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Volumn 5, Issue , 2012, Pages 401-408

Skin permeability and pharmacokinetics of diclofenac epolamine administered by dermal patch in Yorkshire-Landrace pigs

Author keywords

NSAIDs; Systemic absorption; Tissue distribution; Topical patch

Indexed keywords

DICLOFENAC; DICLOFENAC EPOLAMINE;

EID: 84874991162     PISSN: 11787090     EISSN: None     Source Type: Journal    
DOI: 10.2147/JPR.S35450     Document Type: Article
Times cited : (9)

References (22)
  • 1
    • 77956809925 scopus 로고    scopus 로고
    • Topical diclofenac epolamine patch 1.3% for treatment of acute pain caused by soft tissue injury
    • McCarberg BH, Argoff CE. Topical diclofenac epolamine patch 1.3% for treatment of acute pain caused by soft tissue injury. Int J Clin Pract. 2010;64(11):1546-1553.
    • (2010) Int J Clin Pract , vol.64 , Issue.11 , pp. 1546-1553
    • McCarberg, B.H.1    Argoff, C.E.2
  • 2
    • 4344581424 scopus 로고    scopus 로고
    • Effect of a topical diclofenac solution for relieving symptoms of primary osteoarthritis of the knee: A randomized controlled trial
    • Bookman AA, Williams KS, Shainhouse JZ. Effect of a topical diclofenac solution for relieving symptoms of primary osteoarthritis of the knee: a randomized controlled trial. CMAJ. 2004;171(4):333-338.
    • (2004) CMAJ , vol.171 , Issue.4 , pp. 333-338
    • Bookman, A.A.1    Williams, K.S.2    Shainhouse, J.Z.3
  • 3
    • 33847626719 scopus 로고    scopus 로고
    • Topical agents for the management of musculoskeletal pain
    • Stanos SP. Topical agents for the management of musculoskeletal pain. J Pain Symptom Manage. 2007;33(3):342-355.
    • (2007) J Pain Symptom Manage , vol.33 , Issue.3 , pp. 342-355
    • Stanos, S.P.1
  • 4
    • 83355178042 scopus 로고    scopus 로고
    • Topical nonsteroidal anti-inflammatory drugs for the treatment of pain due to soft tissue injury: Diclofenac epolamine topical patch
    • Lionberger DR, Brennan MJ. Topical nonsteroidal anti-inflammatory drugs for the treatment of pain due to soft tissue injury: diclofenac epolamine topical patch. J Pain Res. 2010;3:223-233.
    • (2010) J Pain Res , vol.3 , pp. 223-233
    • Lionberger, D.R.1    Brennan, M.J.2
  • 5
    • 57449098716 scopus 로고    scopus 로고
    • Diclofenac epolamine (Flector) patch: Evidence for topical activity
    • Petersen B, Rovati S. Diclofenac epolamine (Flector) patch: evidence for topical activity. Clin Drug Investig. 2009;29(1):1-9.
    • (2009) Clin Drug Investig , vol.29 , Issue.1 , pp. 1-9
    • Petersen, B.1    Rovati, S.2
  • 6
    • 55549148761 scopus 로고    scopus 로고
    • Review of the pharmaceutical properties and clinical effects of the topical NSAID formulation, diclofenac epolamine
    • Rainsford KD, Kean WF, Ehrlich GE. Review of the pharmaceutical properties and clinical effects of the topical NSAID formulation, diclofenac epolamine. Curr Med Res Opin. 2008;24(10):2967-2992.
    • (2008) Curr Med Res Opin , vol.24 , Issue.10 , pp. 2967-2992
    • Rainsford, K.D.1    Kean, W.F.2    Ehrlich, G.E.3
  • 7
    • 0034104082 scopus 로고    scopus 로고
    • Topical diclofenac patch relieves minor sports injury pain: Results of a multicenter controlled clinical trial
    • Galer BS, Rowbotham M, Perander J, Devers A, Friedman E. Topical diclofenac patch relieves minor sports injury pain: results of a multicenter controlled clinical trial. J Pain Symptom Manage. 2000;19(4): 287-294.
    • (2000) J Pain Symptom Manage , vol.19 , Issue.4 , pp. 287-294
    • Galer, B.S.1    Rowbotham, M.2    Perander, J.3    Devers, A.4    Friedman, E.5
  • 9
    • 56749155996 scopus 로고    scopus 로고
    • Topical diclofenac: Clinical effectiveness and current uses in osteoarthritis of the knee and soft tissue injuries
    • Banning M. Topical diclofenac: clinical effectiveness and current uses in osteoarthritis of the knee and soft tissue injuries. Expert Opin Pharmacother. 2008;9(16):2921-2929.
    • (2008) Expert Opin Pharmacother , vol.9 , Issue.16 , pp. 2921-2929
    • Banning, M.1
  • 10
    • 0033623754 scopus 로고    scopus 로고
    • Evaluation of Göttingen minipig skin for transdermal in vitro permeation studies
    • Qvist MH, Hoeck U, Kreilgaard B, Madsen F, Frokjaer S. Evaluation of Göttingen minipig skin for transdermal in vitro permeation studies. Eur J Pharm Sci. 2000;11(1):59-68.
    • (2000) Eur J Pharm Sci , vol.11 , Issue.1 , pp. 59-68
    • Qvist, M.H.1    Hoeck, U.2    Kreilgaard, B.3    Madsen, F.4    Frokjaer, S.5
  • 11
    • 34247843033 scopus 로고    scopus 로고
    • Key elements of bioanalytical method validation for small molecules
    • Bansal S, DeStefano A. Key elements of bioanalytical method validation for small molecules. AAPS J. 2007;9(1):E109-E114.
    • (2007) AAPS J , vol.9 , Issue.1
    • Bansal, S.1    DeStefano, A.2
  • 12
    • 0034469255 scopus 로고    scopus 로고
    • Bioanalytical method validation-a revisit with a decade of progress
    • Shah VP, Midha KK, Findlay JW, et al. Bioanalytical method validation-a revisit with a decade of progress. Pharm Res. 2000;17(12): 1551-1557.
    • (2000) Pharm Res , vol.17 , Issue.12 , pp. 1551-1557
    • Shah, V.P.1    Midha, K.K.2    Findlay, J.W.3
  • 13
    • 34548550429 scopus 로고    scopus 로고
    • Quantitative bioanalytical methods validation and implementation: Best practices forchromatographic and ligand binding assays
    • Viswanathan CT, Bansal S, Booth B, et al. Quantitative bioanalytical methods validation and implementation: best practices forchromatographic and ligand binding assays. Pharm Res. 2007;24(10): 1962-1973.
    • (2007) Pharm Res , vol.24 , Issue.10 , pp. 1962-1973
    • Viswanathan, C.T.1    Bansal, S.2    Booth, B.3
  • 14
    • 0003484310 scopus 로고    scopus 로고
    • Accessed June 5, Food and Drug Administration, US Department of Health and Human Services, FDA, Center for Drug Evaluation and Research; 2001. Available from
    • Food and Drug Administration. Guidance for Industry: Bioanalytical Method Validation. US Department of Health and Human Services, FDA, Center for Drug Evaluation and Research; 2001. Available from: http://www.fda.gov/downloads/Drugs/GuidanceComplianceRegulatory Information/Guidances/UCM070107.pdf. Accessed June 5, 2012.
    • (2012) Guidance for Industry: Bioanalytical Method Validation
  • 16
    • 0028352236 scopus 로고
    • Pharmacokinetics and metabolism of diclofenac sodium in Yucatan miniature pigs
    • Oberle RL, Das H, Wong SL, Chan KK, Sawchuk RJ. Pharmacokinetics and metabolism of diclofenac sodium in Yucatan miniature pigs. Pharm Res. 1994;11(5):698-703.
    • (1994) Pharm Res , vol.11 , Issue.5 , pp. 698-703
    • Oberle, R.L.1    Das, H.2    Wong, S.L.3    Chan, K.K.4    Sawchuk, R.J.5
  • 17
    • 77957220519 scopus 로고    scopus 로고
    • The utility of the minipig as an animal model in regulatory toxicology
    • for Steering Group of the RETHINK Project
    • Bode G, Clausing P, Gervais F, et al; for Steering Group of the RETHINK Project. The utility of the minipig as an animal model in regulatory toxicology. J Pharmacol Toxicol Methods. 2010;62(3):196-220.
    • (2010) J Pharmacol Toxicol Methods , vol.62 , Issue.3 , pp. 196-220
    • Bode, G.1    Clausing, P.2    Gervais, F.3
  • 18
    • 22544441127 scopus 로고    scopus 로고
    • Determination of the transdermal bioavailability of a newly developed diclofenac sodium patch in comparison with a reference preparation
    • Gschwend MH, Martin W, Arnold P, et al. Determination of the transdermal bioavailability of a newly developed diclofenac sodium patch in comparison with a reference preparation. Arzneimittelforschung. 2005;55(7):403-413.
    • (2005) Arzneimittelforschung , vol.55 , Issue.7 , pp. 403-413
    • Gschwend, M.H.1    Martin, W.2    Arnold, P.3
  • 19
    • 0033778512 scopus 로고    scopus 로고
    • Oral versus topical NSAIDs in rheumatic diseases: A comparison
    • Heyneman CA, Lawless-Liday C, Wall GC. Oral versus topical NSAIDs in rheumatic diseases: a comparison. Drugs. 2000;60(3):555-574.
    • (2000) Drugs , vol.60 , Issue.3 , pp. 555-574
    • Heyneman, C.A.1    Lawless-Liday, C.2    Wall, G.C.3
  • 20
    • 0028140550 scopus 로고
    • Skin permeability and local tissue concentrations of nonsteroidal anti-inflammatory drugs after topical application
    • Singh P, Roberts MS. Skin permeability and local tissue concentrations of nonsteroidal anti-inflammatory drugs after topical application. J Pharmacol Exp Ther. 1994;268(1):144-151.
    • (1994) J Pharmacol Exp Ther , vol.268 , Issue.1 , pp. 144-151
    • Singh, P.1    Roberts, M.S.2
  • 22
    • 0027144979 scopus 로고
    • A trial with diclofenac HEP plaster as topical treatment in minor sport injuries
    • Jenoure P, Segesser B, Lühti U, Gremion G. A trial with diclofenac HEP plaster as topical treatment in minor sport injuries. Drugs Exp Clin Res. 1993;19(3):125-131.
    • (1993) Drugs Exp Clin Res , vol.19 , Issue.3 , pp. 125-131
    • Jenoure, P.1    Segesser, B.2    Lühti, U.3    Gremion, G.4


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