메뉴 건너뛰기




Volumn 9, Issue 2, 2013, Pages 211-220

A method to prepare solid lipid nanoparticles with improved entrapment efficiency of hydrophilic drugs

Author keywords

Entrapment efficiency; Excipient selection; Isoniazid; Lipid combination; Solid lipid nanoparticle

Indexed keywords

ENTRAPMENT EFFICIENCY; EXCIPIENT SELECTION; FAVORABLE INTERACTIONS; GLYCERYL MONOSTEARATE; ISONIAZID; METHODS AND MATERIALS; SOLID LIPID NANOPARTICLE (SLN); SOLID LIPID NANOPARTICLES;

EID: 84878649087     PISSN: 15734137     EISSN: 18756786     Source Type: Journal    
DOI: 10.2174/1573413711309020008     Document Type: Article
Times cited : (69)

References (47)
  • 1
    • 0042918919 scopus 로고
    • Solid lipid nanoparticles (SLN)-an alternative parenteral drug carrier system
    • Lucks, J.S.; Müller, R.H.; Konig, B. Solid lipid nanoparticles (SLN)-an alternative parenteral drug carrier system. Eur. J. Pharm. Biopharm., 1992, 38, 33S.
    • (1992) Eur. J. Pharm. Biopharm , vol.38
    • Lucks, J.S.1    Müller, R.H.2    Konig, B.3
  • 2
    • 28744441355 scopus 로고    scopus 로고
    • Preparation and Characterization of Nano-Liposomes Using Phosphatidylcholine
    • Kang, K.C.; Lee, C.I.; Pyo, H.B.; Jeong, N.H. Preparation and Characterization of Nano-Liposomes Using Phosphatidylcholine. J. Ind. Eng. Chem., 2005, 11, 847-851.
    • (2005) J. Ind. Eng. Chem , vol.11 , pp. 847-851
    • Kang, K.C.1    Lee, C.I.2    Pyo, H.B.3    Jeong, N.H.4
  • 3
    • 0028285718 scopus 로고
    • Solid lipid nanoparticles for controlled drug delivery. I. Production, characterization and sterlization
    • Schwarz, C.; Mehnert, W.; Lucks, JS.; Muller, RH. Solid lipid nanoparticles for controlled drug delivery. I. Production, characterization and sterlization. J. Control Release, 1994, 30, 83-96.
    • (1994) J. Control Release , vol.30 , pp. 83-96
    • Schwarz, C.1    Mehnert, W.2    Lucks, J.S.3    Muller, R.H.4
  • 4
    • 71549120801 scopus 로고    scopus 로고
    • Preparation and characterization of bis-ethylhexyloxyphenolmethoxyphenyltriazine (BEMT) loaded solid lipid nano-particles (SLN)
    • Lee, G.S.; Lee, D.H.; Kang, K.C.; Lee, C.I.; Pyo, H.B.; Choi, T.B. Preparation and characterization of bis-ethylhexyloxyphenolmethoxyphenyltriazine (BEMT) loaded solid lipid nano-particles (SLN). J. Ind. Eng. Chem., 2007, 13, 1180-1187.
    • (2007) J. Ind. Eng. Chem , vol.13 , pp. 1180-1187
    • Lee, G.S.1    Lee, D.H.2    Kang, K.C.3    Lee, C.I.4    Pyo, H.B.5    Choi, T.B.6
  • 5
    • 67349126442 scopus 로고    scopus 로고
    • Stability of oil-in-water emulsions prepared using the phase inversion composition method
    • Yang, H.J.; Cho, W.G.; Park, S.N. Stability of oil-in-water emulsions prepared using the phase inversion composition method. J. Ind. Eng. Chem., 2009, 15, 331.
    • (2009) J. Ind. Eng. Chem , vol.15 , pp. 331
    • Yang, H.J.1    Cho, W.G.2    Park, S.N.3
  • 6
    • 41449091856 scopus 로고    scopus 로고
    • Potential of solid lipid nanoparticles in brain targeting
    • Kaur, I.P.; Bhandari, R.; Bhandari, S.; Kakkar, V. Potential of solid lipid nanoparticles in brain targeting. J. Control Release, 2008, 127, 97-109.
    • (2008) J. Control Release , vol.127 , pp. 97-109
    • Kaur, I.P.1    Bhandari, R.2    Bhandari, S.3    Kakkar, V.4
  • 7
    • 0036153211 scopus 로고    scopus 로고
    • Medium scale production of solid lipid nanoparticles (SLN) by high pressure homogenization
    • Jenning, V.; Lippacher, A.; Gohla, SH. Medium scale production of solid lipid nanoparticles (SLN) by high pressure homogenization. J. Microencapsul, 2002, 19, 1-10.
    • (2002) J. Microencapsul , vol.19 , pp. 1-10
    • Jenning, V.1    Lippacher, A.2    Gohla, S.H.3
  • 8
    • 0034032145 scopus 로고    scopus 로고
    • Preparation and characterization of solid lipid nanospheres containing paclitaxel
    • Cavalli, R.; Caputo, O.; Gasco, M.R. Preparation and characterization of solid lipid nanospheres containing paclitaxel. Eur. J. Pharm. Biopharm., 2000, 10, 305-330.
    • (2000) Eur. J. Pharm. Biopharm , vol.10 , pp. 305-330
    • Cavalli, R.1    Caputo, O.2    Gasco, M.R.3
  • 9
    • 0030944482 scopus 로고    scopus 로고
    • Peptide-loaded solid lipid nanoparticles (SLN): Influence of production parameters
    • Almeida, A.J.; Runge, S.; Miiller, R.H. Peptide-loaded solid lipid nanoparticles (SLN): Influence of production parameters. Int. J. Pharm., 1997, 149, 255-265.
    • (1997) Int. J. Pharm , vol.149 , pp. 255-265
    • Almeida, A.J.1    Runge, S.2    Miiller, R.H.3
  • 10
    • 39049139244 scopus 로고    scopus 로고
    • Lipid carriers: A versatile delivery vehicle for proteins and peptides
    • Rawat, M.; Manju, S.; Singh, D.; Saraf, S. Lipid carriers: a versatile delivery vehicle for proteins and peptides. Yakugaku Zasshi, 2008, 128, 269-280.
    • (2008) Yakugaku Zasshi , vol.128 , pp. 269-280
    • Rawat, M.1    Manju, S.2    Singh, D.3    Saraf, S.4
  • 11
    • 0030866983 scopus 로고    scopus 로고
    • Physicochemical characterization of lipid nanoparticles and evaluation of their drug loading capacity and sustained release potential
    • Westesen, K.; Bunjas, H.; Koch, M.H.J. Physicochemical characterization of lipid nanoparticles and evaluation of their drug loading capacity and sustained release potential. J. Control Release, 1997, 48, 223-236.
    • (1997) J. Control Release , vol.48 , pp. 223-236
    • Westesen, K.1    Bunjas, H.2    Koch, M.H.J.3
  • 12
    • 10044223246 scopus 로고    scopus 로고
    • Solid lipid Nanoparticles. (SLNs) to improve oral bioavaility of poorly soluble drug
    • Hu, L.; Tang, X.; Cui, F. Solid lipid Nanoparticles. (SLNs) to improve oral bioavaility of poorly soluble drug. J. Pharm. Pharmacol., 2004, 56, 1527-1535.
    • (2004) J. Pharm. Pharmacol , vol.56 , pp. 1527-1535
    • Hu, L.1    Tang, X.2    Cui, F.3
  • 13
    • 7444255422 scopus 로고    scopus 로고
    • Altered chemical and biological activities of alltrans retinoic acid incorporated in solid lipid nanoparticle powders
    • Lim, S.; Lee, M.; Kim, C. Altered chemical and biological activities of alltrans retinoic acid incorporated in solid lipid nanoparticle powders. J. Control Release, 2004, 100, 53-61.
    • (2004) J. Control Release , vol.100 , pp. 53-61
    • Lim, S.1    Lee, M.2    Kim, C.3
  • 14
    • 2942518501 scopus 로고    scopus 로고
    • Transfection with different colloidal systems: Comparison of solid lipid nanoparticles and liposomes
    • Tabatt, K.; Kneuer, C.; Sameti, M.; Olbrich, C.; Müller, R.H.; Lehr, C.M.; Bakowsky, U. Transfection with different colloidal systems: comparison of solid lipid nanoparticles and liposomes. J. Control Release, 2004, 97, 321-332.
    • (2004) J. Control Release , vol.97 , pp. 321-332
    • Tabatt, K.1    Kneuer, C.2    Sameti, M.3    Olbrich, C.4    Müller, R.H.5    Lehr, C.M.6    Bakowsky, U.7
  • 15
    • 0036130944 scopus 로고    scopus 로고
    • Production of lipospheres as carriers for bioactive compounds
    • Cortesi, R.; Esposito, E.; Luca, G.; Nastruzzi, C. Production of lipospheres as carriers for bioactive compounds. Biomaterials, 2002, 23, 2283-2294.
    • (2002) Biomaterials , vol.23 , pp. 2283-2294
    • Cortesi, R.1    Esposito, E.2    Luca, G.3    Nastruzzi, C.4
  • 16
    • 2142812902 scopus 로고    scopus 로고
    • Lipid-drug conjugate nanoparticles of the hydrophilic drug diminazene-cytotoxicity testing and mouse serum adsorption
    • Olbrich, C.; Gessner, A.; Schröder, W.; Kayser, O.; Müller, R.H. Lipid-drug conjugate nanoparticles of the hydrophilic drug diminazene-cytotoxicity testing and mouse serum adsorption. J. Control Release, 2004, 96, 425-435.
    • (2004) J. Control Release , vol.96 , pp. 425-435
    • Olbrich, C.1    Gessner, A.2    Schröder, W.3    Kayser, O.4    Müller, R.H.5
  • 17
    • 34447259574 scopus 로고    scopus 로고
    • Solid lipid nanoparticles loaded with insulin by sodium cholate-phosphatidylcholinebased mixed micelles: Preparation and characterization
    • Jie, L.; Tao, G.; Changguang, W.; Zhirong, Z.; Zhirong, Z. Solid lipid nanoparticles loaded with insulin by sodium cholate-phosphatidylcholinebased mixed micelles: preparation and characterization. Int. J. Pharm., 2007, 340, 153-162.
    • (2007) Int. J. Pharm , vol.340 , pp. 153-162
    • Jie, L.1    Tao, G.2    Changguang, W.3    Zhirong, Z.4    Zhirong, Z.5
  • 19
    • 0035850227 scopus 로고    scopus 로고
    • Lipid microparticles as a parenteral controlled release device for peptides
    • Reithmeier, H.; Herrmann, J.; Gopferich, A. Lipid microparticles as a parenteral controlled release device for peptides. J. Control Release, 2001, 73, 339-350.
    • (2001) J. Control Release , vol.73 , pp. 339-350
    • Reithmeier, H.1    Herrmann, J.2    Gopferich, A.3
  • 20
    • 77951710606 scopus 로고    scopus 로고
    • Formulation and evaluation of solid lipid nanoparticles of a water soluble drug: Zidovudine
    • Singh, S.; Dobhal, A.K.; Jain, A.; Pandit, J.K.; Chakraborty, S. Formulation and evaluation of solid lipid nanoparticles of a water soluble drug: zidovudine. Chem. Pharm. Bull., 2010, 58, 650-655.
    • (2010) Chem. Pharm. Bull , vol.58 , pp. 650-655
    • Singh, S.1    Dobhal, A.K.2    Jain, A.3    Pandit, J.K.4    Chakraborty, S.5
  • 21
    • 79959679559 scopus 로고    scopus 로고
    • Formulation and Evaluation of Solid Lipid Nanoparticles of Water Soluble Drug: Isoniazid
    • Nair, R.; Priya, K.V.; Kumar; Badivaddin, T.M.; M, S. Formulation and Evaluation of Solid Lipid Nanoparticles of Water Soluble Drug: Isoniazid. J. Pharm. Sci. Res., 2011, 3, 1256-1264.
    • (2011) J. Pharm. Sci. Res , vol.3 , pp. 1256-1264
    • Nair, R.1    Priya, K.V.2    Kumar3    Badivaddin, T.M.4
  • 23
    • 43249131662 scopus 로고    scopus 로고
    • TBAlliance. Isoniazid
    • TBAlliance. Isoniazid. Tuberculosis, 2008, 88, 112-116.
    • (2008) Tuberculosis , vol.88 , pp. 112-116
  • 24
    • 0030918970 scopus 로고    scopus 로고
    • Therapeutic efficacies of isoniazid and rifampin encapsulated in lung-specific stealth liposomes against Mycobacterium tuberculosis Infection Induced in Mice
    • Deol, P.; Khuller, G.K.; Joshi, K. Therapeutic efficacies of isoniazid and rifampin encapsulated in lung-specific stealth liposomes against Mycobacterium tuberculosis Infection Induced in Mice. Antimicrob. Agents Chemother., 1997, 41, 1211-1214.
    • (1997) Antimicrob. Agents Chemother , vol.41 , pp. 1211-1214
    • Deol, P.1    Khuller, G.K.2    Joshi, K.3
  • 25
    • 49049084290 scopus 로고    scopus 로고
    • Alginate nanoparticles as antituberculosis drug carriers: Formulation, development, pharmacokinetics and therapeutic potential
    • Ahmad, Z.; Pandey, R.; Sharma, S.; Khuller, G.K. Alginate nanoparticles as antituberculosis drug carriers: formulation, development, pharmacokinetics and therapeutic potential. Indian J. Chest. Dis. Allied. Sci., 2006, 48, 171-176.
    • (2006) Indian J. Chest. Dis. Allied. Sci , vol.48 , pp. 171-176
    • Ahmad, Z.1    Pandey, R.2    Sharma, S.3    Khuller, G.K.4
  • 27
    • 40649120076 scopus 로고    scopus 로고
    • Polymerassociated liposomes as a novel delivery system for cyclodextrin-bound drugs
    • Lim, H.J.; Cho, E.C.; Shim, J.; Kim, D-H.; An, E.J.; Kim, J. Polymerassociated liposomes as a novel delivery system for cyclodextrin-bound drugs. J. Colloid Interface Sci., 2008, 320, 460-468.
    • (2008) J. Colloid Interface Sci , vol.320 , pp. 460-468
    • Lim, H.J.1    Cho, E.C.2    Shim, J.3    Kim, D.-H.4    An, E.J.5    Kim, J.6
  • 28
    • 27744539034 scopus 로고    scopus 로고
    • Oral solid lipid nanoparticle-based antitubercular chemotherapy
    • Pandey, R.; Sharma, S.; Khuller, G.K. Oral solid lipid nanoparticle-based antitubercular chemotherapy. Tuberculosis, 2005, 85, 415-420.
    • (2005) Tuberculosis , vol.85 , pp. 415-420
    • Pandey, R.1    Sharma, S.2    Khuller, G.K.3
  • 29
    • 0031929391 scopus 로고    scopus 로고
    • Drug retention and stability of solid lipid nanoparticles containing azidothymidine palmitate after autoclaving, storage and lyopholization
    • Heiati, H.; Tawashi, R.; Phillips, N.C. Drug retention and stability of solid lipid nanoparticles containing azidothymidine palmitate after autoclaving, storage and lyopholization. J. Microencapsul., 1998, 15, 173-184.
    • (1998) J. Microencapsul , vol.15 , pp. 173-184
    • Heiati, H.1    Tawashi, R.2    Phillips, N.C.3
  • 30
    • 0029876015 scopus 로고    scopus 로고
    • Crystallization tendency and polymorphic transitions in triglyceride nanoparticles
    • Bunjes, H.; Westesen, K.; Koch, M.H.J. Crystallization tendency and polymorphic transitions in triglyceride nanoparticles. Int. J. Pharm., 1996, 129, 159-173.
    • (1996) Int. J. Pharm , vol.129 , pp. 159-173
    • Bunjes, H.1    Westesen, K.2    Koch, M.H.J.3
  • 31
    • 0027081624 scopus 로고
    • Behaviour of timolol incorporated in lipospheres in the presence of a series of phosphate esters
    • Cavalli, R.; Gasco, M.R.; Morel, S. Behaviour of timolol incorporated in lipospheres in the presence of a series of phosphate esters. STP Pharma Sci., 1992, 2, 514-518.
    • (1992) STP Pharma Sci , vol.2 , pp. 514-518
    • Cavalli, R.1    Gasco, M.R.2    Morel, S.3
  • 32
    • 0035946615 scopus 로고    scopus 로고
    • Solid Lipid Nanoparticles Production, Characterization and applications
    • Mehnert, W.; Mader, K. Solid Lipid Nanoparticles Production, Characterization and applications. Adv. Drug Deliv. Rev., 2001, 47, 165-196.
    • (2001) Adv. Drug Deliv. Rev , vol.47 , pp. 165-196
    • Mehnert, W.1    Mader, K.2
  • 33
    • 0001469131 scopus 로고
    • Submicron-sized parenteral carrier systems based on solid lipids
    • Siekmann, B.; Westesen, K. Submicron-sized parenteral carrier systems based on solid lipids. Pharm. Pharmacol. Lett., 1992, 1, 123-126.
    • (1992) Pharm. Pharmacol. Lett , vol.1 , pp. 123-126
    • Siekmann, B.1    Westesen, K.2
  • 38
    • 84878632467 scopus 로고
    • US Patent 5250236
    • Gasco, M.R. In US Patent 5250236, 1993.
    • (1993)
    • Gasco, M.R.1
  • 39
    • 84878653523 scopus 로고    scopus 로고
    • USP30NF25
    • USP30NF25. Solubility. 2007, 1689.
    • (2007) Solubility
  • 40
    • 84878643748 scopus 로고    scopus 로고
    • Merck & Co., Inc.: White House Station, NJ, USA
    • Isoniazid, Merck & Co., Inc.: White House Station, NJ, USA 2002.
    • (2002) Isoniazid
  • 42
    • 84878666215 scopus 로고    scopus 로고
    • USEPA
    • USEPA, 1996.
    • (1996)
  • 43
    • 1542611547 scopus 로고    scopus 로고
    • Preparation, characterization and in vitro release kinetics of clozapine solid lipid nanoparticles
    • Venkateswarlu, V.; Manjunath, K. Preparation, characterization and in vitro release kinetics of clozapine solid lipid nanoparticles. J. Control Release, 2004, 95, 627-638.
    • (2004) J. Control Release , vol.95 , pp. 627-638
    • Venkateswarlu, V.1    Manjunath, K.2
  • 44
    • 27744443754 scopus 로고    scopus 로고
    • Etoposide-loaded nanoparticles made from glyceride lipids: Formulation, characterization, in vitro drug release, and stability evaluation
    • Reddy, H.; Murthy, R.S.R. Etoposide-loaded nanoparticles made from glyceride lipids: formulation, characterization, in vitro drug release, and stability evaluation. AAPS Pharm. Sci. Tech., 2005, 6, E158-166.
    • (2005) AAPS Pharm. Sci. Tech , vol.6
    • Reddy, H.1    Murthy, R.S.R.2
  • 45
    • 77951710606 scopus 로고    scopus 로고
    • Formulation and evaluation of solid lipid nanoparticles of a water soluble drug: Zidovudine
    • Singh, S.; Dobhal, A.K.; Jain, A.; Pandit, P.K.; Chakarborty, S. Formulation and evaluation of solid lipid nanoparticles of a water soluble drug: Zidovudine. Chem. Pharm. Bull., 2010, 58, 650-655.
    • (2010) Chem. Pharm. Bull , vol.58 , pp. 650-655
    • Singh, S.1    Dobhal, A.K.2    Jain, A.3    Pandit, P.K.4    Chakarborty, S.5
  • 47
    • 67349203156 scopus 로고    scopus 로고
    • Effect of lipid core material on characteristics of solid lipid nanoparticles designed for oral lymphatic delivery
    • Paliwal, R.; Rai, S.; Vaidya, B.; Khatri, K.; Goyal, A.K.; Mishra, N.; Mehta, A.; Vyas, S.P. Effect of lipid core material on characteristics of solid lipid nanoparticles designed for oral lymphatic delivery. Nanomedicine, 2009, 5, 184-191.
    • (2009) Nanomedicine , vol.5 , pp. 184-191
    • Paliwal, R.1    Rai, S.2    Vaidya, B.3    Khatri, K.4    Goyal, A.K.5    Mishra, N.6    Mehta, A.7    Vyas, S.P.8


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.