Extended release of metoprolol succinate from hpmc reinforced alginate microparticle

Fabad Journal of Pharmaceutical Sciences

Volumn 36, Issue 1, 2011, Pages 1-10

  Parhi, Rabinarayan ^a   Suresh, Padilam ^a  

^a GITAM UNIVERSITY   (India)

Author keywords

Alginate; Burst release; Extended release; Hydroxypropyl methylcellulose; Metoprolol succinate

Indexed keywords

CALCIUM ALGINATE; HYDROXYPROPYLMETHYLCELLULOSE; METOPROLOL SUCCINATE;

AQUEOUS SOLUTION; ARTICLE; DRUG DELIVERY SYSTEM; DRUG RELEASE; IN VITRO STUDY; INFRARED SPECTROSCOPY; MICROENCAPSULATION; PARTICLE SIZE; SCANNING ELECTRON MICROSCOPY; X RAY ANALYSIS; X RAY DIFFRACTION;

EID: 84876239630     PISSN: 13004182     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (30)

1. Krishnaiah, Y.S.R., Karthikeyan, R.S., Satyanarayana, V., A three-layer guar gum matrix tablet for oral controlled delivery of highly soluble metoprolol tartrate, Int J Pharm, 2002, 241: 353-366.
2. Kumaravelrajan, R., Narayanan, N., Suba, V., Bhaskar, K., Simultaneous delivery of Nifedipine and Metoprolol tartarate using sandwiched osmotic pump tablet system, Int J Pharm, 2010, 399: 60-70.
3. Ye, Z-W., Rombout, P., Remon, J.P., Vervaet, C., Mooter, G.V., Correlation between the permeability of metoprolol tartrate through plasticized isolated ethylcellulose/hydroxypropyl methylcellulose films and drug release from reservoir pellets, Eur J Pharm Biopharm, 2007, 67: 485-490.
4. Al-Saidan, S.M., Krishnaiah, Y.S.R., Satyanarayana, V., Bhaskar, P., Karthikeyan, R.S., Pharmacokinetic evaluation of guar gum-based three-layer matrix tablets for oral controlled delivery of highly soluble metoprolol tartrate as a model drug, Eur J Pharm Biopharm,2004, 58: 697-703.
5. Kendall, M.J., Maxwell, S.R., Westergren, S.A., Controlled release metoprolol. Clinical pharmacokinetic and therapeutic implications. Clin Pharmcokinet, 1991, 5: 319-330.
6. Lennard, M.S., Silas, J.H., Freestone, S., Trevethick, J., Defective metabolism of metoprolol in poor hydroxylators of debrisoquine, Br J Clin Pharmacol, 1982, 14: 301-303.
7. Sandberg, A., Ragnarsson, G., Johnson, U.E., Sjogren, J., Design of a new multiple unit controlled release formulation of metoprolol-metoprolol CR, Eur J Clin Pharmacol, 1998, 33: S3-S7.
8. Kendall, M.J., Metoprolol-controlled release, zero order kinetics, J Clin Pharm Ther, 1989, 24: 159-179.
9. Abrahamsson, B., Alpsten, M., Jonsson, U.E., Lundberg, P.J., Sandberg, A., Sundgren, M., Svenheden, A., Tolli, J., Gastro-intestinal transit of a multiple-unit formulation (metoprolol CR/ZOK) and a non-disintegrating tablet with emphasis on colon, Int J Pharm, 1996, 140: 229-235.
10. Eddington, N.D., Marroum, P., Uppoor, R., Hussain, A., Development and internal validation of an in vitro-in vivo correlation for a hydrophilic metoprolol tartrate extended-release tablet formulation, Pharm Res, 1998, 15: 466-473.
11. Ghosh, L.K., Sairam, P., Gupta, B.K., Development and evaluation of an oral controlled release multiple emulsion drug delivery system of a specific beta blocker metoprolol tartrate, Bulletino Chemico Farmaceutico,1996, 135: 468-471.
12. Okabe, K., Yamoguchi, H., Kawai, Y., New iontophoretic transdermal administration of the beta-blocker-metoprolol, J Control Release, 1987, 4: 79-85.
13. Breimer, D.D., Gastrointestinal drug delivery systems, Pharm Tech, 1983, 7: 18-23.
14. Pillay, V., Fassihi, R., A novel approach for constant rate delivery of highly soluble bioactives from a simple monolithic system, J Control Release, 2000, 67: 67-78.
15. Narendra, C., Srinath, M.S., Rao, B.P., Development of three layered buccal compact containing metoprolol tartrate by statistical optimization technique, Int J Pharm, 2005, 304: 102-114.
16. Hasan, A.S., Socha, M., Lamprecht, A., Gazhouani, F., Sapin, A., Hoffman, M., Maincent, P., Ubrich, N., Effect of the microencapsulation of nanoparticles on the reduction of burst release, Int J Pharm, 2007, 344: 53-61.
17. Bazzo, G.C., Lemos-Senna, E., Pires, A.T.N., Poly (3-hydroxybutyrate) /chitosan /ketoprofen or piroxicam composite microparticles: preparation and controlled drug release evaluation, Carbohydrate Polymers, 2009, 77: 839-844.
18. Moebus, K., Siepmann, J., Bodmeier, R., Alginate-poloxamer microparticles for controlled drug delivery to mucosal tissue, Eur J Pharm Biopharm, 2009, 72: 42-53.
19. Nellore, R.V., Rekhi, G.S., Hussain, A.S., Tillman, L.G., Augsburger, L.L., Development of metoprolol tartrate extended-release matrix tablet formulations for regulatory policy consideration, J Control Release, 1998, 50: 247-256.
20. Rekhi, G.S., Nellore, R.V., Hussain, A.S., Tillman, L.G., Malinowski, H.J., Augsburger, L.L., Identification of critical formulation and processing variables for metoprolol tartrate extended-release (ER) matrix tablets, J Control Release, 1999, 59: 327-342.
21. Chan, L.W., Heng, P.W.S., Effects of aldehydes and methods of cross-linking on properties of calcium alginate microspheres prepared by emulsification, Biomaterials, 2002, 23: 1319-1326.
22. Coppi, G., Iannuccelli, V., Alginate/chitosan microparticles for tamoxifen delivery to the lymphatic system, Int J Pharm, 2009, 367: 127-132.
23. Stockwell, A.F., Davis, S.S., Walker, S.E., In vitro evaluation of alginate gel system as sustained release drug delivery system, J Control Release, 1986, 3: 167-175.
24. Jay, S.M., Saltzman, W.M., Controlled delivery of VEGF via modulation of alginate microparticle ionic crosslinking, J Control Release, 2009, 134: 26-34.
25. Siepmann, J., Siepmann, F., Mathematical modeling of drug delivery, Int J Pharm, 2008, 364: 328-343.
26. Morch, Y.A., Donati, I., Strand, B.L., Skjak-Braek, G., Effect of Ca2+, Ba2+, and Sr2+ on alginate microbeads, Biomacromol, 2006, 7: 1471-1480
27. Hurteaux, R., Edwards-Ly, F., Laurent-Maquin, D., Levy, M.-C., Coating alginate microspheres with a serum albumin-alginate membrane: application to the encapsulation of a peptide, Eur J Pharm Sci, 2005, 24: 187-197.
28. Yu, C.-Y., Zhang, X.-C., Zhou, F.-Z., Zhang, X.-Z., Cheng, S.-X., Zhuo, R.-X., Sustained release of antineoplastic drugs from chitosan-reinforced alginate microparticle drug delivery system, Int J Pharm, 2008, 357: 15-21.
29. Ritger, P.L., Peppas, N.A., A simple equation for description of solute release. I. Fickian and non-Fickian release fromnon-swellable devices in the formof slabs, spheres, cylinders or discs, J Control Release, 1987a, 5: 23-36.
30. Ritger, P.L., Peppas, N.A., A simple equation for description of solute release. II. Fickian and anomalous release from swellable devices, J Control Release, 1987b, 5: 37-42.