메뉴 건너뛰기




Volumn 84, Issue 3, 2013, Pages 449-455

The transdermal delivery of fentanyl

Author keywords

Fentanyl; Matrix; Pharmacokinetics; Reservoir; Transdermal patch

Indexed keywords

ADHESIVE AGENT; ALCOHOL; ALOE VERA EXTRACT; DESPROPIONYLFENTANYL; DRUG METABOLITE; DUROGESIC DTRANS; ETHYLENE VINYL ACETATE COPOLYMER; FENCINO; FENTALIS; FENTANYL; HYDROXYETHYLCELLULOSE; HYDROXYFENTANYL; HYDROXYNORFENTANYL; MATRIFEN; MORPHINE; NORFENTANYL; PETHIDINE; POLYMER; PROPYLENE GLYCOL; ROSIN; SILICONE; UNCLASSIFIED DRUG;

EID: 84879114355     PISSN: 09396411     EISSN: 18733441     Source Type: Journal    
DOI: 10.1016/j.ejpb.2013.01.018     Document Type: Review
Times cited : (57)

References (46)
  • 1
    • 0000060541 scopus 로고
    • A review of the chemical features associated with strong morphine-likeactivity
    • P.A. Janssen A review of the chemical features associated with strong morphine-likeactivity Br. J. Anaesth. 34 1962 260 268
    • (1962) Br. J. Anaesth. , vol.34 , pp. 260-268
    • Janssen, P.A.1
  • 2
    • 10644239664 scopus 로고    scopus 로고
    • A.C. Moffat, M.D. Osselton, B. Widdop, 3rd ed. The Pharmaceutical Press London, United Kingdom
    • Fentanyl A.C. Moffat, M.D. Osselton, B. Widdop, Clarke's Analysis of Drugs and Poisons 3rd ed. 2004 The Pharmaceutical Press London, United Kingdom 1029 1030
    • (2004) Clarke's Analysis of Drugs and Poisons , pp. 1029-1030
    • Fentanyl1
  • 3
    • 0020508539 scopus 로고
    • Clinical pharmacokinetics of fentanyl and its newer derivatives
    • L.E. Mather Clinical pharmacokinetics of fentanyl and its newer derivatives Clin. Pharmacokinet. 8 1983 422 446
    • (1983) Clin. Pharmacokinet. , vol.8 , pp. 422-446
    • Mather, L.E.1
  • 4
    • 0242504308 scopus 로고
    • Origin and rationale of neurolept analgesia
    • E. Nilsson Origin and rationale of neurolept analgesia Anaesthesiology 24 1963 267 268
    • (1963) Anaesthesiology , vol.24 , pp. 267-268
    • Nilsson, E.1
  • 5
    • 0018840881 scopus 로고
    • The role of diazepam and fentanyl in the production of balanced anaesthesia
    • U. Aromaa, K. Korttila, and T. Tammisto The role of diazepam and fentanyl in the production of balanced anaesthesia Acta Anaesthesiol. Scand. 24 1980 36 40
    • (1980) Acta Anaesthesiol. Scand. , vol.24 , pp. 36-40
    • Aromaa, U.1    Korttila, K.2    Tammisto, T.3
  • 6
    • 0018906382 scopus 로고
    • The role of thiopental and fentanyl in the production of balanced anaesthesia
    • T. Tammisto, U. Aromaa, and K. Korttila The role of thiopental and fentanyl in the production of balanced anaesthesia Acta Anaesthesiol. Scand. 24 1980 31 35
    • (1980) Acta Anaesthesiol. Scand. , vol.24 , pp. 31-35
    • Tammisto, T.1    Aromaa, U.2    Korttila, K.3
  • 7
    • 0016545625 scopus 로고
    • Drug permeation through human skin: Theory and in vitro experimental measurement
    • A.S. Michaels, S.K. Chandrasekaran, and J.E. Shaw Drug permeation through human skin: theory and in vitro experimental measurement AIChE J. 21 1975 985 996
    • (1975) AIChE J. , vol.21 , pp. 985-996
    • Michaels, A.S.1    Chandrasekaran, S.K.2    Shaw, J.E.3
  • 8
    • 0006617311 scopus 로고
    • Pharmacokinetics and dynamics of narcotic analgesics
    • C. Prys-Roberts, C.C. Hug, Blackwell Oxford
    • C.C. Hug Pharmacokinetics and dynamics of narcotic analgesics C. Prys-Roberts, C.C. Hug, Pharmacokinetics of Anaesthesia 1984 Blackwell Oxford 187 234
    • (1984) Pharmacokinetics of Anaesthesia , pp. 187-234
    • Hug, C.C.1
  • 10
    • 0030041685 scopus 로고    scopus 로고
    • Identification of human liver cytochrome P-450 3A4 as the enzyme responsible for fentanyl and sufentanil N-dealkylation
    • T. Tateishi, Y. Krivoruk, Y.-F. Ueng, A.J.J. Wood, F.P. Guengerich, and M. Wood Identification of human liver cytochrome P-450 3A4 as the enzyme responsible for fentanyl and sufentanil N-dealkylation Anest. Analg. 82 1996 167 172
    • (1996) Anest. Analg. , vol.82 , pp. 167-172
    • Tateishi, T.1    Krivoruk, Y.2    Ueng, Y.-F.3    Wood, A.J.J.4    Guengerich, F.P.5    Wood, M.6
  • 11
    • 0021152878 scopus 로고
    • Identification and quantitative determination of fentanyl metabolites in patients by gas chromatography-mass spectrometry
    • T. Goromaru, H. Matsuraa, N. Yoshimura, T. Miyawaki, T. Sameshima, J. Miyao, T. Furuta, and S. Baba Identification and quantitative determination of fentanyl metabolites in patients by gas chromatography-mass spectrometry Anesthesiology 61 1984 73 77
    • (1984) Anesthesiology , vol.61 , pp. 73-77
    • Goromaru, T.1    Matsuraa, H.2    Yoshimura, N.3    Miyawaki, T.4    Sameshima, T.5    Miyao, J.6    Furuta, T.7    Baba, S.8
  • 12
    • 0019829884 scopus 로고
    • The assay of fentanyl and its metabolites in plasma of patients using gas chromatography with alkali flame ionisation detection and gas chromatography-mass spectrometry
    • H.H. Van Rooy, M.P. Vermeulen, and J.G. Bovill The assay of fentanyl and its metabolites in plasma of patients using gas chromatography with alkali flame ionisation detection and gas chromatography-mass spectrometry J. Chromatogr. 223 1981 85 93
    • (1981) J. Chromatogr. , vol.223 , pp. 85-93
    • Van Rooy, H.H.1    Vermeulen, M.P.2    Bovill, J.G.3
  • 13
    • 0027476762 scopus 로고
    • An analysis of the duration of fentanyl and its metabolites in urine and saliva
    • J.H. Silverstein, M.F. Rieders, M. McMullin, S. Schulman, and K. Zahl An analysis of the duration of fentanyl and its metabolites in urine and saliva Anesth. Analg. 76 1993 618 621
    • (1993) Anesth. Analg. , vol.76 , pp. 618-621
    • Silverstein, J.H.1    Rieders, M.F.2    McMullin, M.3    Schulman, S.4    Zahl, K.5
  • 14
    • 0019063415 scopus 로고
    • Analgesic plasma concentrations
    • 52-52
    • R.F. Cookson Analgesic plasma concentrations Br. J. Anaesth. 52 1980 52-52
    • (1980) Br. J. Anaesth. , vol.52
    • Cookson, R.F.1
  • 15
    • 0018776545 scopus 로고
    • Postoperative analgesia: A comparison of intravenous on-demand fentanyl with epidural bupivacaine
    • W.D. White, D.J. Pearce, and J. Norman Postoperative analgesia: a comparison of intravenous on-demand fentanyl with epidural bupivacaine Br. Med. J. 2 1979 166 167
    • (1979) Br. Med. J. , vol.2 , pp. 166-167
    • White, W.D.1    Pearce, D.J.2    Norman, J.3
  • 16
    • 0018872478 scopus 로고
    • Analgesic action of extradural fentanyl
    • M.J. Wolfe, and G.K. Davies Analgesic action of extradural fentanyl Br. J. Anaesth. 52 1980 357 358
    • (1980) Br. J. Anaesth. , vol.52 , pp. 357-358
    • Wolfe, M.J.1    Davies, G.K.2
  • 17
    • 0012788682 scopus 로고
    • Opioids and adjuvants: Principles of use
    • M.J. Cousins, G.D. Phillips, Churchill Livingstone New York
    • L.E. Mather, and G.D. Phillips Opioids and adjuvants: principles of use M.J. Cousins, G.D. Phillips, Acute Pain Management 1986 Churchill Livingstone New York 77 103
    • (1986) Acute Pain Management , pp. 77-103
    • Mather, L.E.1    Phillips, G.D.2
  • 18
    • 0023791101 scopus 로고
    • Solubility and related physicochemical properties of narcotic analgesics
    • S.D. Roy, and G.L. Flynn Solubility and related physicochemical properties of narcotic analgesics Pharm. Res. 5 1988 580 586
    • (1988) Pharm. Res. , vol.5 , pp. 580-586
    • Roy, S.D.1    Flynn, G.L.2
  • 19
    • 0024510075 scopus 로고
    • Solubility behavior of narcotic analgesics in aqueous media: Solubilities and dissociation constants of morphine, fentanyl, and sufentanil
    • S.D. Roy, and G.L. Flynn Solubility behavior of narcotic analgesics in aqueous media: solubilities and dissociation constants of morphine, fentanyl, and sufentanil Pharm. Res. 6 1989 147 151
    • (1989) Pharm. Res. , vol.6 , pp. 147-151
    • Roy, S.D.1    Flynn, G.L.2
  • 20
    • 0024347402 scopus 로고
    • Transdermal delivery of narcotic analgesics: Comparative permeabilities of narcotic analgesics through human cadaver skin
    • S.D. Roy, and G.L. Flynn Transdermal delivery of narcotic analgesics: comparative permeabilities of narcotic analgesics through human cadaver skin Pharm. Res. 6 1989 825 832
    • (1989) Pharm. Res. , vol.6 , pp. 825-832
    • Roy, S.D.1    Flynn, G.L.2
  • 21
    • 0001089725 scopus 로고
    • The process of diffusion through a rubber membrane
    • H.A. Daynes The process of diffusion through a rubber membrane Proc. Roy. Soc. Ser. A 97 1920 286 307
    • (1920) Proc. Roy. Soc. Ser. A , vol.97 , pp. 286-307
    • Daynes, H.A.1
  • 22
    • 37049166629 scopus 로고
    • Permeation, diffusion and solution of gases in organic polymers
    • R.M. Barrer, and E.K. Rideal Permeation, diffusion and solution of gases in organic polymers Trans. Faraday Soc. 35 1939 628
    • (1939) Trans. Faraday Soc. , vol.35 , pp. 628
    • Barrer, R.M.1    Rideal, E.K.2
  • 23
    • 0025000624 scopus 로고
    • Transdermal delivery of narcotic analgesics: PH, anatomical, and subject influences on cutaneous permeability of fentanyl and sufentanil
    • S.D. Roy, and G.L. Flynn Transdermal delivery of narcotic analgesics: pH, anatomical, and subject influences on cutaneous permeability of fentanyl and sufentanil Pharm. Res. 7 1990 842 847
    • (1990) Pharm. Res. , vol.7 , pp. 842-847
    • Roy, S.D.1    Flynn, G.L.2
  • 24
    • 0023935630 scopus 로고
    • Plasma fentanyl concentrations during transdermal delivery of fentanyl to surgical patients
    • D.J. Duthie, D.J. Rowbotham, R. Wyld, P.D. Henderson, and W.S. Nimmo Plasma fentanyl concentrations during transdermal delivery of fentanyl to surgical patients Br. J. Anaesth. 60 1988 614 618
    • (1988) Br. J. Anaesth. , vol.60 , pp. 614-618
    • Duthie, D.J.1    Rowbotham, D.J.2    Wyld, R.3    Henderson, P.D.4    Nimmo, W.S.5
  • 25
    • 0023877926 scopus 로고
    • Postoperative analgesia with fentanyl: Pharmacokinetics and pharmacodynamics of constant-rate I.V. and transdermal delivery
    • F.O. Holley, and C. van Steenis Postoperative analgesia with fentanyl: pharmacokinetics and pharmacodynamics of constant-rate I.V. and transdermal delivery Br. J. Anaesth. 60 1988 608 613
    • (1988) Br. J. Anaesth. , vol.60 , pp. 608-613
    • Holley, F.O.1    Van Steenis, C.2
  • 27
    • 0026521395 scopus 로고
    • System functionality and physicochemical model of fentanyl transdermal system
    • S.K. Gupta, M. Southam, R. Gale, and S.S. Hwang System functionality and physicochemical model of fentanyl transdermal system J. Pain Symptom Manage. 7 1992 S17 S26
    • (1992) J. Pain Symptom Manage. , vol.7
    • Gupta, S.K.1    Southam, M.2    Gale, R.3    Hwang, S.S.4
  • 29
    • 0000651234 scopus 로고    scopus 로고
    • Assessing the impact of heat on the systemic delivery of fentanyl through the transdermal fentanyl delivery system
    • T.S. Shomaker, J. Zhang, and M.A. Ashburn Assessing the impact of heat on the systemic delivery of fentanyl through the transdermal fentanyl delivery system Pain Med. 1 2000 225 230
    • (2000) Pain Med. , vol.1 , pp. 225-230
    • Shomaker, T.S.1    Zhang, J.2    Ashburn, M.A.3
  • 30
    • 0041469971 scopus 로고    scopus 로고
    • The pharmacokinetics of transdermal fentanyl delivered with and without controlled heat
    • M.A. Ashburn, L.L. Ogden, J. Zhang, G. Love, and S.V. Basta The pharmacokinetics of transdermal fentanyl delivered with and without controlled heat J. Pain. 4 2003 291 297
    • (2003) J. Pain. , vol.4 , pp. 291-297
    • Ashburn, M.A.1    Ogden, L.L.2    Zhang, J.3    Love, G.4    Basta, S.V.5
  • 32
    • 56449126995 scopus 로고    scopus 로고
    • Fentanyl post-mortem redistribution: Preliminary findings regarding the relationship among femoral blood and liver and heart tissue concentrations
    • K. Luckenbill, J. Thompson, O. Middleton, J. Kloss, and F. Apple Fentanyl post-mortem redistribution: preliminary findings regarding the relationship among femoral blood and liver and heart tissue concentrations J. Anal. Toxicol. 32 2008 639 643
    • (2008) J. Anal. Toxicol. , vol.32 , pp. 639-643
    • Luckenbill, K.1    Thompson, J.2    Middleton, O.3    Kloss, J.4    Apple, F.5
  • 35
    • 84859745649 scopus 로고    scopus 로고
    • Toxicological implications of the delivery of fentanyl from gel extracted from a commercial transdermal reservoir patch
    • G. Oliveira, J. Hadgraft, and M.E. Lane Toxicological implications of the delivery of fentanyl from gel extracted from a commercial transdermal reservoir patch Toxicol. in Vitro. 26 2012 645 648
    • (2012) Toxicol. in Vitro. , vol.26 , pp. 645-648
    • Oliveira, G.1    Hadgraft, J.2    Lane, M.E.3
  • 36
    • 0029875895 scopus 로고    scopus 로고
    • Controlled transdermal delivery of fentanyl: Characterizations of pressure-sensitive adhesives for matrix patch design
    • S.D. Roy, M. Gutierrez, G.L. Flynn, and G.W. Cleary Controlled transdermal delivery of fentanyl: characterizations of pressure-sensitive adhesives for matrix patch design J. Pharm. Sci. 85 1996 491 495
    • (1996) J. Pharm. Sci. , vol.85 , pp. 491-495
    • Roy, S.D.1    Gutierrez, M.2    Flynn, G.L.3    Cleary, G.W.4
  • 39
    • 29144442167 scopus 로고    scopus 로고
    • Evaluation of the bioequivalence of two transdermal fentanyl systems following single and repeat applications
    • G. Sathyan, C. Guo, K. Sivakumar, S. Gidwani, and S. Gupta Evaluation of the bioequivalence of two transdermal fentanyl systems following single and repeat applications Curr. Med. Res. Opin. 21 2005 1961 1968
    • (2005) Curr. Med. Res. Opin. , vol.21 , pp. 1961-1968
    • Sathyan, G.1    Guo, C.2    Sivakumar, K.3    Gidwani, S.4    Gupta, S.5
  • 40
    • 79955937048 scopus 로고    scopus 로고
    • Bioequivalence and safety of a novel fentanyl transdermal matrix system compared with a transdermal reservoir system
    • K.T. Moore, H.D. Adams, J. Natarajan, J. Ariyawansa, and H.M. Richards Bioequivalence and safety of a novel fentanyl transdermal matrix system compared with a transdermal reservoir system J. Opioid Manage. 7 2011 99 107
    • (2011) J. Opioid Manage. , vol.7 , pp. 99-107
    • Moore, K.T.1    Adams, H.D.2    Natarajan, J.3    Ariyawansa, J.4    Richards, H.M.5
  • 41
    • 84864416378 scopus 로고    scopus 로고
    • Randomized 5-treatment crossover study to assess the effects of external heat on serumfentanyl concentrations during treatment with transdermal fentanyl systems
    • K.T. Moore, G. Sathyan, U. Richarz, J. Natarajan, and J. Vandenbossche Randomized 5-treatment crossover study to assess the effects of external heat on serumfentanyl concentrations during treatment with transdermal fentanyl systems J. Clin. Pharmacol. 52 2012 1174 1185
    • (2012) J. Clin. Pharmacol. , vol.52 , pp. 1174-1185
    • Moore, K.T.1    Sathyan, G.2    Richarz, U.3    Natarajan, J.4    Vandenbossche, J.5
  • 42
    • 51449109808 scopus 로고    scopus 로고
    • Transdermal matrix fentanyl membrane patch (matrifen): In severe cancer-related chronic pain
    • P.I. Hair, G.M. Keating, and K. McKeage Transdermal matrix fentanyl membrane patch (matrifen): in severe cancer-related chronic pain Drugs 68 2008 2001 2009
    • (2008) Drugs , vol.68 , pp. 2001-2009
    • Hair, P.I.1    Keating, G.M.2    McKeage, K.3
  • 43
    • 0035834196 scopus 로고    scopus 로고
    • In vitro study of low-frequency ultrasound-enhanced transdermal transport of fentanyl and caffeine across human and hairless rat skin
    • A. Boucaud, L. Machet, B. Arbeille, M.C. Machet, M. Sournac, A. Mavon, F. Patat, and L. Vaillant In vitro study of low-frequency ultrasound-enhanced transdermal transport of fentanyl and caffeine across human and hairless rat skin Int. J. Pharm. 228 2001 69 77
    • (2001) Int. J. Pharm. , vol.228 , pp. 69-77
    • Boucaud, A.1    Machet, L.2    Arbeille, B.3    Machet, M.C.4    Sournac, M.5    Mavon, A.6    Patat, F.7    Vaillant, L.8
  • 44
    • 80051789757 scopus 로고    scopus 로고
    • Formulation issues associated with transdermal fentanyl delivery
    • P. Santos, A.C. Watkinson, J. Hadgraft, and M.E. Lane Formulation issues associated with transdermal fentanyl delivery Int. J. Pharm. 416 2011 155 159
    • (2011) Int. J. Pharm. , vol.416 , pp. 155-159
    • Santos, P.1    Watkinson, A.C.2    Hadgraft, J.3    Lane, M.E.4
  • 45
    • 82255179362 scopus 로고    scopus 로고
    • Transdermal delivery using a novel electrochemical device, Part 1: Device design and in vitro release/permeation of fentanyl
    • B. Schröder, U. Nickel, E. Meye, and G. Lee Transdermal delivery using a novel electrochemical device, Part 1: Device design and in vitro release/permeation of fentanyl J. Pharm. Sci. 101 2012 245 255
    • (2012) J. Pharm. Sci. , vol.101 , pp. 245-255
    • Schröder, B.1    Nickel, U.2    Meye, E.3    Lee, G.4
  • 46
    • 84859738752 scopus 로고    scopus 로고
    • Transdermal delivery using a novel electrochemical device, Part 2: In vivo study in humans
    • B. Schröder, U. Nickel, E. Meye, and G. Lee Transdermal delivery using a novel electrochemical device, Part 2: In vivo study in humans J. Pharm. Sci. 101 2012 2262 2268
    • (2012) J. Pharm. Sci. , vol.101 , pp. 2262-2268
    • Schröder, B.1    Nickel, U.2    Meye, E.3    Lee, G.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.