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Volumn 23, Issue 20, 2013, Pages 5740-5743
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Discovery of thiazolyl-phthalazinone acetamides as potent glucose uptake activators via high-throughput screening
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Author keywords
Glucose uptake activators; Obesity; PPAR ; Thiazolyl phthalazinone acetamides; Type 2 diabetes
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Indexed keywords
ACETAMIDE DERIVATIVE;
ADIPIC ACID;
ANTIDIABETIC AGENT;
GLUCOSE;
HETEROCYCLIC AMINE;
HYDRAZINE;
INSULIN;
PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA AGONIST;
ROSIGLITAZONE;
THIAZOLYL PHTHALAZINONE ACETAMIDE;
UNCLASSIFIED DRUG;
ANTIDIABETIC ACTIVITY;
ARTICLE;
BIOLOGICAL ACTIVITY;
DOSE RESPONSE;
DRUG SYNTHESIS;
GLUCOSE TRANSPORT;
HIGH THROUGHPUT SCREENING;
MUSCLE CELL;
SKELETAL MUSCLE;
STRUCTURE ACTIVITY RELATION;
GLUCOSE UPTAKE ACTIVATORS;
OBESITY;
PPAR-Γ;
THIAZOLYL-PHTHALAZINONE ACETAMIDES;
TYPE 2 DIABETES;
ACETAMIDES;
ANIMALS;
CELL LINE;
CERCOPITHECUS AETHIOPS;
DRUG EVALUATION, PRECLINICAL;
GLUCOSE;
HIGH-THROUGHPUT SCREENING ASSAYS;
HUMANS;
HYPOGLYCEMIC AGENTS;
INSULIN;
MUSCLE, SKELETAL;
PHTHALAZINES;
PPAR GAMMA;
STRUCTURE-ACTIVITY RELATIONSHIP;
THIAZOLES;
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EID: 84884280908
PISSN: 0960894X
EISSN: 14643405
Source Type: Journal
DOI: 10.1016/j.bmcl.2013.07.067 Document Type: Article |
Times cited : (15)
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References (8)
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