메뉴 건너뛰기




Volumn 14, Issue 7, 2013, Pages 564-565

A selective ALK inhibitor in ALK-rearranged patients

Author keywords

[No Author keywords available]

Indexed keywords

CH 5424802; CRIZOTINIB; DOCETAXEL; PEMETREXED; PROTEIN TYROSINE KINASE INHIBITOR; UNCLASSIFIED DRUG;

EID: 84878348650     PISSN: 14702045     EISSN: 14745488     Source Type: Journal    
DOI: 10.1016/S1470-2045(13)70170-0     Document Type: Letter
Times cited : (7)

References (10)
  • 1
    • 0028198206 scopus 로고
    • Fusion of a kinase gene, ALK, to a nucleolar protein gene, NPM, in non-Hodgkin's lymphoma
    • Morris SW, Kirstein MN, Valentine MB, et al. Fusion of a kinase gene, ALK, to a nucleolar protein gene, NPM, in non-Hodgkin's lymphoma. Science 1994, 263:1281-1284.
    • (1994) Science , vol.263 , pp. 1281-1284
    • Morris, S.W.1    Kirstein, M.N.2    Valentine, M.B.3
  • 2
    • 34547638047 scopus 로고    scopus 로고
    • Identification of the transforming EML4-ALK fusion gene in non-small-cell lung cancer
    • Soda M, Choi YL, Enomoto M, et al. Identification of the transforming EML4-ALK fusion gene in non-small-cell lung cancer. Nature 2007, 448:561-566.
    • (2007) Nature , vol.448 , pp. 561-566
    • Soda, M.1    Choi, Y.L.2    Enomoto, M.3
  • 3
    • 84866934606 scopus 로고    scopus 로고
    • Activity and safety of crizotinib in patients with ALK-positive non-small-cell lung cancer: updated results from a phase 1 study
    • Camidge DR, Bang YJ, Kwak EL, et al. Activity and safety of crizotinib in patients with ALK-positive non-small-cell lung cancer: updated results from a phase 1 study. Lancet Oncol 2012, 13:1011-1019.
    • (2012) Lancet Oncol , vol.13 , pp. 1011-1019
    • Camidge, D.R.1    Bang, Y.J.2    Kwak, E.L.3
  • 4
    • 84872569905 scopus 로고    scopus 로고
    • Phase III study of crizotinib versus pemetrexed or docetaxel chemotherapy in patients with advanced ALK-positive non-small cell lung cancer (NSCLC) (PROFILE 1007)
    • Abstr LBA1_PR.
    • Shaw AT, Kim DW, Nakagawa K, Seto T Phase III study of crizotinib versus pemetrexed or docetaxel chemotherapy in patients with advanced ALK-positive non-small cell lung cancer (NSCLC) (PROFILE 1007). Ann Oncol 2012, Abstr LBA1_PR.
    • (2012) Ann Oncol
    • Shaw, A.T.1    Kim, D.W.2    Nakagawa, K.3    Seto, T.4
  • 5
    • 84875936053 scopus 로고    scopus 로고
    • ALK in lung cancer: past, present, and future
    • Shaw AT, Engelman JA ALK in lung cancer: past, present, and future. J Clin Oncol 2013, 31:1105-1111.
    • (2013) J Clin Oncol , vol.31 , pp. 1105-1111
    • Shaw, A.T.1    Engelman, J.A.2
  • 6
    • 84856990335 scopus 로고    scopus 로고
    • Mechanisms of resistance to crizotinib in patients with ALK gene rearranged non-small cell lung cancer
    • Doebele RC, Pilling AB, Aisner DL, et al. Mechanisms of resistance to crizotinib in patients with ALK gene rearranged non-small cell lung cancer. Clin Cancer Res 2012, 18:1472-1482.
    • (2012) Clin Cancer Res , vol.18 , pp. 1472-1482
    • Doebele, R.C.1    Pilling, A.B.2    Aisner, D.L.3
  • 7
    • 84856233310 scopus 로고    scopus 로고
    • Design and synthesis of a highly selective, orally active and potent anaplastic lymphoma kinase inhibitor (CH5424802)
    • Kinoshita K, Asoh K, Furuichi N, et al. Design and synthesis of a highly selective, orally active and potent anaplastic lymphoma kinase inhibitor (CH5424802). Bioorg Med Chem 2012, 20:1271-1280.
    • (2012) Bioorg Med Chem , vol.20 , pp. 1271-1280
    • Kinoshita, K.1    Asoh, K.2    Furuichi, N.3
  • 8
    • 79955964568 scopus 로고    scopus 로고
    • CH5424802, a selective ALK inhibitor capable of blocking the resistant gatekeeper mutant
    • Sakamoto H, Tsukaguchi T, Hiroshima S, et al. CH5424802, a selective ALK inhibitor capable of blocking the resistant gatekeeper mutant. Cancer cell 2011, 19:679-690.
    • (2011) Cancer cell , vol.19 , pp. 679-690
    • Sakamoto, H.1    Tsukaguchi, T.2    Hiroshima, S.3
  • 9
    • 84878347085 scopus 로고    scopus 로고
    • CH5424802 (RO5424802) for patients with ALK-rearranged advanced non-small-cell lung cancer (AF-001JP study): a single-arm, open-label, phase 1-2 study
    • published online April 30.
    • Seto T, Kiura K, Nishio M, Nakagawa K CH5424802 (RO5424802) for patients with ALK-rearranged advanced non-small-cell lung cancer (AF-001JP study): a single-arm, open-label, phase 1-2 study. Lancet Oncol 2013, published online April 30. http://dx.doi.org/10.1016/S1470-2045(13)70142-6.
    • (2013) Lancet Oncol
    • Seto, T.1    Kiura, K.2    Nishio, M.3    Nakagawa, K.4
  • 10
    • 84877679409 scopus 로고    scopus 로고
    • Targeted inhibition of the molecular chaperone Hsp90 overcomes ALK inhibitor resistance in non-small cell lung cancer
    • published online March 26.
    • Sang J, Acquaviva J, Friedland JC, et al. Targeted inhibition of the molecular chaperone Hsp90 overcomes ALK inhibitor resistance in non-small cell lung cancer. Cancer Discov 2013, published online March 26. 10.1158/2159-8290.cd-12-0440.
    • (2013) Cancer Discov
    • Sang, J.1    Acquaviva, J.2    Friedland, J.C.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.