Inhibitory effects of cytoskeleton disrupting drugs and GDP-locked Rab mutants on bradykinin B2 receptor cycling

Pharmacological Research

Volumn 71, Issue , 2013, Pages 44-52

  Charest Morin, Xavier ^a   Fortin, Sébastien ^b   Lodge, Robert ^c   Roy, Caroline ^a   Gera, Lajos ^d   C Gaudreault, René ^a   Marceau, François ^a  

^a LAVAL UNIVERSITY   (Canada)

^b UNIVERSITÉ DU QUÉBEC À TROIS RIVIÈRES   (Canada)

^c LAVAL UNIVERSITY   (Canada)

^d UNIVERSITY OF COLORADO   (United States)

Author keywords

Actin; Arrestin; Bradykinin; Bradykinin B2 receptors; Microtubules; Rab proteins

Indexed keywords

3,4,5 TRIMETHOXYPHENYL 4 (2 OXOIMIDAZOLIDIN 1 YL)BENZENESULFONATE; ACTIN; BETA ARRESTIN 2; BRADYKININ B2 RECEPTOR; BRADYKININ B2 RECEPTOR AGONIST; CYTOCHALASIN D; FTC B 9972; GREEN FLUORESCENT PROTEIN; IMZ 602; MYC PROTEIN; PACLITAXEL; PROTEIN INHIBITOR; RAB PROTEIN; RAB11 PROTEIN; RAB4 PROTEIN; RAB5 PROTEIN; TUBULIN; UNCLASSIFIED DRUG;

ACTIN FILAMENT; ARTICLE; CELL ASSAY; CELL SURFACE; CONTROLLED STUDY; CYTOFLUOROMETRY; DNA SEQUENCE; DRUG EFFECT; DRUG SELECTIVITY; ENDOCYTOSIS; FLUORESCENCE IMAGING; MICROTUBULE; MOLECULAR PROBE; NUCLEOTIDE SEQUENCE; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN FUNCTION; PROTEIN PROTEIN INTERACTION; PROTEIN SYNTHESIS INHIBITION; PROTEIN TARGETING;

ACTINS; BRADYKININ; CYTOCHALASIN D; CYTOSKELETON; ENDOCYTOSIS; GUANOSINE DIPHOSPHATE; HEK293 CELLS; HUMANS; MUTATION; PROTEIN TRANSPORT; RAB GTP-BINDING PROTEINS; RAB5 GTP-BINDING PROTEINS; RECEPTOR, BRADYKININ B2; TUBULIN MODULATORS;

EID: 84876145234     PISSN: 10436618     EISSN: 10961186     Source Type: Journal    
DOI: 10.1016/j.phrs.2013.02.007     Document Type: Article

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