Isothermal titration calorimetry with micelles: Thermodynamics of inhibitor binding to carnitine palmitoyltransferase 2 membrane protein

FEBS Open Bio

Volumn 3, Issue , 2013, Pages 204-211

  Perspicace, Samantha ^a   Rufer, Arne C ^b   Thoma, Ralf ^b   Mueller, Francis ^b   Hennig, Michael ^b   Ceccarelli, Simona ^b   Schulz Gasch, Tanja ^b   Seelig, Joachim ^a  

^a UNIVERSITY OF BASEL   (Switzerland)

^b F HOFFMANN LA ROCHE LTD   (Switzerland)

Author keywords

OG (n octyl D glucopyranoside); CMC (critical micellar concentration); ITC (isothermal titration calorimetry); RCPT 2 (rat carnitine palmitoyltransferase)

Indexed keywords

CARNITINE PALMITOYLTRANSFERASE; CARNITINE PALMITOYLTRANSFERASE 2; COENZYME A; OCTYL GLUCOSIDE; TEGLICAR; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; BINDING SITE; CRITICAL MICELLE CONCENTRATION; CRYSTAL STRUCTURE; DISSOCIATION CONSTANT; ENTHALPY; IC 50; ISOTHERMAL TITRATION CALORIMETRY; LIGAND BINDING; MICELLE; MOLECULAR DOCKING; MOLECULAR INTERACTION; MOLECULAR MODEL; MOLECULAR WEIGHT; NONHUMAN; PRIORITY JOURNAL; PROTEIN STABILITY; PROTON TRANSPORT; RAT; SOLUBILIZATION; STOICHIOMETRY; THERMODYNAMICS; X RAY CRYSTALLOGRAPHY;

EID: 84877121934     PISSN: 22115463     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.fob.2013.04.003     Document Type: Article

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