolo, D.¹ Logu, A.D.² Radi, M.³ Bechi, B.⁴ Manetti, F.⁵ Magnani, M.⁶ Supino, S.⁷ Meleddu, R.⁸ Chisu, L.⁹ Botta, M.¹⁰

24
- 84885190750
- WO 2012049161 A1
- Castro, P. J.; Fernandez, M. R.; Fernandez, V. E. P.; Gonzalez, D. V. S.; Mallo-Rubio, A. WO 2012049161 A1, 2012.
- (2012)
- Castro, P.J.¹ Fernandez, M.R.² Fernandez, V.E.P.³ Gonzalez, D.V.S.⁴ Mallo-Rubio, A.⁵

25
- 84880542677
- H.K. Maurya, P.G. Vasudev, and A. Gupta RSC Adv. 3 2013 12955
- (2013) RSC Adv. , vol.3 , pp. 12955
- Maurya, H.K.¹ Vasudev, P.G.² Gupta, A.³

26
- 84880606283
- P. Mishra, S. Kumar, H.K. Maurya, S.K. Gautam, B. Kumar, V.K. Tandon, and V.J. Ram Heterocycles 82 2012 189
- (2012) Heterocycles , vol.82 , pp. 189
- Mishra, P.¹ Kumar, S.² Maurya, H.K.³ Gautam, S.K.⁴ Kumar, B.⁵ Tandon, V.K.⁶ Ram, V.J.⁷

27
- 3242782912
- V.J. Ram, M. Verma, F.A. Hussaini, and A. Shoeb Chem. Res. (S) 1991 98 Technology
- (1991) Chem. Res. (S) , pp. 98
- Ram, V.J.¹ Verma, M.² Hussaini, F.A.³ Shoeb, A.⁴

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