De novo tyrosinase inhibitor: 4-(6,7-Dihydro-5H-indeno[5,6-d]thiazol-2-yl) benzene-1,3-diol (MHY1556)

Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 14, 2013, Pages 4172-4176

  Park, June Whan ^a   Ha, Young Mi ^b   Moon, Kyung Mi ^a   Kim, So Ra ^a   Jeong, Hyoung Oh ^a   Park, Yun Jung ^a   Lee, Hye Jin ^a   Park, Ji Young ^a   Song, Yu Min ^a   Chun, Pusoon ^c   Byun, Youngjoo ^d   Moon, Hyung Ryong ^a   Chung, Hae Young ^a  

^a Pusan National University   (South Korea)

^b Dong A University   (South Korea)

^c Inje University   (South Korea)

^d Korea University   (South Korea)

Author keywords

Kojic acid; Melanogenesis; Skin whitening product; Tyrosinase inhibitor 4 (6,7 Dihydro 5H indeno 5,6 d thiazol 2 yl)benzene 1,3 diol

Indexed keywords

4 (6,7 DIHYDRO 5H INDENO[5,6 D] THIAZOL 2 YL)BENZENE 1,3 DIOL; AMINO ACID; COSMETIC; KOJIC ACID; MHY 1556; OXYGENASE INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL STRUCTURE; HYDROGEN BOND; IC 50; IN VITRO STUDY; MELANOGENESIS; MELANOMA CELL; SYNTHESIS;

AGARICALES; ANIMALS; BENZOTHIAZOLES; BINDING SITES; CELL LINE, TUMOR; CELL SURVIVAL; ENZYME INHIBITORS; MICE; MOLECULAR DOCKING SIMULATION; MONOPHENOL MONOOXYGENASE; PROTEIN BINDING; PROTEIN STRUCTURE, TERTIARY; PYRONES; RESORCINOLS;

BASIDIOMYCOTA;

EID: 84879415446     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2013.05.029     Document Type: Article

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