Synthesis and bioactivities of some new 1H-pyrazole derivatives containing an aryl sulfonate moiety

Chinese Chemical Letters

Volumn 24, Issue 4, 2013, Pages 325-328

  Kendre, Babasaheb V ^a   Landge, Mahadev G ^a   Jadhav, Wamanrao N ^a   Bhusare, Sudhakar R ^a  

^a DNYANOPASAK COLLEGE   (India)

Author keywords

Anti inflammatory activity; COX 2 inhibitors; Enaminone; p Toluene sulfonyl chloride; Pyrazole

Indexed keywords

EID: 84876688002     PISSN: 10018417     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.cclet.2013.02.016     Document Type: Article

References (21)

1. C.E. Dugowson, and P. Gnanashanmugam Nonsteroidal anti-inflammatory drugs Phys. Med. Rehabil. Clin. N. Am. 17 2006 347 354
2. J.R. Vane, and R.M. Botting The mechanism of action of aspirin Thromb. Res. 110 2003 255 258
3. S. Hernandez-Diaz, and L.A.G. Rodriguez Association between nonsteroidal anti-inflammatory drugs and upper gastrointestinal tract bleeding/perforation Arch. Intern. Med. 160 2000 2093 2099
4. F. Krotz, T.M. Schiele, and V. Klauss Selective COX-2 inhibitors and risk of myocardial infarction J. Vasc. Res. 42 2005 312 324
5. S.M. El-Moghazy, F.F. Barsoum, H.M. Abdel-Rahman, and A.A. Marzouk Synthesis and anti-inflammatory activity of some pyrazole derivatives Med. Chem. Res. 21 2012 1722 1733
6. S.R. Shih, T.Y. Chu, and G.R. Reddy Pyrazole compound BPR1P0034 with potent and selective anti-influenza virus activity J. Biomed. Sci. 17 2010 13
7. H. Naito, S. Ohsuki, M. Sugimori, and R. Atsumi Synthesis and antitumor activity of novel pyrimidinyl pyrazole derivatives. II. Optimization of the phenylpiperazine moiety of 1-[5-methyl-1-(2-pyrimidinyl)-4-pyrazolyl]-3- phenylpiperazinyl-1-trans-propenes Chem. Pharm. Bull. 50 2002 453 462
8. M. Abdel-Aziz, G.A. Abuo-Rahma, and A.A. Hassan Synthesis of novel pyrazole derivatives and evaluation of their antidepressant and anticonvulsant activities Eur. J. Med. Chem. 44 2009 3480 3487
9. P.B.R. Kumar, S. Subramaniyan, K. Yamini, and R. Suthakaran Synthesis of some novel 1-H pyrazoles derivatives and their antibacterial activity studies Russ. J. Chem. 4 2011 400 404
10. A. Balbi, M. Anzaldi, and C. Macciò Synthesis and biological evaluation of novel pyrazole derivatives with anticancer activity Eur. J. Med. Chem. 46 2011 5293 5309
11. H.A. Saad, N.A. Osman, and A.H. Moustafa Synthesis and analgesic activity of some new pyrazoles and triazoles bearing a 6,8-dibromo-2-methylquinazoline moiety Molecules 16 2011 10187 10201
12. H. Joshi, P. Upadhyay, D. Karia, and A. Baxi Synthesis of some novel imidazolinones as potent anticonvulsant agents Eur. J. Med. Chem. 38 2003 837 840
13. R.N. Mistry, and K.R. Desai Studies on synthesis of some novel heterocyclic azlactone derivatives and imidazolinone derivatives and their antimicrobial activity Eur. J. Chem. 2 2005 42 51
14. N.D. Christensen, C.A. Reed, and T.D. Culp Papillomavirus microbicidal activities of high-molecular-weight cellulose sulfate, dextran sulfate, and polystyrene sulfonate Antimicrob. Agents Chemother. 45 2001 3427 3432
15. S. Rusconi, M. Moonis, and D.P. Merrill Naphthalene sulfonate polymers with CD4-blocking and anti-human immunodeficiency virus type 1 activities Antimicrob. Agents Chemother. 40 1996 234 236
16. M.A. Hanna, M.M. Girges, and M.A. Berghot Sulfonate ester-containing (imidazol-1-yl)-n-substituted benzene sulfonamides of anticipated antineoplastic activity Phosphorus Sulfur Silicon Relat. Elem. 61 1991 239 246
17. L.M. Betts, N.C. Tam, S.M.H. Kabir, R.F. Langler, and I. Crandall Ether aryl sulfonic acid esters with improved antimalarial/anticancer activities Aust. J. Chem. 59 2006 277 282
18. O.M.O. Habib, H.M. Hassan, E.B. Moawad, and A. El-Mekabaty Synthetic approaches and biological evaluation of some new sulfonate ester-containing imidazolone derivatives Am. J. Org. Chem. 2 2012 79 86
19. B.R. Patil, S.R. Bhusare, R.P. Pawar, and Y.B. Vibhute Iodine and iodic acid: an efficient reagent combination for iodination of aryl hydroxy ketones Tetrahedron Lett. 46 2005 7179 7181
20. S.B. Patwari, M.A. Baseer, Y.B. Vibhute, and S.R. Bhusare Pyridinium bromochromate: a new and efficient reagent for bromination of hydroxy aromatics Tetrahedron Lett. 44 2003 4893 4894
21. Indian Pharmacopoeia Microbiological Assays and Tests vol. 2 1996 Publication & Information Directorate India pp. A-100-A-116