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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 5, 2013, Pages 1182-1186

Discovery of novel inhibitors targeting the Mycobacterium tuberculosis O-acetylserine sulfhydrylase (CysK1) using virtual high-throughput screening

(7) Jean Kumar, Variam Ullas a Poyraz, Ömer b Saxena, Shalini a Schnell, Robert b Yogeeswari, Perumal a Schneider, Gunter b Sriram, Dharmarajan a

a BIRLA INSTITUTE OF TECHNOLOGY AND SCIENCE (India)

b KAROLINSKA INSTITUTE (Sweden)

Author keywords

CysK1; O Acetylserine sulfhydrylase; Tuberculosis

Indexed keywords

CYSTEINE SYNTHASE; ENZYME INHIBITOR;

ARTICLE; CRYSTAL STRUCTURE; CYTOTOXICITY TEST; DRUG SYNTHESIS; ENZYME INHIBITION; HIGH THROUGHPUT SCREENING; IC 50; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; STRUCTURE ACTIVITY RELATION; VIRTUAL REALITY;

CYSTEINE SYNTHASE; DRUG DESIGN; ENZYME INHIBITORS; HIGH-THROUGHPUT SCREENING ASSAYS; HUMANS; MICROBIAL SENSITIVITY TESTS; MODELS, MOLECULAR; MYCOBACTERIUM TUBERCULOSIS; STRUCTURE-ACTIVITY RELATIONSHIP;

MYCOBACTERIUM TUBERCULOSIS;

EID: 84873723914 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.01.031 Document Type: Article

Times cited : (33)

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